JPS6363682A - ２―（１―オキソ―１―イミノ―１―チアシクロアルキル）―チオペネム誘導体および組成物 - Google Patents

２―（１―オキソ―１―イミノ―１―チアシクロアルキル）―チオペネム誘導体および組成物

Info

Publication number
JPS6363682A
JPS6363682A JP62221811A JP22181187A JPS6363682A JP S6363682 A JPS6363682 A JP S6363682A JP 62221811 A JP62221811 A JP 62221811A JP 22181187 A JP22181187 A JP 22181187A JP S6363682 A JPS6363682 A JP S6363682A
Authority
JP
Japan
Prior art keywords
oxo
compound
formula
imino
cis
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP62221811A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0529356B2 (https=
Inventor
アーネスト・セイイチ・ハマナカ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of JPS6363682A publication Critical patent/JPS6363682A/ja
Publication of JPH0529356B2 publication Critical patent/JPH0529356B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
JP62221811A 1986-09-04 1987-09-04 ２―（１―オキソ―１―イミノ―１―チアシクロアルキル）―チオペネム誘導体および組成物 Granted JPS6363682A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8601813 1986-09-04
WO86/01813 1986-09-04

Publications (2)

Publication Number Publication Date
JPS6363682A true JPS6363682A (ja) 1988-03-22
JPH0529356B2 JPH0529356B2 (https=) 1993-04-30

Family

ID=22195624

Family Applications (1)

Application Number Title Priority Date Filing Date
JP62221811A Granted JPS6363682A (ja) 1986-09-04 1987-09-04 ２―（１―オキソ―１―イミノ―１―チアシクロアルキル）―チオペネム誘導体および組成物

Country Status (7)

Country Link
EP (1) EP0260042B1 (https=)
JP (1) JPS6363682A (https=)
AT (1) ATE70841T1 (https=)
DE (1) DE3775504D1 (https=)
DK (1) DK459087A (https=)
IE (1) IE60293B1 (https=)
PT (1) PT85645B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX20084A (es) * 1989-03-28 1993-03-01 Pfizer Derivados de 2 -carbapenem antibacterianos
US5321020A (en) * 1989-03-28 1994-06-14 Pfizer Inc. Antibacterial 2-carbapenem derivatives
WO2017162661A1 (en) 2016-03-22 2017-09-28 Bayer Pharma Aktiengesellschaft 1h-benzo[de]isoquinoline-1,3(2h)-diones

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0130025B1 (en) * 1983-06-21 1987-07-08 Pfizer Inc. 2-alkylthiopenem derivatives

Also Published As

Publication number Publication date
PT85645A (en) 1987-10-01
PT85645B (pt) 1991-02-08
IE872365L (en) 1988-03-04
DK459087A (da) 1988-03-05
EP0260042A1 (en) 1988-03-16
DE3775504D1 (en) 1992-02-06
DK459087D0 (da) 1987-09-03
EP0260042B1 (en) 1991-12-27
ATE70841T1 (de) 1992-01-15
JPH0529356B2 (https=) 1993-04-30
IE60293B1 (en) 1994-06-29

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