JPWO2020195437A1 - - Google Patents

Info

Publication number
JPWO2020195437A1
JPWO2020195437A1 JP2021508823A JP2021508823A JPWO2020195437A1 JP WO2020195437 A1 JPWO2020195437 A1 JP WO2020195437A1 JP 2021508823 A JP2021508823 A JP 2021508823A JP 2021508823 A JP2021508823 A JP 2021508823A JP WO2020195437 A1 JPWO2020195437 A1 JP WO2020195437A1
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021508823A
Other languages
Japanese (ja)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of JPWO2020195437A1 publication Critical patent/JPWO2020195437A1/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C405/00—Compounds containing a five-membered ring having two side-chains in ortho position to each other, and having oxygen atoms directly attached to the ring in ortho position to one of the side-chains, one side-chain containing, not directly attached to the ring, a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, and the other side-chain having oxygen atoms attached in gamma-position to the ring, e.g. prostaglandins ; Analogues or derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B61/00—Other general methods
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/93—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems condensed with a ring other than six-membered
    • C07D307/935—Not further condensed cyclopenta [b] furans or hydrogenated cyclopenta [b] furans
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2021508823A 2019-03-27 2020-02-21 Pending JPWO2020195437A1 (enExample)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2019060295 2019-03-27
PCT/JP2020/007196 WO2020195437A1 (ja) 2019-03-27 2020-02-21 プロスタグランジンの製造方法

Publications (1)

Publication Number Publication Date
JPWO2020195437A1 true JPWO2020195437A1 (enExample) 2020-10-01

Family

ID=72609003

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021508823A Pending JPWO2020195437A1 (enExample) 2019-03-27 2020-02-21

Country Status (7)

Country Link
US (1) US20220169600A1 (enExample)
EP (1) EP3950672A4 (enExample)
JP (1) JPWO2020195437A1 (enExample)
CN (1) CN113557227A (enExample)
CA (1) CA3132572A1 (enExample)
TW (1) TWI838487B (enExample)
WO (1) WO2020195437A1 (enExample)

Citations (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS63174938A (ja) * 1987-01-13 1988-07-19 Toray Ind Inc 光学活性アリルアルコ−ル誘導体の製造方法
JP2005503354A (ja) * 2001-05-24 2005-02-03 レゾリューション ケミカルズ リミテッド プロスタグランジン及びそれらの類縁体の製法
JP2008037782A (ja) * 2006-08-04 2008-02-21 Daiichi Fine Chemical Co Ltd プロスタグランジン誘導体の製造方法
CA2557401A1 (en) * 2006-08-25 2008-02-25 Alphora Research Inc. Prostaglandin intermediates and their synthesis
JP2011246435A (ja) * 2010-04-28 2011-12-08 Takasago Internatl Corp 新規ルテニウム錯体及びこれを触媒とする光学活性アルコール化合物の製造方法
WO2012011128A1 (en) * 2010-07-23 2012-01-26 Aptuit Laurus Private Limited Preparation of prostaglandin derivatives
JP2015506343A (ja) * 2011-12-21 2015-03-02 キノイン・ジヨージセル・エーシユ・ベジエーセテイ・テルメーケク・ジヤーラ・ゼー・エル・テー トラボプロストの調製方法
WO2015133405A1 (ja) * 2014-03-06 2015-09-11 日産化学工業株式会社 光学活性アゼチジノン化合物の製造方法
CN109232494A (zh) * 2018-10-29 2019-01-18 常州博海威医药科技股份有限公司 一种比马前列腺素关键中间体的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3726983A (en) 1971-05-14 1973-04-10 Alza Corp Pharmaceutical compositions comprising tetrahydropyran-2{40 -yl prostaglandin ethers
US6248783B1 (en) 2000-09-20 2001-06-19 Allergan Sales, Inc. Cyclopentane 1-hydroxy alkyl or alkenyl-2-one or 2-hydroxy derivatives as therapeutic agents
US7511168B2 (en) 2006-01-18 2009-03-31 Shih-Yi Wei Processes and intermediates for the preparations of prostaglandins
JP4851467B2 (ja) 2006-02-07 2012-01-11 株式会社アールテック・ウエノ プロスタグランジン誘導体の製造法
CN101555221B (zh) 2008-04-09 2013-01-23 明德国际仓储贸易(上海)有限公司 一种前列腺素f型衍生物的制造方法
WO2014200094A1 (ja) * 2013-06-14 2014-12-18 日産化学工業株式会社 光学活性アルコール化合物の製造方法
US9115109B2 (en) 2013-08-15 2015-08-25 Chirogate International Inc. Processes and intermediates for the preparations of isomer free prostaglandins
CN105985371B (zh) 2015-02-11 2019-06-18 常州博海威医药科技股份有限公司 制备利马前列腺素的关键中间体及其应用
KR102754527B1 (ko) * 2017-05-30 2025-01-14 데이 원 바이오파마슈티칼즈, 인크. 광학 활성 화합물의 제조법

