KR20060032598A - 세로토닌 재흡수 억제제 및 아고멜라틴의 조합 - Google Patents
세로토닌 재흡수 억제제 및 아고멜라틴의 조합 Download PDFInfo
- Publication number
- KR20060032598A KR20060032598A KR1020057024442A KR20057024442A KR20060032598A KR 20060032598 A KR20060032598 A KR 20060032598A KR 1020057024442 A KR1020057024442 A KR 1020057024442A KR 20057024442 A KR20057024442 A KR 20057024442A KR 20060032598 A KR20060032598 A KR 20060032598A
- Authority
- KR
- South Korea
- Prior art keywords
- serotonin reuptake
- reuptake inhibitor
- serotonin
- pharmaceutical composition
- pharmaceutically acceptable
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
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- Hospice & Palliative Care (AREA)
- Addiction (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Child & Adolescent Psychology (AREA)
- Nutrition Science (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| DKPA200301031 | 2003-07-04 | ||
| DKPA200301031 | 2003-07-04 | ||
| US48547903P | 2003-07-07 | 2003-07-07 |
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| KR20060032598A true KR20060032598A (ko) | 2006-04-17 |
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Country Status (17)
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| EP (1) | EP1643985B1 (enExample) |
| JP (1) | JP2007513052A (enExample) |
| KR (1) | KR20060032598A (enExample) |
| CN (1) | CN1852706A (enExample) |
| AR (1) | AR047553A1 (enExample) |
| AT (1) | ATE499096T1 (enExample) |
| AU (1) | AU2004253225A1 (enExample) |
| BR (1) | BRPI0411665A (enExample) |
| CA (1) | CA2530880A1 (enExample) |
| DE (1) | DE602004031527D1 (enExample) |
| DK (1) | DK1643985T3 (enExample) |
| IL (1) | IL172965A0 (enExample) |
| IS (1) | IS8154A (enExample) |
| MX (1) | MXPA06000018A (enExample) |
| NO (1) | NO20060242L (enExample) |
| WO (1) | WO2005002562A1 (enExample) |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
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| FR2884714B1 (fr) * | 2005-04-20 | 2011-05-06 | Servier Lab | Utilisation de l'agomelatine pour l'obtention de medicaments destines au traitement des troubles bipolaires |
| FR2890564B1 (fr) * | 2005-09-09 | 2007-10-19 | Servier Lab | Nouvelle association entre l'agomelatine et un inhibiteur de la recapture de la noradrenaline et les compositions pharmaceutiques qui la contiennent |
| FR2890563B1 (fr) * | 2005-09-09 | 2007-10-19 | Servier Lab | Nouvelle association entre l'agomelatine et un agent thymoregulateur et les compositions pharmaceutiques qui la contiennent |
| FR2899472B1 (fr) | 2006-04-07 | 2008-09-12 | Servier Lab | Utilisation de l'agomelatine pour l'obtention de medicaments destines au traitement du trouble anxiete generalisee |
| WO2008035177A2 (en) * | 2006-09-18 | 2008-03-27 | Copharm | Combination of mt1 and mt2 melatonin receptor agonists and a norepinephrine/dopamine reuptake inhibitor |
| CA2685924A1 (en) * | 2007-05-01 | 2008-11-13 | Concert Pharmaceuticals Inc. | Naphthyl(ethyl)acetamides |
| WO2008141033A1 (en) * | 2007-05-08 | 2008-11-20 | Auspex Pharmaceuticals Inc. | Substituted naphthalenes |
| FR2956031B1 (fr) * | 2010-02-11 | 2012-03-02 | Servier Lab | Utilisation de l'agomelatine pour l'obtention de medicaments destines au traitement du trouble obsessionnel compulsif (toc) |
| EP2629615B1 (en) | 2010-10-22 | 2018-10-10 | Duke University | Slow-release formulations of 5-hydroxytryptophan as an adjunct to pro-serotonergic therapies |
| EP2517700B1 (en) * | 2011-04-28 | 2013-07-17 | Zentiva, k.s. | Pharmaceutically acceptable cocrystals of N-[2-(7-methoxy-1-naphthyl]acetamide and methods of their preparation |
| PH12012000132B1 (en) * | 2011-06-09 | 2014-10-20 | Servier Lab | New co-crystals of agomelatine, a process for their preparation and pharmaceutical compositions containing them |
| WO2013013060A1 (en) * | 2011-07-19 | 2013-01-24 | Lycus, Llc | Agomelatine derivatives |
| EP2551257A1 (en) * | 2011-07-28 | 2013-01-30 | Laboratorios Del. Dr. Esteve, S.A. | Co-crystals of agomelatine with co-crystal-formers |
| WO2014024896A1 (ja) * | 2012-08-08 | 2014-02-13 | 株式会社メドレックス | アゴメラチンを含有する貼付剤組成物 |
| US20250134902A1 (en) * | 2022-02-09 | 2025-05-01 | Univesrity Of North Texas Health Science Center | Drug repurposing for delayed treatment of ischemic stroke |
