JPS57212154A - Novel aminosulfonylbenzoic acid derivative - Google Patents

Novel aminosulfonylbenzoic acid derivative

Info

Publication number
JPS57212154A
JPS57212154A JP56096377A JP9637781A JPS57212154A JP S57212154 A JPS57212154 A JP S57212154A JP 56096377 A JP56096377 A JP 56096377A JP 9637781 A JP9637781 A JP 9637781A JP S57212154 A JPS57212154 A JP S57212154A
Authority
JP
Japan
Prior art keywords
acid
acid derivative
novel
formulai
deoxidizer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP56096377A
Other languages
Japanese (ja)
Inventor
Hideo Maeda
Shoichi Kono
Haruo Onishi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hodogaya Chemical Co Ltd
Mochida Pharmaceutical Co Ltd
Original Assignee
Hodogaya Chemical Co Ltd
Mochida Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hodogaya Chemical Co Ltd, Mochida Pharmaceutical Co Ltd filed Critical Hodogaya Chemical Co Ltd
Priority to JP56096377A priority Critical patent/JPS57212154A/en
Priority to GB08133391A priority patent/GB2100720A/en
Priority to DE19813144688 priority patent/DE3144688A1/en
Priority to FR8121018A priority patent/FR2508038A1/en
Priority to AU85096/82A priority patent/AU539797B2/en
Priority to NL8220204A priority patent/NL8220204A/en
Priority to SE8203877A priority patent/SE8203877L/en
Priority to PCT/JP1982/000241 priority patent/WO1983000044A1/en
Priority to EP82105459A priority patent/EP0068407A1/en
Publication of JPS57212154A publication Critical patent/JPS57212154A/en
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/48—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups having nitrogen atoms of sulfonamide groups further bound to another hetero atom
    • C07C311/49—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups having nitrogen atoms of sulfonamide groups further bound to another hetero atom to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C311/50—Compounds containing any of the groups, X being a hetero atom, Y being any atom
    • C07C311/52—Y being a hetero atom
    • C07C311/64—X and Y being nitrogen atoms, e.g. N-sulfonylguanidine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/20—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

NEW MATERIAL:An amiosulfonylhalogenobenzoic acid derivative shown by the formulaI(X and Y are Cl, Br, H, amino, or nitro; R1 is H, or lower alkyl; R2 is H, amino, lowr alkyl, hydroxyalkyl, etc.).
EXAMPLE: 5-Aminosulfonyl-2,4-dichlorobenzoic acid.
USE: A virucide.
PROCESS: A halogenobenzoic acid is heated in chlorosulfonic acid to give chlorosulfonylbenzoic acid, which is reacted with an amine shown by the formula II at room temperature, and, if necessary, under heating, in a solvent such as water, dioxane THF, etc. in the presence of a deoxidizer (e.g., TEA) or with the amine shown by the formula II itself as the deoxidizer, to give a compound shown by the formulaI.
COPYRIGHT: (C)1982,JPO&Japio
JP56096377A 1981-06-22 1981-06-22 Novel aminosulfonylbenzoic acid derivative Pending JPS57212154A (en)

Priority Applications (9)

Application Number Priority Date Filing Date Title
JP56096377A JPS57212154A (en) 1981-06-22 1981-06-22 Novel aminosulfonylbenzoic acid derivative
GB08133391A GB2100720A (en) 1981-06-22 1981-11-05 Aminosulfonylbenzoic acid derivatives
DE19813144688 DE3144688A1 (en) 1981-06-22 1981-11-10 AMINOSULFONYLBENZOESAEUR DERIVATIVES
FR8121018A FR2508038A1 (en) 1981-06-22 1981-11-10 AMINOSULFONYLBENZOIC ACID DERIVATIVES USEFUL AS MEDICAMENTS
AU85096/82A AU539797B2 (en) 1981-06-22 1982-06-22 Aminosulfonyl benzoic acid derivatives
NL8220204A NL8220204A (en) 1981-06-22 1982-06-22 NEW AMINOSULPHONYLBENZOIC ACID DERIVATIVES AND PROCESS FOR PREPARING THEREOF.
SE8203877A SE8203877L (en) 1981-06-22 1982-06-22 AMINOSULFONYLBENSOESYRADERIVAT
PCT/JP1982/000241 WO1983000044A1 (en) 1981-06-22 1982-06-22 Novel aminosulfonylbenzoic acid derivatives and process for their preparation
EP82105459A EP0068407A1 (en) 1981-06-22 1982-06-22 Aminosulfonylbenzoic acid derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP56096377A JPS57212154A (en) 1981-06-22 1981-06-22 Novel aminosulfonylbenzoic acid derivative

Publications (1)

Publication Number Publication Date
JPS57212154A true JPS57212154A (en) 1982-12-27

Family

ID=14163267

Family Applications (1)

Application Number Title Priority Date Filing Date
JP56096377A Pending JPS57212154A (en) 1981-06-22 1981-06-22 Novel aminosulfonylbenzoic acid derivative

Country Status (4)

Country Link
JP (1) JPS57212154A (en)
DE (1) DE3144688A1 (en)
FR (1) FR2508038A1 (en)
GB (1) GB2100720A (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003004461A1 (en) * 2001-07-02 2003-01-16 Schering Corporation Drugs for treating viral infections

Also Published As

Publication number Publication date
GB2100720A (en) 1983-01-06
FR2508038A1 (en) 1982-12-24
DE3144688A1 (en) 1983-01-05

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