JPWO2022250108A5 - - Google Patents
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- Publication number
- JPWO2022250108A5 JPWO2022250108A5 JP2023524226A JP2023524226A JPWO2022250108A5 JP WO2022250108 A5 JPWO2022250108 A5 JP WO2022250108A5 JP 2023524226 A JP2023524226 A JP 2023524226A JP 2023524226 A JP2023524226 A JP 2023524226A JP WO2022250108 A5 JPWO2022250108 A5 JP WO2022250108A5
- Authority
- JP
- Japan
- Prior art keywords
- alkoxy
- alkyl
- same
- halogen atoms
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2021088034 | 2021-05-26 | ||
| PCT/JP2022/021531 WO2022250108A1 (ja) | 2021-05-26 | 2022-05-26 | フェニルウレア誘導体 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2022250108A1 JPWO2022250108A1 (https=) | 2022-12-01 |
| JPWO2022250108A5 true JPWO2022250108A5 (https=) | 2025-06-02 |
Family
ID=84228903
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023524226A Pending JPWO2022250108A1 (https=) | 2021-05-26 | 2022-05-26 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20240308960A1 (https=) |
| EP (1) | EP4353309A4 (https=) |
| JP (1) | JPWO2022250108A1 (https=) |
| CN (1) | CN117561238A (https=) |
| AU (1) | AU2022282786A1 (https=) |
| BR (1) | BR112023024311A2 (https=) |
| CA (1) | CA3219888A1 (https=) |
| IL (1) | IL308659A (https=) |
| MX (1) | MX2023013975A (https=) |
| TW (1) | TW202313598A (https=) |
| WO (1) | WO2022250108A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US11760747B2 (en) | 2020-12-21 | 2023-09-19 | Alkermes, Inc. | Substituted piperidino compounds and related methods of treatment |
| US12006330B2 (en) | 2020-12-21 | 2024-06-11 | Alkermes, Inc. | Substituted macrocyclic compounds and related methods of treatment |
| CA3248959A1 (en) * | 2022-04-22 | 2025-02-03 | Sumitomo Pharma Co., Ltd. | BICYCLOAMINE CARBOXAMIDE DERIVATIVE |
| WO2025010314A1 (en) * | 2023-07-05 | 2025-01-09 | Vertex Pharmaceuticals Incorporated | Urea-containing agonists of orexin receptor type 2 |
| WO2025010311A1 (en) * | 2023-07-05 | 2025-01-09 | Vertex Pharmaceuticals Incorporated | Urea-containing agonists of orexin receptor type 2 |
| WO2025124698A1 (en) | 2023-12-12 | 2025-06-19 | Idorsia Pharmaceuticals Ltd | Aryl sulfone and sulfanone derivatives as orexin receptor modulators |
| TW202542165A (zh) | 2023-12-19 | 2025-11-01 | 瑞士商愛杜西亞製藥有限公司 | 大環食慾素激動劑 |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6331545B1 (en) * | 1998-12-18 | 2001-12-18 | Soo S. Ko | Heterocycyclic piperidines as modulators of chemokine receptor activity |
| DE69926806D1 (de) * | 1998-12-18 | 2005-09-22 | Bristol Myers Squibb Pharma Co | N-ureidoalkylpiperidine als modulatoren der aktivität der chemokinrezeptoren |
| ES2300376T3 (es) * | 2000-10-27 | 2008-06-16 | Ortho-Mcneil Pharmaceutical, Inc. | Nuevas benzimidazol-2-onas sustituidas utilizadas como antagonistas del receptor de la vasopresina y como moduladores del neuropeptido y. |
| EA006507B1 (ru) * | 2001-10-15 | 2005-12-29 | Янссен Фармацевтика Н.В. | Новые замещенные 4-фенил-4-[1h-имидазол-2-ил] пиперидиновые производные и их применение в качестве селективных непептидных агонистов дельта-опиоидов |
| TW200418466A (en) * | 2002-11-06 | 2004-10-01 | Smithkline Beecham Corp | Chemical compounds |
| WO2006007864A1 (en) * | 2004-07-17 | 2006-01-26 | Max Planck Geselllschaft Zur Förderung Der Wissenschaft | Treating neurodegenerative conditions |
| WO2006127550A1 (en) * | 2005-05-23 | 2006-11-30 | Merck & Co., Inc. | Proline bis-amide orexin receptor antagonists |
| JP2009506061A (ja) * | 2005-08-26 | 2009-02-12 | メルク エンド カムパニー インコーポレーテッド | ジアザスピロデカンオレキシン受容体拮抗薬 |
| MX2009002920A (es) * | 2006-09-15 | 2009-04-01 | Schering Corp | Tratamiento del dolor, diabetes y trastornos del metabolismo de los lipidos. |
| WO2008098859A1 (en) * | 2007-02-15 | 2008-08-21 | F. Hoffmann-La Roche Ag | Hcv polymerase inhibitors |
| GB0813740D0 (en) * | 2008-07-28 | 2008-09-03 | Angeletti P Ist Richerche Biologica | Therapeutic compounds |
| JP2010155827A (ja) * | 2008-12-04 | 2010-07-15 | Takeda Chem Ind Ltd | スピロ環化合物 |
| CA2863413A1 (en) * | 2012-02-07 | 2013-08-15 | Eolas Therapeutics, Inc. | Substituted prolines / piperidines as orexin receptor antagonists |
| PL3411358T3 (pl) | 2016-02-04 | 2022-02-28 | Takeda Pharmaceutical Company Limited | Podstawiony związek piperydynowy i jego zastosowanie |
| US12048703B2 (en) * | 2018-04-13 | 2024-07-30 | University Of North Dakota | Use of small molecule FAK activators to promote mucosal healing |
| US20240024333A1 (en) * | 2020-10-26 | 2024-01-25 | Regents Of The University Of Minnesota | Use of small molecule fak activators to promote mucosal healing |
-
2022
- 2022-05-26 CA CA3219888A patent/CA3219888A1/en active Pending
- 2022-05-26 MX MX2023013975A patent/MX2023013975A/es unknown
- 2022-05-26 BR BR112023024311A patent/BR112023024311A2/pt unknown
- 2022-05-26 US US18/563,776 patent/US20240308960A1/en active Pending
- 2022-05-26 IL IL308659A patent/IL308659A/en unknown
- 2022-05-26 JP JP2023524226A patent/JPWO2022250108A1/ja active Pending
- 2022-05-26 AU AU2022282786A patent/AU2022282786A1/en active Pending
- 2022-05-26 EP EP22811378.3A patent/EP4353309A4/en active Pending
- 2022-05-26 TW TW111119648A patent/TW202313598A/zh unknown
- 2022-05-26 WO PCT/JP2022/021531 patent/WO2022250108A1/ja not_active Ceased
- 2022-05-26 CN CN202280037665.2A patent/CN117561238A/zh active Pending
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