JPWO2021071812A5 - - Google Patents
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- JPWO2021071812A5 JPWO2021071812A5 JP2022546590A JP2022546590A JPWO2021071812A5 JP WO2021071812 A5 JPWO2021071812 A5 JP WO2021071812A5 JP 2022546590 A JP2022546590 A JP 2022546590A JP 2022546590 A JP2022546590 A JP 2022546590A JP WO2021071812 A5 JPWO2021071812 A5 JP WO2021071812A5
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- JP
- Japan
- Prior art keywords
- cr6r7
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- occurrence
- alkyl
- independently
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962911652P | 2019-10-07 | 2019-10-07 | |
| US62/911,652 | 2019-10-07 | ||
| PCT/US2020/054360 WO2021071812A1 (en) | 2019-10-07 | 2020-10-06 | Arylmethylene heterocyclic compounds as kv1.3 potassium shaker channel blockers |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| JP2022551198A JP2022551198A (ja) | 2022-12-07 |
| JP2022551198A5 JP2022551198A5 (https=) | 2024-05-15 |
| JPWO2021071812A5 true JPWO2021071812A5 (https=) | 2024-05-15 |
| JP7822940B2 JP7822940B2 (ja) | 2026-03-03 |
Family
ID=75436856
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022546590A Active JP7822940B2 (ja) | 2019-10-07 | 2020-10-06 | Ｋｖ１．３カリウムシェーカーチャネル遮断薬としてのアリールメチレン複素環式化合物 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US20220411367A1 (https=) |
| EP (1) | EP4041228A4 (https=) |
| JP (1) | JP7822940B2 (https=) |
| KR (1) | KR20220079881A (https=) |
| CN (1) | CN114727993B (https=) |
| AU (1) | AU2020363360A1 (https=) |
| BR (1) | BR112022006226A2 (https=) |
| CA (1) | CA3157031A1 (https=) |
| IL (1) | IL291869A (https=) |
| MX (1) | MX2022004145A (https=) |
| WO (1) | WO2021071812A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN116782894A (zh) * | 2020-10-06 | 2023-09-19 | D.E.肖研究有限责任公司 | 作为Kv1.3钾Shaker通道阻断剂的内酰胺化合物 |
| WO2025029769A1 (en) | 2023-07-31 | 2025-02-06 | Eli Lilly And Company | Solid forms of a kv1.3 potassium shaker channel blockers and method of using the same |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PL208928B1 (pl) * | 2001-04-16 | 2011-06-30 | Pharmacopeia | 3, 4-di-podstawione cyklobuten-1, 2-diony jako ligandy receptora CXC chemokiny |
| WO2008115118A1 (en) * | 2007-03-21 | 2008-09-25 | Innate Pharmaceuticals Ab | Method and means for preventing and inhibiting type iii secretion in infections caused by gram-negative bacteria |
| TW201026708A (en) | 2008-12-12 | 2010-07-16 | Solvay Pharm Bv | Spiro azepane-oxazolidinones as Kv1.3 potassium channel blockers |
| WO2013056153A1 (en) | 2011-10-13 | 2013-04-18 | Kung Charles | Activators of pyruvate kinase m2 and methods of treating disease |
| CA2969295A1 (en) | 2016-06-06 | 2017-12-06 | Pfizer Inc. | Substituted carbonucleoside derivatives, and use thereof as a prmt5 inhibitor |
| AU2017367086A1 (en) * | 2016-11-29 | 2019-07-18 | Epizyme, Inc. | Compounds containing a sulfonic group as KAT inhibitors |
| US11529338B2 (en) * | 2017-08-22 | 2022-12-20 | Cedars-Sinai Medical Center | Compositions and methods for treating cancer |
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2020
- 2020-10-06 JP JP2022546590A patent/JP7822940B2/ja active Active
- 2020-10-06 CN CN202080084714.9A patent/CN114727993B/zh active Active
- 2020-10-06 MX MX2022004145A patent/MX2022004145A/es unknown
- 2020-10-06 BR BR112022006226A patent/BR112022006226A2/pt not_active IP Right Cessation
- 2020-10-06 KR KR1020227013512A patent/KR20220079881A/ko not_active Withdrawn
- 2020-10-06 EP EP20874457.3A patent/EP4041228A4/en active Pending
- 2020-10-06 AU AU2020363360A patent/AU2020363360A1/en not_active Abandoned
- 2020-10-06 US US17/766,889 patent/US20220411367A1/en active Pending
- 2020-10-06 IL IL291869A patent/IL291869A/en unknown
- 2020-10-06 CA CA3157031A patent/CA3157031A1/en active Pending
- 2020-10-06 WO PCT/US2020/054360 patent/WO2021071812A1/en not_active Ceased