KR101638999B1 - 피리미딘 함유 ｎｎｒｔｉ와 ｒｔ 저해제의 배합물 - Google Patents

피리미딘 함유 ｎｎｒｔｉ와 ｒｔ 저해제의 배합물 Download PDF

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Publication number
KR101638999B1
KR101638999B1 KR1020137024817A KR20137024817A KR101638999B1 KR 101638999 B1 KR101638999 B1 KR 101638999B1 KR 1020137024817 A KR1020137024817 A KR 1020137024817A KR 20137024817 A KR20137024817 A KR 20137024817A KR 101638999 B1 KR101638999 B1 KR 101638999B1
Authority
KR
South Korea
Prior art keywords
tmc278
reverse transcriptase
hiv
amino
inhibitor
Prior art date
Application number
KR1020137024817A
Other languages
English (en)
Korean (ko)
Other versions
KR20130127515A (ko
Inventor
파울 스토펠스
Original Assignee
얀센 사이언시즈 아일랜드 유씨
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43778148&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR101638999(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 얀센 사이언시즈 아일랜드 유씨 filed Critical 얀센 사이언시즈 아일랜드 유씨
Priority claimed from PCT/EP2004/052028 external-priority patent/WO2005021001A1/en
Publication of KR20130127515A publication Critical patent/KR20130127515A/ko
Application granted granted Critical
Publication of KR101638999B1 publication Critical patent/KR101638999B1/ko

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1020137024817A 2003-09-03 2004-09-03 피리미딘 함유 ｎｎｒｔｉ와 ｒｔ 저해제의 배합물 KR101638999B1 (ko)

Applications Claiming Priority (13)

Application Number Priority Date Filing Date Title
US49977103P 2003-09-03 2003-09-03
EP03103275.8 2003-09-03
EP03103275 2003-09-03
US60/499,771 2003-09-03
EP03103319.4 2003-09-08
EP03103319 2003-09-08
EP03103335 2003-09-10
EP03103335.0 2003-09-10
EP03103668 2003-10-02
EP03103668.4 2003-10-02
US50848603P 2003-10-03 2003-10-03
US60/508,486 2003-10-03
PCT/EP2004/052028 WO2005021001A1 (en) 2003-09-03 2004-09-03 Combinations of a pyrimidine containing nnrti with rt inhibitors

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020117025799A Division KR101539245B1 (ko) 2003-09-03 2004-09-03 피리미딘 함유 ｎｎｒｔｉ와 ｒｔ 저해제의 배합물

Publications (2)

Publication Number Publication Date
KR20130127515A KR20130127515A (ko) 2013-11-22
KR101638999B1 true KR101638999B1 (ko) 2016-07-12

Family

ID=43778148

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020117025799A KR101539245B1 (ko) 2003-09-03 2004-09-03 피리미딘 함유 ｎｎｒｔｉ와 ｒｔ 저해제의 배합물
KR1020137024817A KR101638999B1 (ko) 2003-09-03 2004-09-03 피리미딘 함유 ｎｎｒｔｉ와 ｒｔ 저해제의 배합물

Family Applications Before (1)

Application Number Title Priority Date Filing Date
KR1020117025799A KR101539245B1 (ko) 2003-09-03 2004-09-03 피리미딘 함유 ｎｎｒｔｉ와 ｒｔ 저해제의 배합물

Country Status (9)

Country Link
KR (2) KR101539245B1 (ru)
CN (1) CN102319433A (ru)
DK (1) DK1663240T4 (ru)
EA (1) EA014840B1 (ru)
ES (1) ES2542017T5 (ru)
HU (1) HUE025576T2 (ru)
PT (1) PT1663240E (ru)
SI (1) SI1663240T2 (ru)
TW (1) TWI365744B (ru)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003016306A1 (en) 2001-08-13 2003-02-27 Janssen Pharmaceutica N.V. Hiv inhibiting pyrimidines derivatives

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003016306A1 (en) 2001-08-13 2003-02-27 Janssen Pharmaceutica N.V. Hiv inhibiting pyrimidines derivatives

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
Clin. Infect. Dis., Vol. 34, pp. 686-692(2002)

Also Published As

Publication number Publication date
TW200524612A (en) 2005-08-01
DK1663240T4 (da) 2023-04-17
KR101539245B1 (ko) 2015-07-27
HUE025576T2 (en) 2016-04-28
PT1663240E (pt) 2015-09-01
SI1663240T1 (sl) 2015-10-30
EA014840B1 (ru) 2011-02-28
DK1663240T3 (en) 2015-07-20
ES2542017T3 (es) 2015-07-29
ES2542017T5 (es) 2023-06-15
KR20130127515A (ko) 2013-11-22
EA200600522A1 (ru) 2006-08-25
SI1663240T2 (sl) 2023-05-31
TWI365744B (en) 2012-06-11
CN102319433A (zh) 2012-01-18
KR20110132475A (ko) 2011-12-07

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KR101638999B1 (ko) 피리미딘 함유 ｎｎｒｔｉ와 ｒｔ 저해제의 배합물
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