JPS57197270A - Production of 2-hydroxyquinoxaline derivative - Google Patents
Production of 2-hydroxyquinoxaline derivativeInfo
- Publication number
- JPS57197270A JPS57197270A JP8031781A JP8031781A JPS57197270A JP S57197270 A JPS57197270 A JP S57197270A JP 8031781 A JP8031781 A JP 8031781A JP 8031781 A JP8031781 A JP 8031781A JP S57197270 A JPS57197270 A JP S57197270A
- Authority
- JP
- Japan
- Prior art keywords
- sulfite
- hydroxyquinoxaline
- formulai
- compound
- reduced
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Abstract
PURPOSE: 2-Hydroxyquinoxaline-4-oxide derivative, as a starting material, is reduced in an alkaline aqueous solution (using water instead of an organic solvent) to produce the titled substance used as a synthetic intermediate of medicaments with no formation of by-products economically and safely.
CONSTITUTION: 2-Hydroxyquinoxaline-4-oxide derivative of formulaI(X is halogen, trifluoromethyl) is reduced with a hydrogen sulfite and/or sulfite salt in the presence of an aqueous alkali such as aqueous sodium hydroxide and/or potassium hydroxide to give a compound of formula II. The concentration of the above aqueous alkali is 2W15wt%, preferably 5W10wt%. Preferable example of the hidrogen sulfite and sulfite salt is sodium hydrogen sulfite or disodium sulfite. The amount is 2W10, preferably 2W5 times the molar amount of the compound of formulaI.
COPYRIGHT: (C)1982,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP8031781A JPS57197270A (en) | 1981-05-27 | 1981-05-27 | Production of 2-hydroxyquinoxaline derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP8031781A JPS57197270A (en) | 1981-05-27 | 1981-05-27 | Production of 2-hydroxyquinoxaline derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS57197270A true JPS57197270A (en) | 1982-12-03 |
Family
ID=13714875
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP8031781A Pending JPS57197270A (en) | 1981-05-27 | 1981-05-27 | Production of 2-hydroxyquinoxaline derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS57197270A (en) |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3419471A1 (en) * | 1983-05-25 | 1984-11-29 | Nippon Kayaku K.K., Tokio/Tokyo | METHOD FOR PRODUCING 2-CHINOXALINOLS |
EP0745594A4 (en) * | 1994-02-17 | 1997-04-09 | Nissan Chemical Ind Ltd | Process for producing 6-substituted 2(1h)-quinoxalinone |
CN102675233A (en) * | 2012-05-25 | 2012-09-19 | 安徽丰乐农化有限责任公司 | New high-yield production process of 6-chloro-2-hydroxyquinoxaline |
-
1981
- 1981-05-27 JP JP8031781A patent/JPS57197270A/en active Pending
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3419471A1 (en) * | 1983-05-25 | 1984-11-29 | Nippon Kayaku K.K., Tokio/Tokyo | METHOD FOR PRODUCING 2-CHINOXALINOLS |
EP0745594A4 (en) * | 1994-02-17 | 1997-04-09 | Nissan Chemical Ind Ltd | Process for producing 6-substituted 2(1h)-quinoxalinone |
CN102675233A (en) * | 2012-05-25 | 2012-09-19 | 安徽丰乐农化有限责任公司 | New high-yield production process of 6-chloro-2-hydroxyquinoxaline |
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