JPS5752359B2 - - Google Patents
Info
- Publication number
- JPS5752359B2 JPS5752359B2 JP48089358A JP8935873A JPS5752359B2 JP S5752359 B2 JPS5752359 B2 JP S5752359B2 JP 48089358 A JP48089358 A JP 48089358A JP 8935873 A JP8935873 A JP 8935873A JP S5752359 B2 JPS5752359 B2 JP S5752359B2
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F1/00—Compounds containing elements of Groups 1 or 11 of the Periodic Table
- C07F1/005—Compounds containing elements of Groups 1 or 11 of the Periodic Table without C-Metal linkages
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F1/00—Compounds containing elements of Groups 1 or 11 of the Periodic Table
- C07F1/08—Copper compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/06—Phosphorus compounds without P—C bonds
- C07F9/08—Esters of oxyacids of phosphorus
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB3765572A GB1440063A (en) | 1972-08-11 | 1972-08-11 | 17alpha-esters of 17alpha,21-dihydroxy-20-oxo-steroids |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS4985062A JPS4985062A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-08-15 |
| JPS5752359B2 true JPS5752359B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1982-11-06 |
Family
ID=10398029
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP48089358A Expired JPS5752359B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1972-08-11 | 1973-08-10 |
Country Status (16)
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1516095A (en) * | 1974-07-31 | 1978-06-28 | Glaxo Lab Ltd | 17,21-diesters of 17alpha,21-dihydroxy-steroids of the pregnane series |
| GB1593978A (en) * | 1976-12-31 | 1981-07-22 | Lark Spa | Anti-inflammatory steroids |
| US4086254A (en) * | 1977-04-13 | 1978-04-25 | The Upjohn Company | Photocleavable steroids |
| DE2735110A1 (de) * | 1977-08-04 | 1979-02-15 | Hoechst Ag | Corticoid-17-alkylcarbonate und verfahren zu ihrer herstellung |
| DE2759135A1 (de) * | 1977-12-30 | 1979-07-19 | Lark Spa | Neue steroidverbindungen und deren herstellung und verwendung |
| DE2817988A1 (de) * | 1978-04-25 | 1979-11-08 | Hoechst Ag | Corticoid 17-alkylcarbonate und verfahren zu deren herstellung |
| DE3133082A1 (de) | 1981-08-18 | 1983-03-10 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | Neue hydrocortison-derivate, ihre herstellung und verwendung |
| AU558725B2 (en) * | 1983-09-07 | 1987-02-05 | Mitsubishi Kasei Corporation | Corticoid derivatives |
| DE3637806A1 (de) * | 1986-11-06 | 1988-05-19 | Hoechst Ag | Verfahren zur herstellung von prednisolon-17-ethylcarbonat durch umlagerung von prednisolon-21-ethylcarbonat |
| FR2683530B1 (fr) * | 1991-11-08 | 1994-01-21 | Roussel Uclaf | Nouveau procede de preparation de derives 20-oxo 17 alpha, 21-dihydroxyles du pregnane et nouveaux intermediaires. |
| US6777399B2 (en) * | 2000-08-05 | 2004-08-17 | Smithkline Beecham Corporation | Anti-inflammatory androstane derivative compositions |
| BRPI0113042B8 (pt) * | 2000-08-05 | 2021-05-25 | Glaxo Group Ltd | composto da fórmula ou um seu solvato fisiologicamente aceitável, uso do mesmo, composição farmacêutica, formulação farmacêutica, método para o tratamento de um indivíduo humano ou animal com uma condição inflamatória e/ou alérgica, e, processo para preparar um composto ou um seu solvato |
| GB0019172D0 (en) * | 2000-08-05 | 2000-09-27 | Glaxo Group Ltd | Novel compounds |
| US6759398B2 (en) * | 2000-08-05 | 2004-07-06 | Smithkline Beecham Corporation | Anti-inflammatory androstane derivative |
| US6858596B2 (en) * | 2000-08-05 | 2005-02-22 | Smithkline Beecham Corporation | Formulation containing anti-inflammatory androstane derivative |
| JP4446661B2 (ja) * | 2001-04-30 | 2010-04-07 | グラクソ グループ リミテッド | 抗炎症性の、１７α位に環状エステル基を有するアンドロスタンの１７β−カルボチオ酸エステル誘導体 |
| WO2003048181A1 (en) * | 2001-12-01 | 2003-06-12 | Glaxo Group Limited | 17.alpha. -cyclic esters of 16-methylpregnan-3,20-dione as anti-inflammatory agents |
