JPS6254786B2 - - Google Patents

Info

Publication number
JPS6254786B2
JPS6254786B2 JP59105654A JP10565484A JPS6254786B2 JP S6254786 B2 JPS6254786 B2 JP S6254786B2 JP 59105654 A JP59105654 A JP 59105654A JP 10565484 A JP10565484 A JP 10565484A JP S6254786 B2 JPS6254786 B2 JP S6254786B2
Authority
JP
Japan
Prior art keywords
carbomethoxyaminobenzimidazole
mixture
chloroform
methanol
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP59105654A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6023371A (ja
Inventor
Shii Biado Koorin
Ei Edowaazu Jon
Eichi Furaido Jon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Syntex USA LLC
Original Assignee
Syntex USA LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex USA LLC filed Critical Syntex USA LLC
Publication of JPS6023371A publication Critical patent/JPS6023371A/ja
Publication of JPS6254786B2 publication Critical patent/JPS6254786B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/30—Isothioureas
    • C07C335/38—Isothioureas containing any of the groups, X being a hetero atom, Y being any atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30—Nitrogen atoms not forming part of a nitro radical
    • C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
JP59105654A 1972-12-29 1984-05-24 駆虫効果を有するカルバメ−ト誘導体の製造方法 Granted JPS6023371A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US31929972A 1972-12-29 1972-12-29
US319299 1972-12-29
US417963 1973-11-21

Publications (2)

Publication Number Publication Date
JPS6023371A JPS6023371A (ja) 1985-02-05
JPS6254786B2 true JPS6254786B2 (enExample) 1987-11-17

Family

ID=23241674

Family Applications (2)

Application Number Title Priority Date Filing Date
JP10631880A Granted JPS5639016A (en) 1972-12-29 1980-08-01 Veterinary vermifuge composition
JP59105654A Granted JPS6023371A (ja) 1972-12-29 1984-05-24 駆虫効果を有するカルバメ−ト誘導体の製造方法

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP10631880A Granted JPS5639016A (en) 1972-12-29 1980-08-01 Veterinary vermifuge composition

Country Status (5)

Country Link
JP (2) JPS5639016A (enExample)
BE (2) BE809235A (enExample)
DD (1) DD112450A5 (enExample)
PL (1) PL99587B1 (enExample)
ZA (2) ZA739219B (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4002640A (en) * 1972-12-29 1977-01-11 Syntex (U.S.A.) Inc. 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity
US3993769A (en) * 1972-12-29 1976-11-23 Syntex (U.S.A.) Inc. 1,5(6)-Disubstituted benzimidazole-2-carbamate derivatives having anthelmintic activity
US4258198A (en) * 1973-05-29 1981-03-24 Smithkline Corporation 5-Cycloalkyl thio- and oxy-2-carbalkoxyaminobenzimidazoles
DE2518188A1 (de) * 1974-05-02 1975-11-20 Chinoin Gyogyszer Es Vegyeszet Neue benzimidazolderivate
DE2441201C2 (de) * 1974-08-28 1986-08-07 Hoechst Ag, 6230 Frankfurt Anthelminthisch wirksame 2-Carbalkoxyamino-5(6)-phenyl-sulfonyloxy-benzimidazole und Verfahren zu ihrer Herstellung
DE2441202C2 (de) * 1974-08-28 1986-05-28 Hoechst Ag, 6230 Frankfurt 2-Carbalkoxyamino-benzimidazolyl-5(6)-sulfonsäure-phenylester, Verfahren zu ihrer Herstellung und diese enthaltende anthelmintische Mittel
US4025638A (en) * 1975-03-10 1977-05-24 Smithkline Corporation Methods and compositions using 5-cycloalkylthio- and oxy-2-carbalkoxy-aminobenzimidazole
US4093732A (en) * 1977-02-17 1978-06-06 E. R. Squibb & Sons, Inc. Sulfoxide derivatives of benzimidazoles
JPS63154063U (enExample) * 1987-03-31 1988-10-11
EP2606726A1 (de) * 2011-12-21 2013-06-26 Bayer CropScience AG N-Arylamidine-substituierte trifluoroethylsulfid-Derivate als Akarizide und Insektizide

Also Published As

Publication number Publication date
ZA739219B (en) 1975-07-30
JPS5639016A (en) 1981-04-14
PL99587B1 (pl) 1978-07-31
ZA739220B (en) 1975-07-30
DD112450A5 (enExample) 1975-04-12
JPS6023371A (ja) 1985-02-05
BE809235A (fr) 1974-06-28
BE809234A (fr) 1974-06-28
JPS624365B2 (enExample) 1987-01-30

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