JPWO2019160980A5 - - Google Patents

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Publication number
JPWO2019160980A5
JPWO2019160980A5 JP2020543286A JP2020543286A JPWO2019160980A5 JP WO2019160980 A5 JPWO2019160980 A5 JP WO2019160980A5 JP 2020543286 A JP2020543286 A JP 2020543286A JP 2020543286 A JP2020543286 A JP 2020543286A JP WO2019160980 A5 JPWO2019160980 A5 JP WO2019160980A5
Authority
JP
Japan
Prior art keywords
compound according
alkyl
halo
cyano
bromine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2020543286A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021513547A5 (https=
JP2021513547A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/017881 external-priority patent/WO2019160980A1/en
Publication of JP2021513547A publication Critical patent/JP2021513547A/ja
Publication of JP2021513547A5 publication Critical patent/JP2021513547A5/ja
Publication of JPWO2019160980A5 publication Critical patent/JPWO2019160980A5/ja
Pending legal-status Critical Current

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JP2020543286A 2018-02-14 2019-02-13 ソベチロムの誘導体 Pending JP2021513547A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201862630775P 2018-02-14 2018-02-14
US62/630,775 2018-02-14
US201862631442P 2018-02-15 2018-02-15
US62/631,442 2018-02-15
PCT/US2019/017881 WO2019160980A1 (en) 2018-02-14 2019-02-13 Derivatives of sobetirome

Publications (3)

Publication Number Publication Date
JP2021513547A JP2021513547A (ja) 2021-05-27
JP2021513547A5 JP2021513547A5 (https=) 2022-02-17
JPWO2019160980A5 true JPWO2019160980A5 (https=) 2022-02-17

Family

ID=67619583

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020543286A Pending JP2021513547A (ja) 2018-02-14 2019-02-13 ソベチロムの誘導体

Country Status (11)

Country Link
US (1) US11578032B2 (https=)
EP (1) EP3752001A4 (https=)
JP (1) JP2021513547A (https=)
KR (1) KR20200120928A (https=)
CN (1) CN111818798A (https=)
AU (1) AU2019222709A1 (https=)
BR (1) BR112020016599A2 (https=)
CA (1) CA3091021A1 (https=)
IL (1) IL276592B2 (https=)
MX (1) MX2020008498A (https=)
WO (1) WO2019160980A1 (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3894383A1 (en) * 2018-12-12 2021-10-20 Autobahn Therapeutics, Inc. Novel thyromimetics
CA3130371A1 (en) 2019-03-01 2020-09-10 Autobahn Therapeutics, Inc. Novel thyromimetics
KR20220121239A (ko) 2019-11-29 2022-08-31 아우토반 쎄라퓨틱스, 인크. 신규한 갑상선 호르몬 모방제
WO2021247847A1 (en) * 2020-06-03 2021-12-09 Autobahn Therapeutics, Inc. Isotopic thyromimetic compounds
US20230242473A1 (en) * 2020-06-17 2023-08-03 Autobahn Therapeutics, Inc. Thyromimetics
JP7813730B2 (ja) 2020-06-17 2026-02-13 オートバーン セラピューティクス,インク. 甲状腺様作用剤
WO2021257851A1 (en) * 2020-06-17 2021-12-23 Autobahn Therapeutics, Inc. Thyromimetics
JP2024516852A (ja) * 2021-05-06 2024-04-17 オートバーン セラピューティクス,インク. 甲状腺ホルモン模倣薬の、脂肪酸アミド加水分解酵素(faah)により切断可能なプロドラッグ、および末梢制限faah阻害剤との組合せ

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5883294A (en) 1997-06-18 1999-03-16 The Regeants Of The University Of California Selective thyroid hormone analogs
US6436990B1 (en) * 1999-10-27 2002-08-20 Nobex Corporation 6-methoxy-2-naphthylacetic acid prodrugs
US6429223B1 (en) * 2000-06-23 2002-08-06 Medinox, Inc. Modified forms of pharmacologically active agents and uses therefor
WO2006128058A2 (en) * 2005-05-26 2006-11-30 Metabasis Therapeutics, Inc. Thyromimetics for the treatment of fatty liver diseases
WO2006128056A2 (en) 2005-05-26 2006-11-30 Metabasis Therapeutics, Inc. Novel phosphinic acid-containing thyromimetics
EP3259246B1 (en) * 2015-02-20 2023-03-22 Oregon Health & Science University Derivatives of sobetirome
US10532983B2 (en) 2015-07-20 2020-01-14 Oregon Health & Science University Quinolone-3-diarylethers
CN109475121B (zh) * 2016-05-18 2021-06-25 俄勒冈健康科学大学 苏比替罗衍生物
US11325886B2 (en) * 2016-08-12 2022-05-10 Oregon Health & Science University Amide compounds, pharmaceutical compositions thereof, and methods of using the same

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