| US20050175545A1 (en) * | 2002-02-04 | 2005-08-11 | Keith Biggadike | Formulation for inhalation comprising a glucocorticoid and a beta 2-adrenoreceptor agonist |
| GB0202635D0 (en) * | 2002-02-05 | 2002-03-20 | Glaxo Wellcome Mfg Pte Ltd | Formulation containing novel anti-inflammatory androstane derivative |
| GB2389530B (en) * | 2002-06-14 | 2007-01-10 | Cipla Ltd | Pharmaceutical compositions |
| GB0507165D0 (en) * | 2005-04-08 | 2005-05-18 | Glaxo Group Ltd | Novel crystalline pharmaceutical product |
| GB0615108D0 (en) * | 2006-07-28 | 2006-09-06 | Glaxo Group Ltd | Novel formulations |
| NZ603107A (en) | 2008-05-28 | 2014-03-28 | Validus Biopharma Inc | Non-hormonal steroid modulators of nf-kb for treatment of disease |
| WO2011127048A2 (en) | 2010-04-05 | 2011-10-13 | Validus Biopharma | NON-HORMONAL STEROID MODULATORS OF NF-ĸB FOR TREATMENT OF DISEASE |
| WO2017004205A1 (en) | 2015-06-29 | 2017-01-05 | Reveragen Biopharma, Inc. | NON-HORMONAL STEROID MODULATORS OF NF-κB FOR TREATMENT OF DISEASE |
| US11382922B2 (en) | 2019-03-07 | 2022-07-12 | Reveragen Biopharma, Inc. | Aqueous oral pharmaceutical suspension compositions |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3255218A (en) * | 1962-03-28 | 1966-06-07 | Schering Corp | 17(20)-enol-21-aldehydes of the pregnane series |
| US3780177A (en) * | 1967-06-16 | 1973-12-18 | Warner Lambert Co | 17-butyrate,21-ester derivatives of 6alpha,9alpha-difluoroprednisolone,compositions and use |
| IT1034011B (it) * | 1969-06-26 | 1979-09-10 | Vister Vismara Terapeutici S P | Processo per la prapratzione di 17 monoesteri di 17 a 21 diossisteroidi per idrolisi die corpispondenti 17 21 ortoesteri ciclici a ph control lato |
-
1972
- 1972-08-11 GB GB3765572A patent/GB1440063A/en not_active Expired
-
1973
- 1973-08-10 ES ES417738A patent/ES417738A1/es not_active Expired
- 1973-08-10 SE SE7310985A patent/SE387951B/xx unknown
- 1973-08-10 IE IE1382/73A patent/IE38312B1/xx unknown
- 1973-08-10 ZA ZA735453A patent/ZA735453B/xx unknown
- 1973-08-10 ZA ZA735452A patent/ZA735452B/xx unknown
- 1973-08-10 CH CH1159373A patent/CH590884A5/xx not_active IP Right Cessation
- 1973-08-10 US US387487A patent/US3891631A/en not_active Expired - Lifetime
- 1973-08-10 NL NL7311072A patent/NL7311072A/xx not_active Application Discontinuation
- 1973-08-10 JP JP48089358A patent/JPS5752359B2/ja not_active Expired
- 1973-08-10 IL IL42942A patent/IL42942A/en unknown
- 1973-08-10 FR FR7329443A patent/FR2205508B1/fr not_active Expired
- 1973-08-10 BE BE134445A patent/BE803461A/xx unknown
- 1973-08-10 DK DK440673AA patent/DK135998B/da unknown
- 1973-08-10 DE DE19732340591 patent/DE2340591A1/de not_active Ceased
- 1973-08-10 LU LU68212A patent/LU68212A1/xx unknown
- 1973-08-10 CA CA178,554A patent/CA1027109A/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| DK135998C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-12-27 |
| NL7311072A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-02-13 |
| DE2340591A1 (de) | 1974-03-07 |
| IE38312B1 (en) | 1978-02-15 |
| IE38312L (en) | 1974-02-11 |
| AU5914373A (en) | 1975-02-13 |
| JPS4985062A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-08-15 |
| IL42942A0 (en) | 1973-11-28 |
| ZA735453B (en) | 1974-10-30 |
| ZA735452B (en) | 1974-07-31 |
| DK135998B (da) | 1977-07-25 |
| LU68212A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1973-10-16 |
| SE387951B (sv) | 1976-09-20 |
| CH590884A5 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1977-08-31 |
| BE803461A (fr) | 1974-02-11 |
| IL42942A (en) | 1977-05-31 |
| US3891631A (en) | 1975-06-24 |
| FR2205508B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1978-09-15 |
| FR2205508A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-05-31 |
| ES417738A1 (es) | 1976-06-16 |
| GB1440063A (en) | 1976-06-23 |
| CA1027109A (en) | 1978-02-28 |