JPWO2023275337A5 - - Google Patents
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- Publication number
- JPWO2023275337A5 JPWO2023275337A5 JP2023580900A JP2023580900A JPWO2023275337A5 JP WO2023275337 A5 JPWO2023275337 A5 JP WO2023275337A5 JP 2023580900 A JP2023580900 A JP 2023580900A JP 2023580900 A JP2023580900 A JP 2023580900A JP WO2023275337 A5 JPWO2023275337 A5 JP WO2023275337A5
- Authority
- JP
- Japan
- Prior art keywords
- compound
- carried out
- formula
- protecting group
- amino protecting
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (11)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP21182956.9 | 2021-06-30 | ||
| EP21182956 | 2021-06-30 | ||
| EP21183316 | 2021-07-01 | ||
| EP21183316.5 | 2021-07-01 | ||
| US202163217783P | 2021-07-02 | 2021-07-02 | |
| US63/217,783 | 2021-07-02 | ||
| PCT/EP2021/086674 WO2023110138A1 (en) | 2021-12-17 | 2021-12-17 | Inhibitors of transglutaminases |
| EPPCT/EP2021/086674 | 2021-12-17 | ||
| EP2022065435 | 2022-06-07 | ||
| EPPCT/EP2022/065435 | 2022-06-07 | ||
| PCT/EP2022/068217 WO2023275337A1 (en) | 2021-06-30 | 2022-06-30 | Inhibitors of transglutaminases |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2024524457A JP2024524457A (ja) | 2024-07-05 |
| JP2024524457A5 JP2024524457A5 (https=) | 2026-03-25 |
| JPWO2023275337A5 true JPWO2023275337A5 (https=) | 2026-03-25 |
Family
ID=82547278
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023580900A Pending JP2024524457A (ja) | 2021-06-30 | 2022-06-30 | トランスグルタミナーゼの阻害剤 |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20240383856A1 (https=) |
| EP (1) | EP4192814B1 (https=) |
| JP (1) | JP2024524457A (https=) |
| KR (1) | KR20240028466A (https=) |
| CN (1) | CN117616011B (https=) |
| AU (1) | AU2022303109A1 (https=) |
| CL (1) | CL2023003921A1 (https=) |
| DK (1) | DK4192814T3 (https=) |
| ES (1) | ES2993597T3 (https=) |
| FI (1) | FI4192814T3 (https=) |
| HR (1) | HRP20241451T1 (https=) |
| HU (1) | HUE068724T2 (https=) |
| IL (1) | IL309476A (https=) |
| LT (1) | LT4192814T (https=) |
| MX (1) | MX2023015408A (https=) |
| PL (1) | PL4192814T3 (https=) |
| RS (1) | RS66080B1 (https=) |
| SI (1) | SI4192814T1 (https=) |
| WO (1) | WO2023275337A1 (https=) |
| ZA (1) | ZA202400821B (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2022301517A1 (en) * | 2021-06-30 | 2023-12-14 | Zedira Gmbh | Inhibitors of transglutaminases |
| JP7805983B2 (ja) | 2022-03-22 | 2026-01-26 | アッヴィ・インコーポレイテッド | ブルトン型チロシンキナーゼを分解するためのピリミジン |
| EP4637764A1 (en) | 2023-12-22 | 2025-10-29 | Zedira GmbH | Oxo-pyridine derivatives as inhibitors of transglutaminases for use in the treatment of pulmonary fibrosis |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102006052755A1 (de) * | 2006-11-08 | 2008-05-15 | N-Zyme Biotec Gmbh | Michaelsysteme als Transglutaminaseinhibitoren |
| EP2687511A1 (de) | 2012-07-17 | 2014-01-22 | Zedira GmbH | Pyridinonderivate als Gewebetransglutaminaseinhibitoren |
| EP3342779A1 (en) * | 2016-12-27 | 2018-07-04 | Zedira GmbH | Inhibitors of transglutaminases |
| TWI825144B (zh) * | 2018-08-10 | 2023-12-11 | 美商思達利醫藥公司 | 第二型轉麩醯胺酸酶(tg2)抑制劑 |
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2022
- 2022-06-30 KR KR1020247003531A patent/KR20240028466A/ko active Pending
- 2022-06-30 EP EP22741488.5A patent/EP4192814B1/en active Active
- 2022-06-30 MX MX2023015408A patent/MX2023015408A/es unknown
- 2022-06-30 WO PCT/EP2022/068217 patent/WO2023275337A1/en not_active Ceased
- 2022-06-30 LT LTEPPCT/EP2022/068217T patent/LT4192814T/lt unknown
- 2022-06-30 AU AU2022303109A patent/AU2022303109A1/en active Pending
- 2022-06-30 PL PL22741488.5T patent/PL4192814T3/pl unknown
- 2022-06-30 DK DK22741488.5T patent/DK4192814T3/da active
- 2022-06-30 CN CN202280045224.7A patent/CN117616011B/zh active Active
- 2022-06-30 US US18/572,134 patent/US20240383856A1/en active Pending
- 2022-06-30 HU HUE22741488A patent/HUE068724T2/hu unknown
- 2022-06-30 HR HRP20241451TT patent/HRP20241451T1/hr unknown
- 2022-06-30 FI FIEP22741488.5T patent/FI4192814T3/fi active
- 2022-06-30 SI SI202230065T patent/SI4192814T1/sl unknown
- 2022-06-30 IL IL309476A patent/IL309476A/en unknown
- 2022-06-30 RS RS20241159A patent/RS66080B1/sr unknown
- 2022-06-30 JP JP2023580900A patent/JP2024524457A/ja active Pending
- 2022-06-30 ES ES22741488T patent/ES2993597T3/es active Active
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2023
- 2023-12-28 CL CL2023003921A patent/CL2023003921A1/es unknown
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2024
- 2024-01-24 ZA ZA2024/00821A patent/ZA202400821B/en unknown