KR20140071405A - 광민감성 간질의 예방 또는 치료에 사용하기 위한 1h-퀴나졸린-2,4-디온의 용도 - Google Patents
광민감성 간질의 예방 또는 치료에 사용하기 위한 1h-퀴나졸린-2,4-디온의 용도 Download PDFInfo
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- KR20140071405A KR20140071405A KR1020147008752A KR20147008752A KR20140071405A KR 20140071405 A KR20140071405 A KR 20140071405A KR 1020147008752 A KR1020147008752 A KR 1020147008752A KR 20147008752 A KR20147008752 A KR 20147008752A KR 20140071405 A KR20140071405 A KR 20140071405A
- Authority
- KR
- South Korea
- Prior art keywords
- dihydro
- quinazolin
- dioxo
- methanesulfonamide
- trifluoromethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
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- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
- C07D239/96—Two oxygen atoms
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
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- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| PCT/US2011/050687 WO2013036224A1 (en) | 2011-09-07 | 2011-09-07 | Use of 1h-quinazoline- 2, 4 -diones for use in the prevention or treatment photosensitive epilepsy |
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| KR20140071405A true KR20140071405A (ko) | 2014-06-11 |
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| TW201609719A (zh) * | 2014-05-28 | 2016-03-16 | 美國禮來大藥廠 | 作為ＴＡＲＰ－γ８依賴性ＡＭＰＡ受體拮抗劑之６－經取代－３Ｈ－１，３－苯并噻唑－２－酮化合物 |
| US10973783B2 (en) | 2015-12-30 | 2021-04-13 | Adamas Pharmaceuticals, Inc. | Methods and compositions for the treatment of seizure-related disorders |
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| SE0201943D0 (sv) | 2002-06-20 | 2002-06-20 | Astrazeneca Ab | New use |
| JP2007510645A (ja) | 2003-10-31 | 2007-04-26 | アストラゼネカ アクチボラグ | アルキン類ｉ |
| CN1871001A (zh) | 2003-10-31 | 2006-11-29 | 阿斯利康(瑞典)有限公司 | 炔烃ⅲ |
| CA2549969A1 (en) | 2003-10-31 | 2005-05-19 | Astrazeneca Ab | Alkynes ii |
| CA2555402A1 (en) | 2004-02-12 | 2005-09-01 | Celine Bonnefous | Bipyridyl amides as modulators of metabotropic glutamate receptor-5 |
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| GB0508319D0 (en) | 2005-04-25 | 2005-06-01 | Novartis Ag | Organic compounds |
| BRPI0620066A2 (pt) | 2005-12-20 | 2011-11-01 | Novartis Ag | derivados de ácido nicotìnico como moduladores do receptor de glutamato metabotrópico, processo para preparação dos mesmos, composição farmacêutica e uso dos referidos derivados |
| PH12012500886A1 (en) * | 2009-11-03 | 2012-11-26 | Lupin Ltd | Modified release formulation of lacosamide |
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- 2011-09-07 IN IN1791DEN2014 patent/IN2014DN01791A/en unknown
- 2011-09-07 WO PCT/US2011/050687 patent/WO2013036224A1/en not_active Ceased
- 2011-09-07 JP JP2014529647A patent/JP2014525474A/ja not_active Withdrawn
- 2011-09-07 CN CN201180073318.7A patent/CN103889427A/zh active Pending
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- 2011-09-07 KR KR1020147008752A patent/KR20140071405A/ko not_active Withdrawn
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| BR112014005210A2 (pt) | 2017-03-21 |
| CA2846503A1 (en) | 2013-03-14 |
| AU2011376333A1 (en) | 2014-03-13 |
| WO2013036224A1 (en) | 2013-03-14 |
| EP2753331A1 (en) | 2014-07-16 |
| MX2014002693A (es) | 2014-06-04 |
| CN103889427A (zh) | 2014-06-25 |
| IN2014DN01791A (cg-RX-API-DMAC7.html) | 2015-05-15 |
| JP2014525474A (ja) | 2014-09-29 |
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