KR20090047499A - 심근 조영법 동안에 환자의 순응성을 증가시키기 위한 방법및 조성물 - Google Patents

심근 조영법 동안에 환자의 순응성을 증가시키기 위한 방법및 조성물 Download PDF

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Publication number
KR20090047499A
KR20090047499A KR1020097004186A KR20097004186A KR20090047499A KR 20090047499 A KR20090047499 A KR 20090047499A KR 1020097004186 A KR1020097004186 A KR 1020097004186A KR 20097004186 A KR20097004186 A KR 20097004186A KR 20090047499 A KR20090047499 A KR 20090047499A
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South Korea
Prior art keywords
caffeine
receptor agonist
administered
legadenoson
alkyl
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Ceased
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KR1020097004186A
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English (en)
Korean (ko)
Inventor
샤오 디 류
브렌트 블랙번
루이즈 벨라디넬리
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씨브이 쎄러퓨틱스, 인코포레이티드
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Publication of KR20090047499A publication Critical patent/KR20090047499A/ko
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
KR1020097004186A 2006-09-01 2007-08-31 심근 조영법 동안에 환자의 순응성을 증가시키기 위한 방법및 조성물 Ceased KR20090047499A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US84184206P 2006-09-01 2006-09-01
US60/841,842 2006-09-01

Publications (1)

Publication Number Publication Date
KR20090047499A true KR20090047499A (ko) 2009-05-12

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KR1020097004186A Ceased KR20090047499A (ko) 2006-09-01 2007-08-31 심근 조영법 동안에 환자의 순응성을 증가시키기 위한 방법및 조성물

Country Status (12)

Country Link
US (1) US20080213165A1 (https=)
EP (1) EP2056834B1 (https=)
JP (1) JP2010502649A (https=)
KR (1) KR20090047499A (https=)
CN (1) CN101511366B (https=)
AU (1) AU2007289037A1 (https=)
BR (1) BRPI0716174A2 (https=)
CA (1) CA2662278C (https=)
IL (1) IL197267A0 (https=)
MX (1) MX2009002299A (https=)
RU (1) RU2459626C2 (https=)
WO (1) WO2008028140A1 (https=)

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US7732595B2 (en) 2006-02-03 2010-06-08 Gilead Palo Alto, Inc. Process for preparing an A2A-adenosine receptor agonist and its polymorphs
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WO2013028612A2 (en) 2011-08-20 2013-02-28 Volcano Corporation Devices, systems, and methods for visually depicting a vessel and evaluating treatment options
US9339348B2 (en) 2011-08-20 2016-05-17 Imperial Colege of Science, Technology and Medicine Devices, systems, and methods for assessing a vessel
WO2013138617A1 (en) 2012-03-16 2013-09-19 Axikin Pharmaceuticals, Inc. 3,5-diaminopyrazole kinase inhibitors
EP3760637A3 (en) * 2013-04-11 2021-04-07 AMRI Italy S.r.l. Stable solid forms of regadenoson
NZ631142A (en) 2013-09-18 2016-03-31 Axikin Pharmaceuticals Inc Pharmaceutically acceptable salts of 3,5-diaminopyrazole kinase inhibitors
TWI703133B (zh) 2014-12-23 2020-09-01 美商艾克斯基製藥公司 3,5-二胺基吡唑激酶抑制劑

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Also Published As

Publication number Publication date
IL197267A0 (en) 2009-12-24
MX2009002299A (es) 2009-03-20
EP2056834B1 (en) 2012-08-29
CA2662278A1 (en) 2008-03-06
JP2010502649A (ja) 2010-01-28
AU2007289037A1 (en) 2008-03-06
BRPI0716174A2 (pt) 2013-09-24
CN101511366B (zh) 2011-12-28
RU2009106862A (ru) 2010-09-10
US20080213165A1 (en) 2008-09-04
CA2662278C (en) 2011-11-22
EP2056834A1 (en) 2009-05-13
RU2459626C2 (ru) 2012-08-27
WO2008028140A1 (en) 2008-03-06
CN101511366A (zh) 2009-08-19

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