JPWO2020210485A5 - - Google Patents
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- Publication number
- JPWO2020210485A5 JPWO2020210485A5 JP2021559848A JP2021559848A JPWO2020210485A5 JP WO2020210485 A5 JPWO2020210485 A5 JP WO2020210485A5 JP 2021559848 A JP2021559848 A JP 2021559848A JP 2021559848 A JP2021559848 A JP 2021559848A JP WO2020210485 A5 JPWO2020210485 A5 JP WO2020210485A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- compound
- protecting group
- group
- nitrogen protecting
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201962831962P | 2019-04-10 | 2019-04-10 | |
| US62/831,962 | 2019-04-10 | ||
| PCT/US2020/027459 WO2020210485A1 (fr) | 2019-04-10 | 2020-04-09 | Procédé de préparation de dérivés de pyrrolidine alpha-carboxamide |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2022527213A JP2022527213A (ja) | 2022-05-31 |
| JPWO2020210485A5 true JPWO2020210485A5 (fr) | 2023-05-17 |
Family
ID=72750576
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021559848A Withdrawn JP2022527213A (ja) | 2019-04-10 | 2020-04-09 | アルファ－カルボキサミドピロリジン誘導体を調製するためのプロセス |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20220177426A1 (fr) |
| EP (1) | EP3953329A4 (fr) |
| JP (1) | JP2022527213A (fr) |
| KR (1) | KR20210150527A (fr) |
| CN (1) | CN114026066A (fr) |
| AU (1) | AU2020271856A1 (fr) |
| BR (1) | BR112021020345A2 (fr) |
| CA (1) | CA3136536A1 (fr) |
| EA (1) | EA202192762A1 (fr) |
| IL (1) | IL287078A (fr) |
| MX (1) | MX2021012420A (fr) |
| WO (1) | WO2020210485A1 (fr) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112153968A (zh) | 2017-10-05 | 2020-12-29 | 生物基因公司 | 制备α-羧酰胺吡咯烷衍生物的工艺 |
| CN112812048B (zh) * | 2021-01-20 | 2022-08-26 | 北京蓝博特科技有限公司 | 一种钠离子通道阻滞剂cnv1014802盐酸盐形态的制备方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3164597A (en) * | 1962-12-17 | 1965-01-05 | Geigy Chem Corp | 5-carboxylic acid-2-phenyl-pyrrolines, corresponding pyrrolidines and functional derivatives thereof |
| TW200730494A (en) * | 2005-10-10 | 2007-08-16 | Glaxo Group Ltd | Novel compounds |
| WO2008090117A1 (fr) * | 2007-01-24 | 2008-07-31 | Glaxo Group Limited | Nouvelles compositions pharmaceutiques |
| WO2016102967A1 (fr) * | 2014-12-23 | 2016-06-30 | Convergence Pharmaceuticals Limited | Procédé de préparation de dérivés d'alpha-carboxamide de pyrrolidine |
| WO2016160574A2 (fr) * | 2015-03-27 | 2016-10-06 | Scifluor Life Sciences, Inc. | Composés d'aryl-et hétéroaryl-pyrrolidine-2-carboxamide |
-
2020
- 2020-04-09 AU AU2020271856A patent/AU2020271856A1/en not_active Withdrawn
- 2020-04-09 EA EA202192762A patent/EA202192762A1/ru unknown
- 2020-04-09 BR BR112021020345A patent/BR112021020345A2/pt not_active Application Discontinuation
- 2020-04-09 CN CN202080042335.3A patent/CN114026066A/zh not_active Withdrawn
- 2020-04-09 KR KR1020217036558A patent/KR20210150527A/ko unknown
- 2020-04-09 US US17/602,585 patent/US20220177426A1/en active Pending
- 2020-04-09 MX MX2021012420A patent/MX2021012420A/es unknown
- 2020-04-09 EP EP20788448.7A patent/EP3953329A4/fr not_active Withdrawn
- 2020-04-09 WO PCT/US2020/027459 patent/WO2020210485A1/fr unknown
- 2020-04-09 CA CA3136536A patent/CA3136536A1/fr not_active Withdrawn
- 2020-04-09 JP JP2021559848A patent/JP2022527213A/ja not_active Withdrawn
-
2021
- 2021-10-07 IL IL287078A patent/IL287078A/en unknown
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