KR100956898B1 - 인단 아세트산 유도체, 및 이의 약제로서의 용도, 중간체및 제조 방법 - Google Patents

인단 아세트산 유도체, 및 이의 약제로서의 용도, 중간체및 제조 방법 Download PDF

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KR100956898B1
KR100956898B1 KR1020047001188A KR20047001188A KR100956898B1 KR 100956898 B1 KR100956898 B1 KR 100956898B1 KR 1020047001188 A KR1020047001188 A KR 1020047001188A KR 20047001188 A KR20047001188 A KR 20047001188A KR 100956898 B1 KR100956898 B1 KR 100956898B1
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dihydro
methyl
delete delete
ethoxy
oxazol
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Expired - Fee Related
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KR20040028950A (ko
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데렉 비. 로웨
필립 엘. 위킨스
신 마
밍바오 장
윌리엄 에이치. 불록
필립 디.지. 코이쉬
잉고 아. 무게
안드레아스 스톨레
밍 왕
야민. 왕
쳉지 장
하이-준 장
레이 주
마나미 츠츠미
제임스 엔. 리빙스턴
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바이엘 파마슈티칼스 코포레이션
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Publication of KR20040028950A publication Critical patent/KR20040028950A/ko
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Publication of KR100956898B1 publication Critical patent/KR100956898B1/ko
Assigned to 바이엘 헬스케어 엘엘씨 reassignment 바이엘 헬스케어 엘엘씨 권리의 전부이전등록 Assignors: 바이엘 파마슈티칼스 코포레이션
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    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07C59/40—Unsaturated compounds
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    • C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/73—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids
    • C07C69/732—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids of unsaturated hydroxy carboxylic acids
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  • Urology & Nephrology (AREA)
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  • Biochemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
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  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
KR1020047001188A 2001-07-27 2002-07-25 인단 아세트산 유도체, 및 이의 약제로서의 용도, 중간체및 제조 방법 Expired - Fee Related KR100956898B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US30850001P 2001-07-27 2001-07-27
US60/308,500 2001-07-27
US37304802P 2002-04-16 2002-04-16
US60/373,048 2002-04-16
PCT/US2002/023614 WO2003011842A1 (en) 2001-07-27 2002-07-25 Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation

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KR1020097023801A Division KR100987267B1 (ko) 2001-07-27 2002-07-25 인단 아세트산 유도체, 및 이의 약제로서의 용도, 중간체 및 제조 방법

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KR20040028950A KR20040028950A (ko) 2004-04-03
KR100956898B1 true KR100956898B1 (ko) 2010-05-11

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KR1020047001188A Expired - Fee Related KR100956898B1 (ko) 2001-07-27 2002-07-25 인단 아세트산 유도체, 및 이의 약제로서의 용도, 중간체및 제조 방법
KR1020097023801A Expired - Fee Related KR100987267B1 (ko) 2001-07-27 2002-07-25 인단 아세트산 유도체, 및 이의 약제로서의 용도, 중간체 및 제조 방법

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US (4) US6828335B2 (https=)
EP (1) EP1414809B1 (https=)
JP (1) JP4510447B2 (https=)
KR (2) KR100956898B1 (https=)
CN (1) CN100528850C (https=)
AR (1) AR036237A1 (https=)
AT (1) ATE388944T1 (https=)
AU (2) AU2002319693B2 (https=)
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CA (2) CA2455620C (https=)
CO (1) CO5560561A2 (https=)
CY (1) CY1107370T1 (https=)
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IL (3) IL159960A0 (https=)
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PT (1) PT1414809E (https=)
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Publication number Priority date Publication date Assignee Title
US20110065129A1 (en) * 2001-07-27 2011-03-17 Lowe Derek B Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation
AR036237A1 (es) * 2001-07-27 2004-08-25 Bayer Corp Derivados del acido indan acetico, intermediarios, y metodo para su preparacion, composicion farmaceutica y el uso de dichos derivados para la manufactura de un medicamento
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