KR101222774B1 - 수지 상 펩티드 고리화 - Google Patents

수지 상 펩티드 고리화 Download PDF

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Publication number
KR101222774B1
KR101222774B1 KR1020077010506A KR20077010506A KR101222774B1 KR 101222774 B1 KR101222774 B1 KR 101222774B1 KR 1020077010506 A KR1020077010506 A KR 1020077010506A KR 20077010506 A KR20077010506 A KR 20077010506A KR 101222774 B1 KR101222774 B1 KR 101222774B1
Authority
KR
South Korea
Prior art keywords
peptide
resin
cysteine
solid phase
amino acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
KR1020077010506A
Other languages
English (en)
Korean (ko)
Other versions
KR20070084099A (ko
Inventor
스테판 바라이
올레크 베르비츠키
토마스 차이터
Original Assignee
론자 아게
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 론자 아게 filed Critical 론자 아게
Publication of KR20070084099A publication Critical patent/KR20070084099A/ko
Application granted granted Critical
Publication of KR101222774B1 publication Critical patent/KR101222774B1/ko
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Polyamides (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1020077010506A 2004-10-19 2005-10-18 수지 상 펩티드 고리화 Expired - Fee Related KR101222774B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP04024813.0 2004-10-19
EP04024813 2004-10-19
EP05008979 2005-04-25
EP05008979.6 2005-04-25
PCT/EP2005/011182 WO2006045483A2 (en) 2004-10-19 2005-10-18 On-resin peptide cyclization

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020127016164A Division KR101276463B1 (ko) 2004-10-19 2005-10-18 수지 상 펩티드 고리화

Publications (2)

Publication Number Publication Date
KR20070084099A KR20070084099A (ko) 2007-08-24
KR101222774B1 true KR101222774B1 (ko) 2013-01-15

Family

ID=36096370

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020077010506A Expired - Fee Related KR101222774B1 (ko) 2004-10-19 2005-10-18 수지 상 펩티드 고리화
KR1020127016164A Expired - Fee Related KR101276463B1 (ko) 2004-10-19 2005-10-18 수지 상 펩티드 고리화

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR1020127016164A Expired - Fee Related KR101276463B1 (ko) 2004-10-19 2005-10-18 수지 상 펩티드 고리화

Country Status (16)

Country Link
US (1) US7994280B2 (enExample)
EP (1) EP1805203B1 (enExample)
JP (1) JP4927746B2 (enExample)
KR (2) KR101222774B1 (enExample)
CN (1) CN101111510B (enExample)
AT (1) ATE455123T1 (enExample)
AU (1) AU2005298991B2 (enExample)
BR (1) BRPI0516929A (enExample)
CA (1) CA2588098A1 (enExample)
DE (1) DE602005018952D1 (enExample)
DK (1) DK1805203T3 (enExample)
ES (1) ES2339791T3 (enExample)
IL (1) IL182575A (enExample)
PT (1) PT1805203E (enExample)
TW (1) TW200628487A (enExample)
WO (1) WO2006045483A2 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101538316B (zh) * 2009-01-13 2012-09-05 深圳翰宇药业股份有限公司 一种固相法制备Eptifibatide的方法
WO2013112548A1 (en) * 2012-01-23 2013-08-01 University Of South Florida Gamma-aapeptides with potent and broad-spectrum antimicrobial activity
CN108218964A (zh) * 2018-01-30 2018-06-29 江南大学 一种固相载体上酶法合成环肽方法
WO2024234959A1 (en) * 2023-05-18 2024-11-21 Versitech Limited Late-stage peptide cyclization to form disulfide mimetics

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003093302A2 (en) * 2002-05-03 2003-11-13 Avecia Limited Process for the synthesis of peptides amides by side-chain attachement to a solid phase
WO2004092202A1 (en) 2003-04-07 2004-10-28 Novetide, Ltd. Process for production of cyclic peptides
WO2005121164A1 (en) 2004-06-14 2005-12-22 Usv Limited Process for the preparation of peptides
CN100500805C (zh) * 2006-11-07 2009-06-17 武汉钢铁集团鄂城钢铁有限责任公司 除尘焦粉回配煤炼焦方法及其工艺

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4606856A (en) * 1985-03-18 1986-08-19 Seyler Jay K [Des-1-amino, 8-glycine]calcitonin
US5770687A (en) * 1995-06-07 1998-06-23 Peptor Limited Comformationally constrained backbone cyclized somatostatin analogs
CN1222537C (zh) * 2002-11-14 2005-10-12 吉尔生化（上海）有限公司 一种制备依非巴特的工艺

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003093302A2 (en) * 2002-05-03 2003-11-13 Avecia Limited Process for the synthesis of peptides amides by side-chain attachement to a solid phase
WO2004092202A1 (en) 2003-04-07 2004-10-28 Novetide, Ltd. Process for production of cyclic peptides
WO2005121164A1 (en) 2004-06-14 2005-12-22 Usv Limited Process for the preparation of peptides
CN100500805C (zh) * 2006-11-07 2009-06-17 武汉钢铁集团鄂城钢铁有限责任公司 除尘焦粉回配煤炼焦方法及其工艺

Also Published As

Publication number Publication date
WO2006045483A3 (en) 2006-07-13
DK1805203T3 (da) 2010-05-17
IL182575A0 (en) 2007-07-24
KR20070084099A (ko) 2007-08-24
WO2006045483A2 (en) 2006-05-04
AU2005298991B2 (en) 2011-03-03
PT1805203E (pt) 2010-04-19
JP4927746B2 (ja) 2012-05-09
BRPI0516929A (pt) 2008-09-23
TW200628487A (en) 2006-08-16
US20080200647A1 (en) 2008-08-21
US7994280B2 (en) 2011-08-09
AU2005298991A1 (en) 2006-05-04
EP1805203A2 (en) 2007-07-11
ATE455123T1 (de) 2010-01-15
CN101111510A (zh) 2008-01-23
CA2588098A1 (en) 2006-05-04
KR101276463B1 (ko) 2013-06-19
DE602005018952D1 (de) 2010-03-04
KR20120088855A (ko) 2012-08-08
JP2008517016A (ja) 2008-05-22
ES2339791T3 (es) 2010-05-25
EP1805203B1 (en) 2010-01-13
CN101111510B (zh) 2011-09-14
IL182575A (en) 2012-07-31

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