| CN116570579A (zh) * | 2023-06-13 | 2023-08-11 | 深圳市泛谷药业股份有限公司 | 一种含有阿戈美拉汀和氟伏沙明的药物组合物及其应用 |
Family Cites Families (13)
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| FR2658818B1 (fr) | 1990-02-27 | 1993-12-31 | Adir Cie | Nouveaux derives a structure naphtalenique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| US5470846A (en) * | 1994-01-14 | 1995-11-28 | Sandyk; Reuven | Treatment of neurological and mental disorders |
| CA2134038C (en) | 1994-06-16 | 1997-06-03 | David Taiwai Wong | Potentiation of drug response |
| JP3155008B2 (ja) | 1994-07-26 | 2001-04-09 | ファイザー・インコーポレーテッド | セロトニンアゴニストおよびアンタゴニストとしての４−インドール誘導体 |
| US5597826A (en) | 1994-09-14 | 1997-01-28 | Pfizer Inc. | Compositions containing sertraline and a 5-HT1D receptor agonist or antagonist |
| EP0714663A3 (en) | 1994-11-28 | 1997-01-15 | Lilly Co Eli | Potentiation of drug responses by serotonin 1A receptor antagonists |
| FR2744449B1 (fr) | 1996-02-02 | 1998-04-24 | Pf Medicament | Nouvelles piperazines aromatiques derivees de cycloazanes substitues, ainsi que leur procede de preparation, les compositions pharmaceutiques et leur utilisation comme medicaments |
| SE9703375D0 (sv) | 1997-09-18 | 1997-09-18 | Astra Ab | A new combination |
| GB2336534A (en) * | 1998-04-24 | 1999-10-27 | Alec James Coppen | Anti-depressant - Folic Acid Combination |
| UA77650C2 (en) * | 1999-12-06 | 2007-01-15 | Lundbeck & Co As H | Use of serotonin reuptake inhibitor in combination with deramcyclane |
| YU85303A (sh) * | 2001-05-01 | 2006-05-25 | H. Lundbeck A/S | Upotreba enantiomerno čistog escitaloprama |
| US6617891B2 (en) * | 2001-09-26 | 2003-09-09 | Intel Corporation | Slew rate at buffers by isolating predriver from driver |
| FR2834890B1 (fr) * | 2002-01-23 | 2004-02-27 | Servier Lab | Composition pharmaceutique orodispersible d'agomelatine |
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2004
- 2004-06-28 AR ARP040102269A patent/AR047553A1/es unknown
- 2004-06-29 BR BRPI0411665-8A patent/BRPI0411665A/pt not_active Application Discontinuation
- 2004-06-29 MX MXPA06000018A patent/MXPA06000018A/es not_active Application Discontinuation
- 2004-06-29 KR KR1020057024442A patent/KR20060032598A/ko not_active Withdrawn
- 2004-06-29 AT AT04738961T patent/ATE499096T1/de not_active IP Right Cessation
- 2004-06-29 CA CA002530880A patent/CA2530880A1/en not_active Abandoned
- 2004-06-29 JP JP2006517965A patent/JP2007513052A/ja active Pending
- 2004-06-29 US US10/558,494 patent/US20060205754A1/en not_active Abandoned
- 2004-06-29 EP EP04738961A patent/EP1643985B1/en not_active Expired - Lifetime
- 2004-06-29 DK DK04738961.4T patent/DK1643985T3/da active
- 2004-06-29 AU AU2004253225A patent/AU2004253225A1/en not_active Abandoned
- 2004-06-29 WO PCT/DK2004/000464 patent/WO2005002562A1/en not_active Ceased
- 2004-06-29 DE DE602004031527T patent/DE602004031527D1/de not_active Expired - Lifetime
- 2004-06-29 CN CNA2004800191380A patent/CN1852706A/zh active Pending
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2005
- 2005-11-28 IS IS8154A patent/IS8154A/is unknown
-
2006
- 2006-01-03 IL IL172965A patent/IL172965A0/en unknown
- 2006-01-17 NO NO20060242A patent/NO20060242L/no not_active Application Discontinuation
-
2010
- 2010-04-21 US US12/764,348 patent/US20100267772A1/en not_active Abandoned
-
2012
- 2012-07-19 US US13/552,699 patent/US20130217776A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| AU2004253225A1 (en) | 2005-01-13 |
| US20130217776A1 (en) | 2013-08-22 |
| EP1643985A1 (en) | 2006-04-12 |
| EP1643985B1 (en) | 2011-02-23 |
| DK1643985T3 (da) | 2011-06-06 |
| ATE499096T1 (de) | 2011-03-15 |
| CN1852706A (zh) | 2006-10-25 |
| IS8154A (is) | 2005-11-28 |
| US20060205754A1 (en) | 2006-09-14 |
| CA2530880A1 (en) | 2005-01-13 |
| BRPI0411665A (pt) | 2006-08-08 |
| AR047553A1 (es) | 2006-01-25 |
| MXPA06000018A (es) | 2006-03-21 |
| NO20060242L (no) | 2006-01-17 |
| JP2007513052A (ja) | 2007-05-24 |
| IL172965A0 (en) | 2006-06-11 |
| US20100267772A1 (en) | 2010-10-21 |
| WO2005002562A1 (en) | 2005-01-13 |
| DE602004031527D1 (de) | 2011-04-07 |
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