JPWO2024181437A5 - - Google Patents

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Publication number
JPWO2024181437A5
JPWO2024181437A5 JP2025503931A JP2025503931A JPWO2024181437A5 JP WO2024181437 A5 JPWO2024181437 A5 JP WO2024181437A5 JP 2025503931 A JP2025503931 A JP 2025503931A JP 2025503931 A JP2025503931 A JP 2025503931A JP WO2024181437 A5 JPWO2024181437 A5 JP WO2024181437A5
Authority
JP
Japan
Prior art keywords
phenanthrolin
indazol
amino
solvate
fluoro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2025503931A
Other languages
English (en)
Japanese (ja)
Other versions
JP7742517B2 (ja
JPWO2024181437A1 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/JP2024/007072 external-priority patent/WO2024181437A1/ja
Publication of JPWO2024181437A1 publication Critical patent/JPWO2024181437A1/ja
Priority to JP2025148435A priority Critical patent/JP2026000973A/ja
Application granted granted Critical
Publication of JP7742517B2 publication Critical patent/JP7742517B2/ja
Publication of JPWO2024181437A5 publication Critical patent/JPWO2024181437A5/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2025503931A 2023-02-28 2024-02-27 Myt1阻害活性を有する含窒素複素環化合物 Active JP7742517B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2025148435A JP2026000973A (ja) 2023-02-28 2025-09-08 Myt1阻害活性を有する含窒素複素環化合物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2023029673 2023-02-28
JP2023029673 2023-02-28
PCT/JP2024/007072 WO2024181437A1 (ja) 2023-02-28 2024-02-27 Myt1阻害活性を有する含窒素複素環化合物

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025148435A Division JP2026000973A (ja) 2023-02-28 2025-09-08 Myt1阻害活性を有する含窒素複素環化合物

Publications (3)

Publication Number Publication Date
JPWO2024181437A1 JPWO2024181437A1 (https=) 2024-09-06
JP7742517B2 JP7742517B2 (ja) 2025-09-19
JPWO2024181437A5 true JPWO2024181437A5 (https=) 2025-10-02

Family

ID=92589871

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2025503931A Active JP7742517B2 (ja) 2023-02-28 2024-02-27 Myt1阻害活性を有する含窒素複素環化合物
JP2025148435A Pending JP2026000973A (ja) 2023-02-28 2025-09-08 Myt1阻害活性を有する含窒素複素環化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2025148435A Pending JP2026000973A (ja) 2023-02-28 2025-09-08 Myt1阻害活性を有する含窒素複素環化合物

Country Status (15)

Country Link
US (1) US20260062412A1 (https=)
EP (1) EP4647424A1 (https=)
JP (2) JP7742517B2 (https=)
KR (1) KR20250153810A (https=)
CN (1) CN120677145A (https=)
AR (1) AR131956A1 (https=)
AU (1) AU2024229746A1 (https=)
CL (1) CL2025002607A1 (https=)
CO (1) CO2025011476A2 (https=)
CR (1) CR20250376A (https=)
IL (1) IL322675A (https=)
MX (1) MX2025010048A (https=)
PE (1) PE20252436A1 (https=)
TW (1) TW202446768A (https=)
WO (1) WO2024181437A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2025182927A1 (ja) * 2024-02-27 2025-09-04 中外製薬株式会社 Myt1阻害剤の用途
WO2026054022A1 (ja) * 2024-09-05 2026-03-12 中外製薬株式会社 Myt1阻害活性を有する含窒素複素環化合物の製剤

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3202661A (en) * 1962-11-27 1965-08-24 Hoffmann La Roche Substituted 3-amino 4-phenyl quinolones
US4014883A (en) * 1973-09-10 1977-03-29 Hoffmann-La Roche Inc. Indoloquinolines, intermediates and processes
AU742452B2 (en) * 1997-08-28 2002-01-03 Bristol-Myers Squibb Company 4-aryl-3-aminoquinoline-2-one derivatives as potassium channel modulators
WO2002076396A2 (en) * 2001-03-23 2002-10-03 Smithkline Beecham Corporation Compounds useful as kinase inhibitors for the treatment of hyperproliferative diseases
CA2539760C (en) * 2003-09-23 2011-01-25 Merck & Co., Inc. Quinoline potassium channel inhibitors
GB0420970D0 (en) * 2004-09-21 2004-10-20 Smithkline Beecham Corp Novel triazoloquinoline compounds
WO2015088564A1 (en) * 2013-12-13 2015-06-18 Sunovion Pharmaceuticals Inc. P2x4 receptor modulating compounds
US11026937B2 (en) * 2016-09-12 2021-06-08 Padlock Therapeutics, Inc. Heteroaryl inhibitors of PAD4
CN109111426B (zh) * 2017-06-23 2021-12-14 中国科学院上海药物研究所 一类稠合双环杂芳基或芳基化合物,及其用途
US20240398799A1 (en) * 2021-08-19 2024-12-05 Engine Biosciences Pte. Ltd. Compositions and methods for generating synthetic lethality in tumors
CN114369061B (zh) * 2022-01-28 2024-05-03 济南同路医药科技发展有限公司 一种氯硝西泮有关物质b的制备方法
WO2024048687A1 (ja) * 2022-08-31 2024-03-07 中外製薬株式会社 Myt1阻害剤と化学療法剤を併用する、rb1の機能低下が生じている患者のがんの治療剤及び治療方法

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