JPS5982375A - ６−アニリノ−５，８−キノキサリンジオン類 - Google Patents

６−アニリノ−５，８−キノキサリンジオン類

Info

Publication number
JPS5982375A
JPS5982375A JP58182918A JP18291883A JPS5982375A JP S5982375 A JPS5982375 A JP S5982375A JP 58182918 A JP58182918 A JP 58182918A JP 18291883 A JP18291883 A JP 18291883A JP S5982375 A JPS5982375 A JP S5982375A
Authority
JP
Japan
Prior art keywords
alkyl
quinoxalinedione
compound
hydrogen
general formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP58182918A
Other languages
English (en)
Japanese (ja)
Inventor
ウインストン・エス・マ−シヤル
ジエロ−ム・エイチ・フレイシユ
ジヨ−ジ・ジエイ・キユリナン
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of JPS5982375A publication Critical patent/JPS5982375A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/36—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems
    • C07D241/38—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings condensed with carbocyclic rings or ring systems with only hydrogen or carbon atoms directly attached to the ring nitrogen atoms
    • C07D241/40—Benzopyrazines
    • C07D241/42—Benzopyrazines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Immunology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP58182918A 1982-09-30 1983-09-29 ６−アニリノ−５，８−キノキサリンジオン類 Pending JPS5982375A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US06/430,896 US4486432A (en) 1982-09-30 1982-09-30 Quinoxalinedione leukotriene release inhibitors
US430896 1982-09-30

Publications (1)

Publication Number Publication Date
JPS5982375A true JPS5982375A (ja) 1984-05-12

Family

ID=23709539

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58182918A Pending JPS5982375A (ja) 1982-09-30 1983-09-29 ６−アニリノ−５，８−キノキサリンジオン類

Country Status (12)

Country Link
US (1) US4486432A (en:Method)
EP (1) EP0107365B1 (en:Method)
JP (1) JPS5982375A (en:Method)
KR (1) KR860001583B1 (en:Method)
CA (1) CA1212677A (en:Method)
DE (1) DE3372615D1 (en:Method)
DK (1) DK159108C (en:Method)
GB (1) GB2127815B (en:Method)
GR (1) GR78726B (en:Method)
HU (1) HU191639B (en:Method)
IE (1) IE55975B1 (en:Method)
IL (1) IL69816A0 (en:Method)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4692449A (en) * 1986-06-20 1987-09-08 American Cyanamid Company Substituted quinolinediones
US4742059A (en) * 1986-06-20 1988-05-03 American Cyanamide Company Substituted quinoxalinediones and their methods of use
US4808586A (en) * 1987-11-23 1989-02-28 American Cyanamid Company Substituted benzimidazoles and benzothidiazoles having anti-asthmatic and/or anti-inflammatory activities
WO1999052365A1 (en) * 1998-04-13 1999-10-21 Eli Lilly And Company Anticancer agents
AU2006311577B2 (en) 2005-11-09 2013-02-07 Zalicus Inc. Methods, compositions, and kits for the treatment of medical conditions

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE795970A (fr) * 1972-02-29 1973-08-27 Pfizer Nouveaux derives de quinoleine, quinoxaline et quinazoline er composition pharmaceutiques les contenant
DE2860806D1 (en) * 1977-11-10 1981-10-01 Beecham Group Plc 4,9-dihydro-4,9-dioxo-1h-naphtho(2,3-d) triazoles, their preparation and antiallergic compositions containing them

Also Published As

Publication number Publication date
DK159108C (da) 1991-03-11
EP0107365A3 (en) 1985-05-15
IE832277L (en) 1984-03-30
EP0107365B1 (en) 1987-07-22
HU191639B (en) 1987-03-30
DK446683D0 (da) 1983-09-29
DE3372615D1 (de) 1987-08-27
DK446683A (da) 1984-03-31
CA1212677A (en) 1986-10-14
US4486432A (en) 1984-12-04
KR860001583B1 (ko) 1986-10-10
EP0107365A2 (en) 1984-05-02
GB2127815A (en) 1984-04-18
KR840006219A (ko) 1984-11-22
GB2127815B (en) 1985-12-11
GR78726B (en:Method) 1984-10-02
IE55975B1 (en) 1991-03-13
GB8325679D0 (en) 1983-10-26
DK159108B (da) 1990-09-03
IL69816A0 (en) 1983-12-30

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