KR20110002459A - 치료 화합물로서의 치환된 피페리딘 - Google Patents
치료 화합물로서의 치환된 피페리딘 Download PDFInfo
- Publication number
- KR20110002459A KR20110002459A KR1020107022007A KR20107022007A KR20110002459A KR 20110002459 A KR20110002459 A KR 20110002459A KR 1020107022007 A KR1020107022007 A KR 1020107022007A KR 20107022007 A KR20107022007 A KR 20107022007A KR 20110002459 A KR20110002459 A KR 20110002459A
- Authority
- KR
- South Korea
- Prior art keywords
- methoxy
- straight
- methyl
- acid
- chain
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Tropical Medicine & Parasitology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Virology (AREA)
- Neurology (AREA)
- Molecular Biology (AREA)
- Oncology (AREA)
- Hospice & Palliative Care (AREA)
- Communicable Diseases (AREA)
- AIDS & HIV (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08153929 | 2008-04-02 | ||
| EP08153929.8 | 2008-04-02 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20110002459A true KR20110002459A (ko) | 2011-01-07 |
Family
ID=40627638
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020107022007A KR20110002459A (ko) | 2008-04-02 | 2009-04-01 | 치료 화합물로서의 치환된 피페리딘 |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP2271644A1 (es) |
| JP (1) | JP2011516453A (es) |
| KR (1) | KR20110002459A (es) |
| CN (1) | CN101970431A (es) |
| AU (1) | AU2009232012A1 (es) |
| BR (1) | BRPI0910991A2 (es) |
| CA (1) | CA2719070A1 (es) |
| EA (1) | EA201001517A1 (es) |
| MX (1) | MX2010010876A (es) |
| WO (1) | WO2009121914A1 (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011057160A2 (en) * | 2009-11-06 | 2011-05-12 | The Regents Of The Uiversity Of California | Method to improve the immunogenicity of vaccine antigens by modification of cleavage sites in hiv-1 gp 120 |
| MX2012004377A (es) | 2009-10-14 | 2012-06-01 | Merck Sharp & Dohme | Piperidinas sustituidas que aumentan la actividad de p53 y sus usos. |
| GB201008209D0 (en) * | 2010-05-17 | 2010-06-30 | Senexis Ltd | Compounds |
| WO2013062923A1 (en) | 2011-10-28 | 2013-05-02 | Merck Sharp & Dohme Corp. | MACROCYCLES THAT INCREASE p53 ACTIVITY AND THE USES THEREOF |
| ES2707305T3 (es) | 2012-12-20 | 2019-04-03 | Merck Sharp & Dohme | Imidazopiridinas sustituidas como inhibidores de HDM2 |
| CN105001300A (zh) * | 2014-04-17 | 2015-10-28 | 复旦大学 | 组织蛋白酶d抑制剂及其制备方法、药物组合物和应用 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1816122A3 (en) * | 2006-01-19 | 2007-09-19 | Speedel Experimenta AG | 3,4,5-substituted piperidines as therapeutic compounds |
| EP1911758A1 (en) * | 2006-10-04 | 2008-04-16 | Speedel Experimenta AG | Phenyl piperidine derivatives for use as renin inhibitors |
| EP1908761A1 (en) * | 2006-10-04 | 2008-04-09 | Speedel Experimenta AG | Organic compounds |
-
2009
- 2009-04-01 WO PCT/EP2009/053898 patent/WO2009121914A1/en active Application Filing
- 2009-04-01 MX MX2010010876A patent/MX2010010876A/es not_active Application Discontinuation
- 2009-04-01 BR BRPI0910991A patent/BRPI0910991A2/pt not_active Application Discontinuation
- 2009-04-01 CA CA2719070A patent/CA2719070A1/en not_active Abandoned
- 2009-04-01 AU AU2009232012A patent/AU2009232012A1/en not_active Abandoned
- 2009-04-01 CN CN2009801083136A patent/CN101970431A/zh active Pending
- 2009-04-01 EA EA201001517A patent/EA201001517A1/ru unknown
- 2009-04-01 JP JP2011502382A patent/JP2011516453A/ja active Pending
- 2009-04-01 KR KR1020107022007A patent/KR20110002459A/ko not_active Application Discontinuation
- 2009-04-01 EP EP09728288A patent/EP2271644A1/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009121914A1 (en) | 2009-10-08 |
| CN101970431A (zh) | 2011-02-09 |
| AU2009232012A1 (en) | 2009-10-08 |
| CA2719070A1 (en) | 2009-10-08 |
| MX2010010876A (es) | 2010-10-26 |
| JP2011516453A (ja) | 2011-05-26 |
| EA201001517A1 (ru) | 2011-04-29 |
| EP2271644A1 (en) | 2011-01-12 |
| BRPI0910991A2 (pt) | 2016-01-19 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US20070167433A1 (en) | 3,4,5-Substituted piperidines as therapeutic compounds | |
| US8153658B2 (en) | Piperidine derivative or salt thereof | |
| JP5872552B2 (ja) | 化学化合物 | |
| US20070066582A1 (en) | Diaminoalcohols as therapeutic compounds | |
| KR20110002459A (ko) | 치료 화합물로서의 치환된 피페리딘 | |
| JP6609306B2 (ja) | ６，７−ジヒドロピラゾロ［１，５−ａ］ピラジン−４（５Ｈ）−オン化合物およびＭＧＬＵＲ２受容体の負のアロステリック調節因子としてのその使用 | |
| US20070021413A1 (en) | Diamino alcohols as therapeutic compounds | |
| PT2841437T (pt) | Derivados de imidazotiadiazol e imidazopirazina como inibidores de recetor 4 ativado por protease (par4) para o tratamento de agregação plaquetária | |
| JP2017533253A (ja) | アルツハイマー病を治療するための、ｂａｃｅ１阻害剤としての２−アミノ−３，５−ジフルオロ−３，６−ジメチル−６−フェニル−３，４，５，６−テトラヒドロピリジン | |
| TW200302726A (en) | Nitrogen-containing bicyclic compound and medicament containing same as active ingredient | |
| TW201100385A (en) | Substituted isoquinoline derivative | |
| US20220340546A1 (en) | Inhibitors of sarm1 | |
| CA3123215A1 (en) | Inhibitors of sarm1 in combination with neuroprotective agents | |
| EP1958666A1 (en) | Heterocyclic-substituted alkanamides as therapeutic compounds | |
| EP4200293A1 (en) | Inhibitors of sarm1 | |
| US20070021400A1 (en) | Amino alcohols as therapeutic compounds | |
| WO2009106599A2 (en) | Substituted piperidines as therapeutic compounds | |
| ES2519572T3 (es) | Moduladores del receptor de tipo toll y usos de los mismos | |
| TW201111375A (en) | N-substituted cyclic amino derivative | |
| EP1867329A2 (en) | 5-Amino-4-hydroxy-2-isopropyl-7-[4-methoxy-3-(3-methoxypropoxy)benzyl]-8-methylnonanamides as therapeutic compounds | |
| JP2018529647A (ja) | ２−アミノ−３，５，５−トリフルオロ−３，４，５，６−テトラヒドロピリジンの投与を含む併用治療 | |
| US20070021399A1 (en) | Amido-amino alcohols as therapeutic compounds | |
| EP1987834A2 (en) | Substituted piperidines as therapeutic compounds | |
| US20070066604A1 (en) | Diaminoalcohols as therapeutic compounds | |
| EP4259619A1 (en) | Benzopyrazole inhibitors of sarm1 |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| WITN | Withdrawal due to no request for examination |