JPWO2023023112A5 - - Google Patents

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Publication number
JPWO2023023112A5
JPWO2023023112A5 JP2024506883A JP2024506883A JPWO2023023112A5 JP WO2023023112 A5 JPWO2023023112 A5 JP WO2023023112A5 JP 2024506883 A JP2024506883 A JP 2024506883A JP 2024506883 A JP2024506883 A JP 2024506883A JP WO2023023112 A5 JPWO2023023112 A5 JP WO2023023112A5
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JP
Japan
Prior art keywords
compound
further optionally
carried out
optionally
reacting
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024506883A
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English (en)
Japanese (ja)
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JP2024531115A (ja
JP2024531115A5 (https=
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/040540 external-priority patent/WO2023023112A1/en
Publication of JP2024531115A publication Critical patent/JP2024531115A/ja
Publication of JPWO2023023112A5 publication Critical patent/JPWO2023023112A5/ja
Publication of JP2024531115A5 publication Critical patent/JP2024531115A5/ja
Pending legal-status Critical Current

Links

JP2024506883A 2021-08-18 2022-08-17 ヒストン脱メチル化阻害剤を調製するためのプロセス Pending JP2024531115A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163234344P 2021-08-18 2021-08-18
US63/234,344 2021-08-18
PCT/US2022/040540 WO2023023112A1 (en) 2021-08-18 2022-08-17 Process for preparing histone demethylase inhibitors

Publications (3)

Publication Number Publication Date
JP2024531115A JP2024531115A (ja) 2024-08-29
JPWO2023023112A5 true JPWO2023023112A5 (https=) 2025-08-21
JP2024531115A5 JP2024531115A5 (https=) 2025-08-21

Family

ID=85239709

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024506883A Pending JP2024531115A (ja) 2021-08-18 2022-08-17 ヒストン脱メチル化阻害剤を調製するためのプロセス

Country Status (6)

Country Link
US (1) US20250129056A1 (https=)
EP (1) EP4387961A4 (https=)
JP (1) JP2024531115A (https=)
AU (1) AU2022331536A1 (https=)
CA (1) CA3227684A1 (https=)
WO (1) WO2023023112A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20200039938A1 (en) 2017-03-30 2020-02-06 Albert-Ludwigs-University Freiburg Kdm4 inhibitors
WO2022217100A1 (en) * 2021-04-09 2022-10-13 Tachyon Therapeutics, Inc. Treatment of cancer with kdm4 inhibitors
CN120225189A (zh) * 2022-09-21 2025-06-27 细胞基因公司 组蛋白去甲基化酶抑制剂3-({[(4r)-7-{甲基[4-(丙烷-2-基)苯基]氨基}-3,4-二氢-2h-1-苯并吡喃-4-基]甲基}氨基)吡啶-4-甲酸l-赖氨酸盐的结晶形式

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013143597A1 (en) * 2012-03-29 2013-10-03 Glaxo Group Limited Demethylase enzymes inhibitors
AR100997A1 (es) * 2014-06-25 2016-11-16 Quanticel Pharmaceuticals Inc Derivados de piridina como inhibidores de histona demetilasa
US20200039938A1 (en) * 2017-03-30 2020-02-06 Albert-Ludwigs-University Freiburg Kdm4 inhibitors

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