JPWO2022145444A1 - - Google Patents
Info
- Publication number
- JPWO2022145444A1 JPWO2022145444A1 JP2022573099A JP2022573099A JPWO2022145444A1 JP WO2022145444 A1 JPWO2022145444 A1 JP WO2022145444A1 JP 2022573099 A JP2022573099 A JP 2022573099A JP 2022573099 A JP2022573099 A JP 2022573099A JP WO2022145444 A1 JPWO2022145444 A1 JP WO2022145444A1
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
- C07K1/042—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers characterised by the nature of the carrier
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
- C07K1/062—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for alpha- or omega-carboxy functions
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Analytical Chemistry (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020218595 | 2020-12-28 | ||
| PCT/JP2021/048743 WO2022145444A1 (ja) | 2020-12-28 | 2021-12-28 | アミノ酸の固相合成用樹脂への担持方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2022145444A1 true JPWO2022145444A1 (https=) | 2022-07-07 |
| JPWO2022145444A5 JPWO2022145444A5 (https=) | 2024-12-11 |
Family
ID=82260759
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022573099A Pending JPWO2022145444A1 (https=) | 2020-12-28 | 2021-12-28 |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20240067674A1 (https=) |
| EP (1) | EP4249496A4 (https=) |
| JP (1) | JPWO2022145444A1 (https=) |
| KR (1) | KR20230125807A (https=) |
| CN (1) | CN116547295A (https=) |
| WO (1) | WO2022145444A1 (https=) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW202446781A (zh) | 2011-12-28 | 2024-12-01 | 日商中外製藥股份有限公司 | 胜肽化合物之製造方法 |
| KR20250007021A (ko) | 2017-06-09 | 2025-01-13 | 추가이 세이야쿠 가부시키가이샤 | N-치환 아미노산을 포함하는 펩타이드의 합성 방법 |
| EP3878836B1 (en) | 2018-11-07 | 2025-07-23 | Chugai Seiyaku Kabushiki Kaisha | O-substituted serine derivative production method |
| EP3939962A4 (en) | 2019-03-15 | 2022-12-28 | Chugai Seiyaku Kabushiki Kaisha | PROCESS FOR PREPARING AN AROMATIC AMINO ACID DERIVATIVE |
| BR112022007535A2 (pt) | 2019-11-07 | 2022-07-12 | Chugai Pharmaceutical Co Ltd | Composto peptídico cíclico tendo ação inibitória de kras |
| EP4056580A4 (en) | 2019-11-07 | 2023-12-06 | Chugai Seiyaku Kabushiki Kaisha | METHOD FOR PRODUCING A PEPTIDE COMPOUND COMPRISING A STERICALLY HINDERED AMINO ACID |
| US12312379B2 (en) | 2021-05-07 | 2025-05-27 | Chugai Seiyaku Kabushiki Kaisha | Methods for producing cyclic compounds comprising N-substituted amino acid residues |
| JP7823181B2 (ja) | 2022-05-06 | 2026-03-03 | 中外製薬株式会社 | Ｈｒａｓおよびｎｒａｓに対して選択的なｋｒａｓ阻害作用を有する環状化合物 |
| JPWO2024096023A1 (https=) | 2022-11-01 | 2024-05-10 | ||
| WO2024143514A1 (ja) | 2022-12-28 | 2024-07-04 | 中外製薬株式会社 | 環状ペプチドの精製法及び製造法 |
| TW202523345A (zh) | 2023-09-28 | 2025-06-16 | 日商中外製藥股份有限公司 | 使用混合酸酐法的胜肽化合物的製造方法 |
