JPWO2021097009A5 - - Google Patents

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Publication number
JPWO2021097009A5
JPWO2021097009A5 JP2022527989A JP2022527989A JPWO2021097009A5 JP WO2021097009 A5 JPWO2021097009 A5 JP WO2021097009A5 JP 2022527989 A JP2022527989 A JP 2022527989A JP 2022527989 A JP2022527989 A JP 2022527989A JP WO2021097009 A5 JPWO2021097009 A5 JP WO2021097009A5
Authority
JP
Japan
Prior art keywords
methyl
oxy
pyridin
dichlorophenyl
piperidin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022527989A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023503852A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/060108 external-priority patent/WO2021097009A1/en
Publication of JP2023503852A publication Critical patent/JP2023503852A/ja
Publication of JPWO2021097009A5 publication Critical patent/JPWO2021097009A5/ja
Pending legal-status Critical Current

Links

JP2022527989A 2019-11-12 2020-11-12 感染症を処置するための低分子フーリン阻害剤 Pending JP2023503852A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201962934407P 2019-11-12 2019-11-12
US62/934,407 2019-11-12
PCT/US2020/060108 WO2021097009A1 (en) 2019-11-12 2020-11-12 Small molecule furin inhibitors for treating infectious diseases

Publications (2)

Publication Number Publication Date
JP2023503852A JP2023503852A (ja) 2023-02-01
JPWO2021097009A5 true JPWO2021097009A5 (enExample) 2023-11-20

Family

ID=73793799

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022527989A Pending JP2023503852A (ja) 2019-11-12 2020-11-12 感染症を処置するための低分子フーリン阻害剤

Country Status (8)

Country Link
US (1) US20230011571A1 (enExample)
EP (1) EP4058021A1 (enExample)
JP (1) JP2023503852A (enExample)
KR (1) KR20220104744A (enExample)
CN (1) CN114929220A (enExample)
AU (1) AU2020382819A1 (enExample)
CA (1) CA3157892A1 (enExample)
WO (1) WO2021097009A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2019267166C1 (en) 2018-05-11 2023-11-30 Glaxosmithkline Intellectual Property Development Limited Furin inhibitors
DE102023126563A1 (de) 2023-09-28 2025-04-03 Philipps-Universität Marburg, Körperschaft des öffentlichen Rechts Hemmstoffe der Proproteinkonvertase Furin, Verfahren zu deren Herstellung und Verwendung

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003037346A1 (en) * 2001-10-31 2003-05-08 Cell Therapeutics, Inc. 6-phenyl-n-phenyl-(1,3,5) -triazine-2,4-diamine derivatives and related compounds with lysophphosphatidic acid acyltransferase beta (lpaat-beta) inhibitory activity for use in the treatment of cancer
WO2009023306A2 (en) 2007-05-09 2009-02-19 Burnham Institute For Medical Research Targeting host proteinases as a therapeutic strategy against viral and bacterial pathogens
WO2013138666A1 (en) 2012-03-16 2013-09-19 Sanford-Burnham Medical Research Institute Inhibitors of furin and other pro-protein convertases
WO2014152716A1 (en) * 2013-03-15 2014-09-25 President And Fellows Of Harvard College Substituted heterocyclic compounds for treating or preventing viral infections
CN107441094B (zh) * 2017-08-08 2020-05-22 南方医科大学 尼罗替尼作为治疗登革病毒感染的药物及其制药用途
AU2019267166C1 (en) * 2018-05-11 2023-11-30 Glaxosmithkline Intellectual Property Development Limited Furin inhibitors

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