JPS5815997A - 新規なタイロシン誘導体 - Google Patents

新規なタイロシン誘導体

Info

Publication number
JPS5815997A
JPS5815997A JP56107485A JP10748581A JPS5815997A JP S5815997 A JPS5815997 A JP S5815997A JP 56107485 A JP56107485 A JP 56107485A JP 10748581 A JP10748581 A JP 10748581A JP S5815997 A JPS5815997 A JP S5815997A
Authority
JP
Japan
Prior art keywords
chloroform
solution
residue
reduced pressure
under reduced
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP56107485A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6242919B2 (enrdf_load_stackoverflow
Inventor
Hamao Umezawa
梅沢　浜夫
Sumio Umezawa
梅沢　純夫
Osamu Tsuchiya
修 土屋
Tomio Takeuchi
富雄 竹内
Akihiro Tanaka
昭弘 田中
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Microbial Chemistry Research Foundation
Original Assignee
Microbial Chemistry Research Foundation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Microbial Chemistry Research Foundation filed Critical Microbial Chemistry Research Foundation
Priority to JP56107485A priority Critical patent/JPS5815997A/ja
Priority to AU85524/82A priority patent/AU551142B2/en
Priority to US06/395,463 priority patent/US4477443A/en
Priority to KR1019820003045A priority patent/KR840000583A/ko
Priority to ES513827A priority patent/ES8308333A1/es
Priority to EP84201085A priority patent/EP0132895A1/en
Priority to EP82303622A priority patent/EP0070170B1/en
Priority to DE8282303622T priority patent/DE3269164D1/de
Priority to AT82303622T priority patent/ATE18055T1/de
Priority to EP84201086A priority patent/EP0134054A1/en
Publication of JPS5815997A publication Critical patent/JPS5815997A/ja
Priority to ES520905A priority patent/ES520905A0/es
Priority to SU833624073A priority patent/SU1282821A3/ru
Priority to SU833622787A priority patent/SU1200852A3/ru
Publication of JPS6242919B2 publication Critical patent/JPS6242919B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP56107485A 1981-07-09 1981-07-09 新規なタイロシン誘導体 Granted JPS5815997A (ja)

Priority Applications (13)

Application Number Priority Date Filing Date Title
JP56107485A JPS5815997A (ja) 1981-07-09 1981-07-09 新規なタイロシン誘導体
AU85524/82A AU551142B2 (en) 1981-07-09 1982-07-01 Tylosin derivatives
US06/395,463 US4477443A (en) 1981-07-09 1982-07-06 Tylosin derivatives, their preparation and pharmaceutical compositions containing them
KR1019820003045A KR840000583A (ko) 1981-07-09 1982-07-08 타이로신 유도체의 제조방법
ES513827A ES8308333A1 (es) 1981-07-09 1982-07-08 Un metodo de produccion de un derivado de tilosina.
DE8282303622T DE3269164D1 (en) 1981-07-09 1982-07-09 Tylosin derivatives, their preparation and pharmaceutical compositions containing them
EP82303622A EP0070170B1 (en) 1981-07-09 1982-07-09 Tylosin derivatives, their preparation and pharmaceutical compositions containing them
EP84201085A EP0132895A1 (en) 1981-07-09 1982-07-09 Tylosin derivatives, their preparation and pharmaceutical compositions containing them
AT82303622T ATE18055T1 (de) 1981-07-09 1982-07-09 Tylosinderivate, ihre herstellung und sie enthaltende pharmazeutische zusammensetzungen.
EP84201086A EP0134054A1 (en) 1981-07-09 1982-07-09 Tylosin derivatives, their preparation and pharmaceutical compositions containing them
ES520905A ES520905A0 (es) 1981-07-09 1983-03-23 Un metodo para la preparacion de un derivado de tilosina.
SU833624073A SU1282821A3 (ru) 1981-07-09 1983-07-21 Способ получени тилозиновых производных
SU833622787A SU1200852A3 (ru) 1981-07-09 1983-07-21 Способ получени тилозиновых производных

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP56107485A JPS5815997A (ja) 1981-07-09 1981-07-09 新規なタイロシン誘導体

Publications (2)

Publication Number Publication Date
JPS5815997A true JPS5815997A (ja) 1983-01-29
JPS6242919B2 JPS6242919B2 (enrdf_load_stackoverflow) 1987-09-10

Family

ID=14460406

Family Applications (1)

Application Number Title Priority Date Filing Date
JP56107485A Granted JPS5815997A (ja) 1981-07-09 1981-07-09 新規なタイロシン誘導体

Country Status (3)

Country Link
JP (1) JPS5815997A (enrdf_load_stackoverflow)
KR (1) KR840000583A (enrdf_load_stackoverflow)
SU (2) SU1200852A3 (enrdf_load_stackoverflow)

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5933298A (ja) * 1982-08-19 1984-02-23 Microbial Chem Res Found タイロシン誘導体
JPS5944398A (ja) * 1982-08-02 1984-03-12 フアイザ−・インコ−ポレ−テツド 抗菌性マイコサミノシルタイロノライド及び関連マクロライド誘導体
JPS6150993A (ja) * 1984-08-17 1986-03-13 Microbial Chem Res Found ２３位が塩基性基で置換されたマイカミノシルタイロノライド誘導体およびその製造法
JPS61167695A (ja) * 1985-01-18 1986-07-29 イーライ・リリー・アンド・カンパニー マクロライド誘導体
WO2006078032A1 (ja) * 2005-01-24 2006-07-27 Microbial Chemistry Research Foundation 抗ペニシリン耐性肺炎球菌剤及び新規１６員環マクロライド誘導体

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5944398A (ja) * 1982-08-02 1984-03-12 フアイザ−・インコ−ポレ−テツド 抗菌性マイコサミノシルタイロノライド及び関連マクロライド誘導体
JPS5933298A (ja) * 1982-08-19 1984-02-23 Microbial Chem Res Found タイロシン誘導体
JPS6150993A (ja) * 1984-08-17 1986-03-13 Microbial Chem Res Found ２３位が塩基性基で置換されたマイカミノシルタイロノライド誘導体およびその製造法
JPS61167695A (ja) * 1985-01-18 1986-07-29 イーライ・リリー・アンド・カンパニー マクロライド誘導体
WO2006078032A1 (ja) * 2005-01-24 2006-07-27 Microbial Chemistry Research Foundation 抗ペニシリン耐性肺炎球菌剤及び新規１６員環マクロライド誘導体
AU2006206952B2 (en) * 2005-01-24 2011-08-18 Microbial Chemistry Research Foundation Anti-penicillin resistant pneumococci agent and novel 16-membered ring macrolide derivative
US8053418B2 (en) 2005-01-24 2011-11-08 Microbial Chemistry Research Foundation Anti-penicillin resistant pneumococci agent and novel 16-membered macrolide derivative
JP5129485B2 (ja) * 2005-01-24 2013-01-30 公益財団法人微生物化学研究会 抗ペニシリン耐性肺炎球菌剤及び新規１６員環マクロライド誘導体
US8507453B2 (en) 2005-01-24 2013-08-13 Microbial Chemistry Research Foundation Anti-penicillin resistant pneumococci agent and novel 16-membered macrolide derivative

Also Published As

Publication number Publication date
SU1282821A3 (ru) 1987-01-07
SU1200852A3 (ru) 1985-12-23
JPS6242919B2 (enrdf_load_stackoverflow) 1987-09-10
KR840000583A (ko) 1984-02-25

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