Patent Citations (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS63174938A (ja) * 1987-01-13 1988-07-19 Toray Ind Inc 光学活性アリルアルコ−ル誘導体の製造方法
JP2005503354A (ja) * 2001-05-24 2005-02-03 レゾリューション ケミカルズ リミテッド プロスタグランジン及びそれらの類縁体の製法
JP2008037782A (ja) * 2006-08-04 2008-02-21 Daiichi Fine Chemical Co Ltd プロスタグランジン誘導体の製造方法
CA2557401A1 (en) * 2006-08-25 2008-02-25 Alphora Research Inc. Prostaglandin intermediates and their synthesis
JP2011246435A (ja) * 2010-04-28 2011-12-08 Takasago Internatl Corp 新規ルテニウム錯体及びこれを触媒とする光学活性アルコール化合物の製造方法
WO2012011128A1 (en) * 2010-07-23 2012-01-26 Aptuit Laurus Private Limited Preparation of prostaglandin derivatives
JP2015506343A (ja) * 2011-12-21 2015-03-02 キノイン・ジヨージセル・エーシユ・ベジエーセテイ・テルメーケク・ジヤーラ・ゼー・エル・テー トラボプロストの調製方法
WO2015133405A1 (ja) * 2014-03-06 2015-09-11 日産化学工業株式会社 光学活性アゼチジノン化合物の製造方法
CN109232494A (zh) * 2018-10-29 2019-01-18 常州博海威医药科技股份有限公司 一种比马前列腺素关键中间体的制备方法

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
CHANDRSEKHAR, S. ET AL.: "One Pot Conversion of Carboxylic Acids to Aldehydes with DIBAL-H", TETRAHEDRON LETTERS, vol. 39, JPN6020001256, 1998, pages 909 - 910, ISSN: 0005243364 *
MATSUMURA, K. ET AL.: "Chiral Ruthenabicyclic Complexes: Precatalysts for Rapid, Enantioselective, and Wide-Scope Hydrogena", J. AM. CHEM. SOC., vol. 133, JPN6020016096, 2011, pages 10696 - 10699, ISSN: 0005243363 *
NORRIS, M. D. ET AL.: "Biomimetic Total Synthesis of Gracilioethers B and C", ORG. LETT., vol. 17, JPN6020016097, 2015, pages 668 - 671, ISSN: 0005459396 *

Also Published As

Publication number Publication date
CA3132572A1 (en) 2020-10-01
TW202102472A (zh) 2021-01-16
TWI838487B (zh) 2024-04-11
KR20210143744A (ko) 2021-11-29
CN113557227A (zh) 2021-10-26
WO2020195437A1 (ja) 2020-10-01
US20220169600A1 (en) 2022-06-02
EP3950672A1 (en) 2022-02-09
EP3950672A4 (en) 2023-01-11

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