KR20100020479A - 바이사이클로설포닐 산 (ｂｃｓａ) 화합물 및 치료제로서의 이의 용도 - Google Patents
바이사이클로설포닐 산 (ｂｃｓａ) 화합물 및 치료제로서의 이의 용도 Download PDFInfo
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- KR20100020479A KR20100020479A KR1020097026376A KR20097026376A KR20100020479A KR 20100020479 A KR20100020479 A KR 20100020479A KR 1020097026376 A KR1020097026376 A KR 1020097026376A KR 20097026376 A KR20097026376 A KR 20097026376A KR 20100020479 A KR20100020479 A KR 20100020479A
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Classifications
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- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
- C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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Applications Claiming Priority (2)
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| US92451807P | 2007-05-18 | 2007-05-18 | |
| US60/924,518 | 2007-05-18 |
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| KR20100020479A true KR20100020479A (ko) | 2010-02-22 |
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| US (1) | US20100311741A1 (https=) |
| EP (1) | EP2155703A1 (https=) |
| JP (1) | JP2010527344A (https=) |
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| EP2406248B1 (en) * | 2009-03-11 | 2013-12-25 | Msd K.K. | Novel isoindolin-1-one derivative |
| GB2475359A (en) * | 2009-11-11 | 2011-05-18 | Biocopea Ltd | A compound for use in treating a fulminant respiratory disorder |
| DK2597084T3 (en) | 2010-07-08 | 2016-08-15 | Kaken Pharma Co Ltd | N-HYDROXYFORMAMIDE DERIVATIVE AND MEDICINAL CONTAINING SAME |
| US20150125438A1 (en) | 2012-07-20 | 2015-05-07 | Sang Jae Kim | Anti-Inflammatory Peptides and Composition Comprising the Same |
| WO2015091428A1 (en) * | 2013-12-20 | 2015-06-25 | Bayer Pharma Aktiengesellschaft | Glucose transport inhibitors |
| CN110790758A (zh) * | 2018-08-01 | 2020-02-14 | 上海轶诺药业有限公司 | 一类具有免疫调节功能的含n杂环化合物的制备和应用 |
| EP3750878B1 (en) | 2019-06-14 | 2025-05-14 | Vivoryon Therapeutics N.V. | Heteroaromatic inhibitors of astacin proteinases |
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| EP0350163A3 (en) * | 1988-06-09 | 1990-11-22 | Beecham Group Plc | Renin inhibitory peptides |
| CA2006443A1 (en) * | 1988-12-23 | 1990-06-23 | Stephen A. Smith | Compounds |
| AU653279B2 (en) * | 1991-12-30 | 1994-09-22 | Sanofi | Novel 2-saccharinylmethyl heterocyclic carboxylates useful as proteolytic enzyme inhibitors and compositions and method of use thereof |
| WO1999024419A1 (en) * | 1997-11-12 | 1999-05-20 | Darwin Discovery Limited | Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity |
| US6288063B1 (en) * | 1998-05-27 | 2001-09-11 | Bayer Corporation | Substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives as matrix metalloprotease inhibitors |
| US6319912B1 (en) * | 1999-05-04 | 2001-11-20 | American Home Products Corporation | Cyclic regimens using 2,1-benzisothiazoline 2,2-dioxides |
| WO2002081447A1 (en) * | 2001-04-06 | 2002-10-17 | Daewoong Pharmaceutical Co., Ltd. | 3-cyclopentyloxy-4-methoxyphenyl-isothiazolinone derivatives and the use thereof |
| WO2003031431A1 (en) * | 2001-10-09 | 2003-04-17 | Bristol-Myers Squibb Company | Cyclic sulfone derivatives as inhibitors of matrix metalloproteinases and/or tnf-$g(a) converting enzyme (tace) |
| ATE365167T1 (de) * | 2003-07-10 | 2007-07-15 | Neurogen Corp | Aryl-substituierte benzo(d)isothiazol-3-ylamin analoga als capsaicinrezeptormodulatoren |
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Also Published As
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| JP2010527344A (ja) | 2010-08-12 |
| US20100311741A1 (en) | 2010-12-09 |
| RU2472784C2 (ru) | 2013-01-20 |
| MX2009012470A (es) | 2010-02-24 |
| WO2008142376A1 (en) | 2008-11-27 |
| AU2008252628A1 (en) | 2008-11-27 |
| EP2155703A1 (en) | 2010-02-24 |
| BRPI0811651A2 (pt) | 2014-11-11 |
| CA2687415A1 (en) | 2008-11-27 |
| RU2009145296A (ru) | 2011-06-27 |
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