JPS5962594A - ３，５―ジ置換―トリアゾロピリミジン誘導体 - Google Patents

３，５―ジ置換―トリアゾロピリミジン誘導体

Info

Publication number
JPS5962594A
JPS5962594A JP17117282A JP17117282A JPS5962594A JP S5962594 A JPS5962594 A JP S5962594A JP 17117282 A JP17117282 A JP 17117282A JP 17117282 A JP17117282 A JP 17117282A JP S5962594 A JPS5962594 A JP S5962594A
Authority
JP
Japan
Prior art keywords
compound
formula
group
disubstituted
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP17117282A
Other languages
English (en)
Japanese (ja)
Other versions
JPH033675B2 (en, 2012
Inventor
Takeo Tono
東野　武郎
Eisaku Hayashi
林　英作
Tatsuhiko Katori
香取　達彦
Takako Wakabayashi
若林　貴子
Kenichi Kukita
茎田　憲一
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SSP Co Ltd
Original Assignee
SSP Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SSP Co Ltd filed Critical SSP Co Ltd
Priority to JP17117282A priority Critical patent/JPS5962594A/ja
Publication of JPS5962594A publication Critical patent/JPS5962594A/ja
Publication of JPH033675B2 publication Critical patent/JPH033675B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP17117282A 1982-09-30 1982-09-30 ３，５―ジ置換―トリアゾロピリミジン誘導体 Granted JPS5962594A (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP17117282A JPS5962594A (ja) 1982-09-30 1982-09-30 ３，５―ジ置換―トリアゾロピリミジン誘導体

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP17117282A JPS5962594A (ja) 1982-09-30 1982-09-30 ３，５―ジ置換―トリアゾロピリミジン誘導体

Publications (2)

Publication Number Publication Date
JPS5962594A true JPS5962594A (ja) 1984-04-10
JPH033675B2 JPH033675B2 (en, 2012) 1991-01-21

Family

ID=15918328

Family Applications (1)

Application Number Title Priority Date Filing Date
JP17117282A Granted JPS5962594A (ja) 1982-09-30 1982-09-30 ３，５―ジ置換―トリアゾロピリミジン誘導体

Country Status (1)

Country Link
JP (1) JPS5962594A (en, 2012)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005012307A1 (en) * 2003-07-16 2005-02-10 Janssen Pharmaceutica N.V. Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
WO2005012304A3 (en) * 2003-07-16 2007-04-26 Janssen Pharmaceutica Nv Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
WO2006076442A3 (en) * 2005-01-14 2007-08-23 Janssen Pharmaceutica Nv Triazolopyrimidine derivatives
US20120190697A1 (en) * 2004-10-29 2012-07-26 Guillemont Jerome Emile Georges Hiv inhibiting bicyclic pyrimidine derivatives
US8236809B2 (en) 2004-05-18 2012-08-07 Vasopharm Gmbh Substituted 1,2,3-triazolopyrimidines for the inhibition of NAD(P)H oxidases and platelet activation
WO2014135244A1 (en) * 2013-03-05 2014-09-12 Merck Patent Gmbh Triazolo[4,5-d]pyrimidine derivatives for the treatment of diseases such as cancer

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS56131586A (en) * 1980-03-18 1981-10-15 Ss Pharmaceut Co Ltd Triazolopyrimidine derivative and its preparation

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS56131586A (en) * 1980-03-18 1981-10-15 Ss Pharmaceut Co Ltd Triazolopyrimidine derivative and its preparation

Cited By (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN100549014C (zh) 2003-07-16 2009-10-14 詹森药业有限公司 作为糖原合酶激酶3抑制剂的三唑并嘧啶衍生物
WO2005012304A3 (en) * 2003-07-16 2007-04-26 Janssen Pharmaceutica Nv Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
EA010109B1 (ru) * 2003-07-16 2008-06-30 Янссен Фармацевтика Н.В. Триазолопиримидиновые производные в качестве ингибиторов киназы-3 гликогенсинтазы
CN100404536C (zh) * 2003-07-16 2008-07-23 詹森药业有限公司 作为糖原合酶激酶3抑制剂的三唑并嘧啶衍生物
US7449465B2 (en) 2003-07-16 2008-11-11 Janssen Pharmaceutica, N.V. Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
EA011300B1 (ru) * 2003-07-16 2009-02-27 Янссен Фармацевтика Н.В. Производные триазолопиримидина в качестве ингибиторов киназы гликогенсинтазы-3
AU2004260738B2 (en) * 2003-07-16 2009-07-16 Janssen Pharmaceutica N.V. Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
WO2005012307A1 (en) * 2003-07-16 2005-02-10 Janssen Pharmaceutica N.V. Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors
US8236809B2 (en) 2004-05-18 2012-08-07 Vasopharm Gmbh Substituted 1,2,3-triazolopyrimidines for the inhibition of NAD(P)H oxidases and platelet activation
US20120190697A1 (en) * 2004-10-29 2012-07-26 Guillemont Jerome Emile Georges Hiv inhibiting bicyclic pyrimidine derivatives
US9487518B2 (en) * 2004-10-29 2016-11-08 Janssen Sciences Ireland Uc HIV inhibiting bicyclic pyrimidine derivatives
US9802943B2 (en) 2004-10-29 2017-10-31 Janssen Sciences Ireland Uc HIV inhibiting bicyclic pyrimidine derivatives
US10072015B2 (en) 2004-10-29 2018-09-11 Janssen Sciences Ireland Uc HIV inhibiting bicyclic pyrimidine derivatives
US10077270B2 (en) 2004-10-29 2018-09-18 Janssen Sciences Ireland Uc HIV inhibiting bicyclic pyrimidine derivatives
US7563781B2 (en) * 2005-01-14 2009-07-21 Janssen Pharmaceutica Nv Triazolopyrimidine derivatives
WO2006076442A3 (en) * 2005-01-14 2007-08-23 Janssen Pharmaceutica Nv Triazolopyrimidine derivatives
WO2014135244A1 (en) * 2013-03-05 2014-09-12 Merck Patent Gmbh Triazolo[4,5-d]pyrimidine derivatives for the treatment of diseases such as cancer
CN105026398A (zh) * 2013-03-05 2015-11-04 默克专利股份公司 用于治疗疾病诸如癌症的三唑并[4,5-d]嘧啶衍生物
JP2016510044A (ja) * 2013-03-05 2016-04-04 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングＭｅｒｃｋ Ｐａｔｅｎｔ Ｇｅｓｅｌｌｓｃｈａｆｔ ｍｉｔ ｂｅｓｃｈｒａｅｎｋｔｅｒ Ｈａｆｔｕｎｇ 癌などの疾患の処置のためのトリアゾロ［４，５−ｄ］ピリミジン誘導体
AU2014224975B2 (en) * 2013-03-05 2017-09-14 Merck Patent Gmbh Triazolo(4,5-d)pyrimidine derivatives for the treatment of diseases such as cancer
US9855268B2 (en) 2013-03-05 2018-01-02 Merck Patent Gmbh Triazolo[4,5-d]pyrimidine derivatives

Also Published As

Publication number Publication date
JPH033675B2 (en, 2012) 1991-01-21

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