| TW202535901A (zh) | 2023-12-27 | 2025-09-16 | 日商中外製藥股份有限公司 | 使用獨立型縮合劑的胜肽化合物的製造方法 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102643330A (zh) * | 2011-07-09 | 2012-08-22 | 广东医学院 | 一种骨靶向药物天冬氨酸六肽丹参素的合成方法及其医疗用途 |
| JP2013533264A (ja) * | 2010-07-22 | 2013-08-22 | ノヴォ・ノルディスク・ヘルス・ケア・アーゲー | 成長ホルモンコンジュゲート |
| WO2018225851A1 (ja) * | 2017-06-09 | 2018-12-13 | 中外製薬株式会社 | Ｎ－置換アミノ酸を含むペプチドの合成方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1648921A2 (en) * | 2003-06-26 | 2006-04-26 | Carlsberg A/S | Libraries containing heterocyclic organic molecules prepared through intramolecular formation of n-acyliminium ions |
| US20140213759A1 (en) * | 2011-06-16 | 2014-07-31 | Lonza Braine S.A. | Process For Extraction Of Peptides And Its Application In Liquid Phase Peptide Synthesis |
| TW202446781A (zh) | 2011-12-28 | 2024-12-01 | 日商中外製藥股份有限公司 | 胜肽化合物之製造方法 |
| GB201622029D0 (en) | 2016-12-22 | 2017-02-08 | Nederlands Inst Voor Ecologie (Nioo-Knaw) See Scientia Terrae Vzw Nordic Semiconductor Asa | Voltage sampling circuits |
| CN110869544B (zh) | 2017-06-09 | 2024-03-08 | 中外制药株式会社 | 膜透过性高的环状肽化合物及包含其的文库 |
| WO2020111238A1 (ja) | 2018-11-30 | 2020-06-04 | 中外製薬株式会社 | ペプチド化合物、またはアミド化合物の脱保護法および固相反応における脱樹脂方法、並びにペプチド化合物の製造方法 |
| WO2020122182A1 (ja) | 2018-12-12 | 2020-06-18 | 中外製薬株式会社 | 分子内水素結合可能な官能基を有するアミノ酸とそれらのアミノ酸を含むペプチド化合物、およびそれらの製造方法 |
-
2021
- 2021-12-28 CN CN202180083338.6A patent/CN116547295A/zh active Pending
- 2021-12-28 JP JP2022573099A patent/JPWO2022145444A1/ja active Pending
- 2021-12-28 WO PCT/JP2021/048743 patent/WO2022145444A1/ja not_active Ceased
- 2021-12-28 EP EP21915302.0A patent/EP4249496A4/en active Pending
- 2021-12-28 KR KR1020237024024A patent/KR20230125807A/ko active Pending
- 2021-12-28 US US18/269,334 patent/US20240067674A1/en active Pending
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013533264A (ja) * | 2010-07-22 | 2013-08-22 | ノヴォ・ノルディスク・ヘルス・ケア・アーゲー | 成長ホルモンコンジュゲート |
| CN102643330A (zh) * | 2011-07-09 | 2012-08-22 | 广东医学院 | 一种骨靶向药物天冬氨酸六肽丹参素的合成方法及其医疗用途 |
| WO2018225851A1 (ja) * | 2017-06-09 | 2018-12-13 | 中外製薬株式会社 | Ｎ－置換アミノ酸を含むペプチドの合成方法 |
Non-Patent Citations (1)
| Title |
|---|
| JAD, Y. E. ET AL.: "2-Methyltetrahydrofuran and cyclopentyl methyl ether for green solid-phase peptide synthesis", AMINO ACIDS, vol. 48, JPN6022004372, 2016, pages 419 - 426, ISSN: 0005787207 * |
Also Published As
| Publication number | Publication date |
|---|---|
| KR20230125807A (ko) | 2023-08-29 |
| WO2022145444A1 (ja) | 2022-07-07 |
| US20240067674A1 (en) | 2024-02-29 |
| EP4249496A1 (en) | 2023-09-27 |
| EP4249496A4 (en) | 2024-11-13 |
| TW202241921A (zh) | 2022-11-01 |
| CN116547295A (zh) | 2023-08-04 |
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