JPWO2021076514A5 - - Google Patents

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Publication number
JPWO2021076514A5
JPWO2021076514A5 JP2022521584A JP2022521584A JPWO2021076514A5 JP WO2021076514 A5 JPWO2021076514 A5 JP WO2021076514A5 JP 2022521584 A JP2022521584 A JP 2022521584A JP 2022521584 A JP2022521584 A JP 2022521584A JP WO2021076514 A5 JPWO2021076514 A5 JP WO2021076514A5
Authority
JP
Japan
Prior art keywords
compound
use according
treatment period
platelet count
itp
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022521584A
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English (en)
Japanese (ja)
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JP2022550919A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2020/055410 external-priority patent/WO2021076514A1/fr
Publication of JP2022550919A publication Critical patent/JP2022550919A/ja
Publication of JPWO2021076514A5 publication Critical patent/JPWO2021076514A5/ja
Pending legal-status Critical Current

Links

JP2022521584A 2019-10-14 2020-10-13 (r)-2-[3-[4-アミノ-3-(2-フルオロ-4-フェノキシ-フェニル)ピラゾロ[3,4-d]ピリミジン-1-イル]ピペリジン-1-カルボニル]-4-メチル-4-[4-(オキセタン-3-イル)ピペラジン-1-イル]ペンタ-2-エンニトリルを投与することにより免疫性血小板減少症を治療する方法 Pending JP2022550919A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201962914688P 2019-10-14 2019-10-14
US62/914,688 2019-10-14
US201962951302P 2019-12-20 2019-12-20
US62/951,302 2019-12-20
PCT/US2020/055410 WO2021076514A1 (fr) 2019-10-14 2020-10-13 Procédé de traitement de la thrombocytopénie immunitaire par l'administration de (r)-2-[3-[4-amino-3-(2-fluoro-4-phénoxy-phényl)pyrazolo[3,4-d]pyrimidine-1-yl]pipéridine-1-carbonyle]-4-méthyl-4-[4-(oxétane-3-yl)pipérazine-1-yl]pent-2-ènenitrile

Publications (2)

Publication Number Publication Date
JP2022550919A JP2022550919A (ja) 2022-12-05
JPWO2021076514A5 true JPWO2021076514A5 (fr) 2023-10-20

Family

ID=73040359

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022521584A Pending JP2022550919A (ja) 2019-10-14 2020-10-13 (r)-2-[3-[4-アミノ-3-(2-フルオロ-4-フェノキシ-フェニル)ピラゾロ[3,4-d]ピリミジン-1-イル]ピペリジン-1-カルボニル]-4-メチル-4-[4-(オキセタン-3-イル)ピペラジン-1-イル]ペンタ-2-エンニトリルを投与することにより免疫性血小板減少症を治療する方法

Country Status (12)

Country Link
US (2) US20210106584A1 (fr)
EP (1) EP4045051A1 (fr)
JP (1) JP2022550919A (fr)
KR (1) KR20220080179A (fr)
CN (1) CN115209899A (fr)
AU (1) AU2020365951A1 (fr)
CA (1) CA3154257A1 (fr)
CO (1) CO2022006087A2 (fr)
IL (1) IL291994A (fr)
MX (1) MX2022004427A (fr)
TW (1) TW202128175A (fr)
WO (1) WO2021076514A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202308638A (zh) * 2021-04-16 2023-03-01 美商普林斯匹亞生物製藥公司 藉由投予特定化合物治療藥物及疫苗誘發的免疫性血小板減少症之方法
WO2024097667A1 (fr) * 2022-10-31 2024-05-10 Principia Biopharma Inc. Méthodes de traitement de thrombocytopénie immunitaire par administration de (r)-2-[3- [4-amino-3-(2-fluoro-4-phénoxy-phényl)pyrazolo[3,4-d]pyrimidin-l-yl]pipéridine-l-carbonyl]-4-méthyl-4-[4-(oxétan-3-yl)pipérazin-l-yl]pent-2-ènenitrile

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2731833T3 (es) 2012-09-10 2019-11-19 Principia Biopharma Inc Compuestos pirazolopirimidínicos comos inhibidores de cinasas
US10092569B2 (en) 2014-02-21 2018-10-09 Principia Biopharma Inc. Salts and solid form of a BTK inhibitor
MX2017007973A (es) 2014-12-18 2018-02-09 Principia Biopharma Inc Tratamiento de penfigo.
CN107427468B (zh) 2014-12-24 2022-02-25 普林斯匹亚生物制药公司 Btk抑制剂的部位特异性给药
AU2017290354C1 (en) 2016-06-29 2023-07-06 Principia Biopharma Inc. Modified release formulations of 2-[3-[4-amino-3-(2-fluoro-4-phenoxy-phenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl]-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile

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