KR101567969B1 - 벤질페닐 시클로헥산 유도체 및 이의 사용 방법 - Google Patents

벤질페닐 시클로헥산 유도체 및 이의 사용 방법 Download PDF

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Publication number
KR101567969B1
KR101567969B1 KR1020107015420A KR20107015420A KR101567969B1 KR 101567969 B1 KR101567969 B1 KR 101567969B1 KR 1020107015420 A KR1020107015420 A KR 1020107015420A KR 20107015420 A KR20107015420 A KR 20107015420A KR 101567969 B1 KR101567969 B1 KR 101567969B1
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South Korea
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phenyl
diabetes
chloro
rti
compound
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Expired - Fee Related
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KR1020107015420A
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English (en)
Korean (ko)
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KR20100098690A (ko
Inventor
위안웨이 첸
쿤 펭
릴리 장
빈후아 엘브이
바이후아 쉬
지아지아 동
지얀 두
얀 펭
게 수
바산타쿠말 라자판
브라이언 시드
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테라코스, 인코포레이티드
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Publication of KR20100098690A publication Critical patent/KR20100098690A/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/04—Carbocyclic radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biotechnology (AREA)
  • Obesity (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyrane Compounds (AREA)
KR1020107015420A 2007-12-13 2008-12-11 벤질페닐 시클로헥산 유도체 및 이의 사용 방법 Expired - Fee Related KR101567969B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US1351707P 2007-12-13 2007-12-13
US61/013,517 2007-12-13

Publications (2)

Publication Number Publication Date
KR20100098690A KR20100098690A (ko) 2010-09-08
KR101567969B1 true KR101567969B1 (ko) 2015-11-10

Family

ID=40754059

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020107015420A Expired - Fee Related KR101567969B1 (ko) 2007-12-13 2008-12-11 벤질페닐 시클로헥산 유도체 및 이의 사용 방법

Country Status (16)

Country Link
US (1) US8129434B2 (https=)
EP (1) EP2230907B1 (https=)
JP (1) JP5507464B2 (https=)
KR (1) KR101567969B1 (https=)
CN (1) CN101938902B (https=)
AR (2) AR071268A1 (https=)
AU (1) AU2008335080B2 (https=)
BR (1) BRPI0819930A2 (https=)
CA (1) CA2707909C (https=)
IL (1) IL206234A0 (https=)
NZ (1) NZ586639A (https=)
RU (1) RU2505521C2 (https=)
TW (1) TWI426081B (https=)
UA (1) UA101004C2 (https=)
WO (1) WO2009076550A1 (https=)
ZA (1) ZA201004400B (https=)

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TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
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WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
CN103570671B (zh) * 2012-09-26 2016-03-30 上海天慈生物谷生物工程有限公司 一种降糖化合物及其制法和应用
WO2015051484A1 (en) 2013-10-12 2015-04-16 Theracos, Inc. Preparation of hydroxy-benzylbenzene derivatives
MX376097B (es) 2013-12-17 2025-03-07 Boehringer Ingelheim Vetmedica Gmbh Inhibidores de sglt2 para usarse en el tratamiento o prevención de trastornos metabólicos en animales felinos.
US10759729B2 (en) * 2016-11-07 2020-09-01 The Chinese University Of Hong Kong Compounds for treating diabetes
CN116785268A (zh) * 2022-03-14 2023-09-22 江苏万邦生化医药集团有限责任公司 一种sglt-2抑制剂的药物组合物

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Also Published As

Publication number Publication date
NZ586639A (en) 2011-06-30
IL206234A0 (en) 2010-12-30
EP2230907A4 (en) 2015-04-08
RU2010128940A (ru) 2012-01-20
KR20100098690A (ko) 2010-09-08
TW200932755A (en) 2009-08-01
AU2008335080B2 (en) 2014-06-05
US20090156516A1 (en) 2009-06-18
AR113211A2 (es) 2020-02-19
BRPI0819930A2 (pt) 2016-05-17
AR071268A1 (es) 2010-06-09
WO2009076550A1 (en) 2009-06-18
CA2707909A1 (en) 2009-06-18
JP2011506469A (ja) 2011-03-03
ZA201004400B (en) 2014-10-29
EP2230907A1 (en) 2010-09-29
RU2505521C2 (ru) 2014-01-27
UA101004C2 (en) 2013-02-25
CN101938902A (zh) 2011-01-05
EP2230907B1 (en) 2018-05-09
CN101938902B (zh) 2014-07-02
JP5507464B2 (ja) 2014-05-28
CA2707909C (en) 2016-10-18
US8129434B2 (en) 2012-03-06
TWI426081B (zh) 2014-02-11
AU2008335080A1 (en) 2009-06-18

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