EA201001517A1 - Замещенные пиперидины в качестве терапевтических соединений - Google Patents
Замещенные пиперидины в качестве терапевтических соединенийInfo
- Publication number
- EA201001517A1 EA201001517A1 EA201001517A EA201001517A EA201001517A1 EA 201001517 A1 EA201001517 A1 EA 201001517A1 EA 201001517 A EA201001517 A EA 201001517A EA 201001517 A EA201001517 A EA 201001517A EA 201001517 A1 EA201001517 A1 EA 201001517A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- therapeutic compounds
- substituted piperidines
- compounds
- piperidines
- substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
Описываются соединения общей формулы (I)и их фармацевтически приемлемые соли, в которых Rимеет определения, подробно проиллюстрированные в описании, в качестве ингибиторов β-секретазы, катепсина D, плазмепсина II и/или протеазы ВИЧ.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP08153929 | 2008-04-02 | ||
PCT/EP2009/053898 WO2009121914A1 (en) | 2008-04-02 | 2009-04-01 | Substituted piperidines as therapeutic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201001517A1 true EA201001517A1 (ru) | 2011-04-29 |
Family
ID=40627638
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201001517A EA201001517A1 (ru) | 2008-04-02 | 2009-04-01 | Замещенные пиперидины в качестве терапевтических соединений |
Country Status (10)
Country | Link |
---|---|
EP (1) | EP2271644A1 (ru) |
JP (1) | JP2011516453A (ru) |
KR (1) | KR20110002459A (ru) |
CN (1) | CN101970431A (ru) |
AU (1) | AU2009232012A1 (ru) |
BR (1) | BRPI0910991A2 (ru) |
CA (1) | CA2719070A1 (ru) |
EA (1) | EA201001517A1 (ru) |
MX (1) | MX2010010876A (ru) |
WO (1) | WO2009121914A1 (ru) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2011057160A2 (en) * | 2009-11-06 | 2011-05-12 | The Regents Of The Uiversity Of California | Method to improve the immunogenicity of vaccine antigens by modification of cleavage sites in hiv-1 gp 120 |
BR112012008849A2 (pt) | 2009-10-14 | 2015-09-22 | Schering Corp | composto, composição farmacêutica, e, uso de um composto |
GB201008209D0 (en) * | 2010-05-17 | 2010-06-30 | Senexis Ltd | Compounds |
EP2771008A4 (en) | 2011-10-28 | 2015-04-08 | Merck Sharp & Dohme | MACROCYCLES INCREASING P53 ACTIVITY AND USES THEREOF |
BR112015013611A2 (pt) | 2012-12-20 | 2017-11-14 | Merck Sharp & Dohme | composto, e, composição farmacêutica |
CN105001300A (zh) * | 2014-04-17 | 2015-10-28 | 复旦大学 | 组织蛋白酶d抑制剂及其制备方法、药物组合物和应用 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1816122A3 (en) * | 2006-01-19 | 2007-09-19 | Speedel Experimenta AG | 3,4,5-substituted piperidines as therapeutic compounds |
EP1908761A1 (en) * | 2006-10-04 | 2008-04-09 | Speedel Experimenta AG | Organic compounds |
EP1911758A1 (en) * | 2006-10-04 | 2008-04-16 | Speedel Experimenta AG | Phenyl piperidine derivatives for use as renin inhibitors |
-
2009
- 2009-04-01 EA EA201001517A patent/EA201001517A1/ru unknown
- 2009-04-01 AU AU2009232012A patent/AU2009232012A1/en not_active Abandoned
- 2009-04-01 KR KR1020107022007A patent/KR20110002459A/ko not_active Application Discontinuation
- 2009-04-01 EP EP09728288A patent/EP2271644A1/en not_active Withdrawn
- 2009-04-01 BR BRPI0910991A patent/BRPI0910991A2/pt not_active Application Discontinuation
- 2009-04-01 CN CN2009801083136A patent/CN101970431A/zh active Pending
- 2009-04-01 CA CA2719070A patent/CA2719070A1/en not_active Abandoned
- 2009-04-01 JP JP2011502382A patent/JP2011516453A/ja active Pending
- 2009-04-01 WO PCT/EP2009/053898 patent/WO2009121914A1/en active Application Filing
- 2009-04-01 MX MX2010010876A patent/MX2010010876A/es not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
MX2010010876A (es) | 2010-10-26 |
CN101970431A (zh) | 2011-02-09 |
WO2009121914A1 (en) | 2009-10-08 |
EP2271644A1 (en) | 2011-01-12 |
KR20110002459A (ko) | 2011-01-07 |
AU2009232012A1 (en) | 2009-10-08 |
BRPI0910991A2 (pt) | 2016-01-19 |
JP2011516453A (ja) | 2011-05-26 |
CA2719070A1 (en) | 2009-10-08 |
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