KR101575679B1 - 코어 및 하나 이상의 배리어 층을 포함하는 방출 제어형 경구 투여 제제 - Google Patents
코어 및 하나 이상의 배리어 층을 포함하는 방출 제어형 경구 투여 제제 Download PDFInfo
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- KR101575679B1 KR101575679B1 KR1020097006438A KR20097006438A KR101575679B1 KR 101575679 B1 KR101575679 B1 KR 101575679B1 KR 1020097006438 A KR1020097006438 A KR 1020097006438A KR 20097006438 A KR20097006438 A KR 20097006438A KR 101575679 B1 KR101575679 B1 KR 101575679B1
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- 229960004355 vindesine Drugs 0.000 description 1
- UGGWPQSBPIFKDZ-KOTLKJBCSA-N vindesine Chemical compound C([C@@H](C[C@]1(C(=O)OC)C=2C(=CC3=C([C@]45[C@H]([C@@]([C@H](O)[C@]6(CC)C=CCN([C@H]56)CC4)(O)C(N)=O)N3C)C=2)OC)C[C@@](C2)(O)CC)N2CCC2=C1N=C1[C]2C=CC=C1 UGGWPQSBPIFKDZ-KOTLKJBCSA-N 0.000 description 1
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4422—1,4-Dihydropyridines, e.g. nifedipine, nicardipine
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- A61K9/0012—Galenical forms characterised by the site of application
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
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- A—HUMAN NECESSITIES
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- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
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- A—HUMAN NECESSITIES
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- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
- A61K9/2846—Poly(meth)acrylates
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- A—HUMAN NECESSITIES
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- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| ES2547226T5 (es) * | 2006-08-30 | 2020-06-12 | Jagotec Ag | Formulaciones de dosificación oral de liberación controlada que comprenden un núcleo y una o más capas de barrera |
| EP2180883B1 (en) * | 2007-07-23 | 2017-01-11 | Pharmathen S.A. | Pharmaceutical composition containing dihydropyridine calcium channel antagonist and method for the preparation thereof |
| EP2187873B1 (en) | 2007-08-13 | 2018-07-25 | Abuse Deterrent Pharmaceutical Llc | Abuse resistant drugs, method of use and method of making |
| AU2009224254A1 (en) * | 2008-03-11 | 2009-09-17 | Takeda Pharmaceutical Company Limited | Orally-disintegrating solid preparation |
| MX2011001384A (es) | 2008-08-06 | 2011-09-27 | Gosforth Ct Holdings Pty Ltd | Composiciones y metodos para tratar trastornos psiquiatricos. |
| EP2331094A4 (en) * | 2008-08-29 | 2011-10-26 | Uab Research Foundation | NOVEL AGENT AGAINST ARTHHYTHMIA |
| KR20100069170A (ko) * | 2008-12-16 | 2010-06-24 | 삼일제약주식회사 | 라시디핀 함유 과립 및 이를 포함하는 약학 조성물 |
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2007
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- 2007-08-29 US US11/847,012 patent/US20080057123A1/en not_active Abandoned
- 2007-08-29 JP JP2009525973A patent/JP2010501607A/ja not_active Abandoned
- 2007-08-29 CA CA2662123A patent/CA2662123C/en active Active
- 2007-08-29 KR KR1020097006438A patent/KR101575679B1/ko active Active
- 2007-08-29 WO PCT/EP2007/007545 patent/WO2008025532A1/en not_active Ceased
- 2007-08-29 MX MX2009002235A patent/MX2009002235A/es unknown
- 2007-08-29 AU AU2007291506A patent/AU2007291506A1/en not_active Abandoned
- 2007-08-29 EP EP07801970.0A patent/EP2063872B2/en active Active
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- 2007-08-29 JP JP2009525976A patent/JP2010501609A/ja active Pending
- 2007-08-29 KR KR1020097006435A patent/KR20090065519A/ko not_active Withdrawn
- 2007-08-29 MX MX2009002236A patent/MX2009002236A/es active IP Right Grant
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Also Published As
| Publication number | Publication date |
|---|---|
| JP5788547B2 (ja) | 2015-09-30 |
| US20080063711A1 (en) | 2008-03-13 |
| US20080057123A1 (en) | 2008-03-06 |
| EP2063872A1 (en) | 2009-06-03 |
| ZA200901688B (en) | 2014-02-26 |
| WO2008025535A1 (en) | 2008-03-06 |
| AU2007291509B2 (en) | 2013-05-02 |
| EP2063871A1 (en) | 2009-06-03 |
| KR20090065520A (ko) | 2009-06-22 |
| AU2007291509A1 (en) | 2008-03-06 |
| JP2010501609A (ja) | 2010-01-21 |
| CA2662123A1 (en) | 2008-03-06 |
| KR20090065519A (ko) | 2009-06-22 |
| JP2014114323A (ja) | 2014-06-26 |
| MX2009002236A (es) | 2009-03-13 |
| ES2547226T5 (es) | 2020-06-12 |
| JP2010501607A (ja) | 2010-01-21 |
| CA2662122A1 (en) | 2008-03-06 |
| MX2009002235A (es) | 2009-03-13 |
| ES2547226T3 (es) | 2015-10-02 |
| CA2662123C (en) | 2015-12-01 |
| WO2008025532A1 (en) | 2008-03-06 |
| US20160008288A1 (en) | 2016-01-14 |
| EP2063872B2 (en) | 2019-12-04 |
| US9622980B2 (en) | 2017-04-18 |
| US9101544B2 (en) | 2015-08-11 |
| AU2007291506A1 (en) | 2008-03-06 |
| EP2063872B1 (en) | 2015-05-06 |
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