KR20150058159A - 바클로펜 및 아캄프로세이트 기반 황반 변성 장애의 치료 - Google Patents
바클로펜 및 아캄프로세이트 기반 황반 변성 장애의 치료 Download PDFInfo
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- KR20150058159A KR20150058159A KR1020157004145A KR20157004145A KR20150058159A KR 20150058159 A KR20150058159 A KR 20150058159A KR 1020157004145 A KR1020157004145 A KR 1020157004145A KR 20157004145 A KR20157004145 A KR 20157004145A KR 20150058159 A KR20150058159 A KR 20150058159A
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- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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- A—HUMAN NECESSITIES
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| PCT/EP2013/065209 WO2014013025A1 (en) | 2012-07-18 | 2013-07-18 | Baclofen and acamprosate based therapy of macular degeneration disorders |
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| EP3062782A1 (en) | 2013-10-30 | 2016-09-07 | Pharnext | Compositions, methods and uses for the treatment of diabetes and related conditions by controlling blood glucose level |
| AU2015217796B2 (en) | 2014-02-11 | 2020-04-30 | Pharnext | Combination of baclofen, acamprosate and medium chain triglycerides for the treatment of neurological disorders |
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| WO2005019163A2 (en) | 2003-08-20 | 2005-03-03 | Xenoport, Inc. | Acyloxyalkyl carbamate prodrugs, methods of synthesis and use |
| US20050112210A1 (en) * | 2003-09-12 | 2005-05-26 | Terry Grossman | Eye nutritional supplement |
| EP1716115B1 (en) | 2003-12-30 | 2013-02-27 | XenoPort, Inc. | Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof |
| ES2365574T3 (es) | 2007-01-11 | 2011-10-07 | Xenoport, Inc. | Formas de dosificación oral para liberación continua de un profármaco de r-baclofeno y procedimientos de tratamiento. |
| US9308260B2 (en) * | 2007-07-05 | 2016-04-12 | Inserm (Institut National De La Sante Et De La Recherche Medicale) | Anticonvulsive pharmaceutical compositions |
| US20090082464A1 (en) | 2007-09-07 | 2009-03-26 | Bernd Jandeleit | Externally masked neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use |
| WO2009033054A1 (en) | 2007-09-07 | 2009-03-12 | Xenoport, Inc. | Complex pantoic acid ester neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use |
| WO2009052191A1 (en) | 2007-10-15 | 2009-04-23 | Xenoport, Inc. | Internally masked neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use |
| TW200936123A (en) | 2007-11-06 | 2009-09-01 | Xenoport Inc | Use of prodrugs of GABAb agonists for treating neuropathic and musculoskeletal pain |
| WO2009096985A1 (en) | 2008-02-01 | 2009-08-06 | Xenoport, Inc. | Sustained release particulate oral dosage forms of (r)-baclofen prodrugs and methods of treatment |
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| EP2393490A1 (en) * | 2009-02-04 | 2011-12-14 | INSERM - Institut National de la Santé et de la Recherche Médicale | Taurine or taurine-like substances for the prevention and treatment of a disease associated with retinal ganglion cell degeneration |
| JP2012519212A (ja) * | 2009-03-03 | 2012-08-23 | ゼノポート，インコーポレイティド | Ｒ−バクロフェンプロドラッグの持効性放出経口投与形 |
| US8344028B2 (en) | 2009-04-17 | 2013-01-01 | Xenoport, Inc. | Gamma-amino-butyric acid derivatives as GABAB receptor ligands |
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| AU2013291970B2 (en) | 2017-09-28 |
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| JP6271539B2 (ja) | 2018-01-31 |
| BR112015001090A2 (pt) | 2017-06-27 |
| US20150238452A1 (en) | 2015-08-27 |
| WO2014013025A1 (en) | 2014-01-23 |
| MX364232B (es) | 2019-04-16 |
| EP2874617B1 (en) | 2019-02-27 |
| EP2874617A1 (en) | 2015-05-27 |
| AU2013291970A1 (en) | 2015-02-19 |
| CA2879114A1 (en) | 2014-01-23 |
| EA201500143A1 (ru) | 2015-05-29 |
| ZA201500663B (en) | 2016-10-26 |
| CN104780917A (zh) | 2015-07-15 |
| IN2015DN00820A (cg-RX-API-DMAC10.html) | 2015-06-12 |
| ES2729208T3 (es) | 2019-10-30 |
| HK1209335A1 (en) | 2016-04-01 |
| SG11201500309VA (en) | 2015-02-27 |
| US9545389B2 (en) | 2017-01-17 |
| EA029157B1 (ru) | 2018-02-28 |
| IL236737A0 (en) | 2015-02-26 |
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