KR101714820B1 - 11(베타)-ｈｓｄ1의 억제제로서 3,3-이치환된-(8-아자-비시클로[3.2.1]옥트-8-일)-[5-(1h-피라졸-4-일)-티오펜-3-일]-메탄온 - Google Patents

11(베타)-ｈｓｄ1의 억제제로서 3,3-이치환된-(8-아자-비시클로[3.2.1]옥트-8-일)-[5-(1h-피라졸-4-일)-티오펜-3-일]-메탄온 Download PDF

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KR101714820B1
KR101714820B1 KR1020127028597A KR20127028597A KR101714820B1 KR 101714820 B1 KR101714820 B1 KR 101714820B1 KR 1020127028597 A KR1020127028597 A KR 1020127028597A KR 20127028597 A KR20127028597 A KR 20127028597A KR 101714820 B1 KR101714820 B1 KR 101714820B1
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스캇 피터 웹스터
조나단 로버트 섹클
브라이언 로버트 월컬
피터 월드
토마스 데이빗 펠린
헤이즐 조안 디케
트레볼 로버트 퍼리어
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KR1020127028597A 2010-04-29 2011-03-10 11(베타)-ｈｓｄ1의 억제제로서 3,3-이치환된-(8-아자-비시클로[3.2.1]옥트-8-일)-[5-(1h-피라졸-4-일)-티오펜-3-일]-메탄온 Active KR101714820B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US32945310P 2010-04-29 2010-04-29
US61/329,453 2010-04-29
PCT/GB2011/000345 WO2011135276A1 (en) 2010-04-29 2011-03-10 3, 3 -disubstituted- ( 8 - aza - bicyclo [3.2.1] oct- 8 - yl) -[5- (1h - pyrazol - 4 -yl) -thiophen-3 -yl] methanones as inhibitors of 11 (beta) -hsd1

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KR20130079379A KR20130079379A (ko) 2013-07-10
KR101714820B1 true KR101714820B1 (ko) 2017-03-09

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GB0724251D0 (en) 2007-12-12 2008-02-06 Univ Edinburgh Therapeutic compounds and their use
GB0804685D0 (en) 2008-03-13 2008-04-16 Univ Edinburgh Therapeutic compounds and their use
US8642621B2 (en) 2009-09-16 2014-02-04 The University Of Edinburgh (4-phenyl-piperidin-1-yl)-[5-(1H-pyrazol-4-yl)-thiophen-3-yl]-methanone compounds and their use
CN102947295B (zh) 2010-04-29 2016-01-20 爱丁堡大学 作为11β-HSD1抑制剂的3,3-二取代的-(8-氮杂双环[3.2.1]辛烷-8-基)-[5-(1H-吡唑-4基)-噻吩-3-基]-甲酮
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