KR20080095877A - 아자사이클릴-치환된 아릴디하이드로이소퀴놀리논, 이의 제조 방법 및 약제로서 이의 용도 - Google Patents

아자사이클릴-치환된 아릴디하이드로이소퀴놀리논, 이의 제조 방법 및 약제로서 이의 용도 Download PDF

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KR20080095877A
KR20080095877A KR1020087019922A KR20087019922A KR20080095877A KR 20080095877 A KR20080095877 A KR 20080095877A KR 1020087019922 A KR1020087019922 A KR 1020087019922A KR 20087019922 A KR20087019922 A KR 20087019922A KR 20080095877 A KR20080095877 A KR 20080095877A
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alkyl
alkoxy
ring
compound
hydroxy
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Korean (ko)
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로타르 슈빈크
지그프리드 슈텐겔린
마티아스 고셀
게르하르트 헤슬러
토르슈텐 학크
페트라 레니그
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사노피-아벤티스
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/472—Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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    • A61K31/00—Medicinal preparations containing organic active ingredients
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    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4355—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having oxygen as a ring hetero atom
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings
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  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
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KR1020087019922A 2006-02-15 2007-02-13 아자사이클릴-치환된 아릴디하이드로이소퀴놀리논, 이의 제조 방법 및 약제로서 이의 용도 Withdrawn KR20080095877A (ko)

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DE102006007045 2006-02-15
DE102006007045.3 2006-02-15

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KR20080095877A true KR20080095877A (ko) 2008-10-29

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US (1) US8822495B2 (enExample)
EP (1) EP1987020B1 (enExample)
JP (1) JP5175228B2 (enExample)
KR (1) KR20080095877A (enExample)
CN (1) CN101384583A (enExample)
AR (1) AR059458A1 (enExample)
AU (1) AU2007214709A1 (enExample)
BR (1) BRPI0707872A2 (enExample)
CA (1) CA2636873A1 (enExample)
CR (1) CR10160A (enExample)
EC (1) ECSP088680A (enExample)
IL (1) IL193340A0 (enExample)
MA (1) MA30221B1 (enExample)
NI (1) NI200800217A (enExample)
NZ (1) NZ570503A (enExample)
RU (1) RU2008136898A (enExample)
TN (1) TNSN08326A1 (enExample)
TW (1) TW200800908A (enExample)
UY (1) UY30166A1 (enExample)
WO (1) WO2007093364A1 (enExample)
ZA (1) ZA200805939B (enExample)

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AR083718A1 (es) 2010-05-11 2013-03-20 Sanofi Aventis Fenil cicloalquil pirrolidina (piperidina) espirolactamas y amidas sustituidas, preparacion y uso terapeutico de las mismas
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NZ570503A (en) 2010-07-30
MA30221B1 (fr) 2009-02-02
IL193340A0 (en) 2009-05-04
UY30166A1 (es) 2007-09-28
CR10160A (es) 2008-10-06
AU2007214709A1 (en) 2007-08-23
TW200800908A (en) 2008-01-01
US20090264403A1 (en) 2009-10-22
RU2008136898A (ru) 2010-03-20
EP1987020A1 (en) 2008-11-05
EP1987020B1 (en) 2012-10-03
TNSN08326A1 (en) 2009-12-29
BRPI0707872A2 (pt) 2011-05-10
US8822495B2 (en) 2014-09-02
CA2636873A1 (en) 2007-08-23
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JP5175228B2 (ja) 2013-04-03
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