JPS57165357A - Novel optically active azidocarboxylic acid or ester thereof and its preparation - Google Patents
Novel optically active azidocarboxylic acid or ester thereof and its preparationInfo
- Publication number
- JPS57165357A JPS57165357A JP5032381A JP5032381A JPS57165357A JP S57165357 A JPS57165357 A JP S57165357A JP 5032381 A JP5032381 A JP 5032381A JP 5032381 A JP5032381 A JP 5032381A JP S57165357 A JPS57165357 A JP S57165357A
- Authority
- JP
- Japan
- Prior art keywords
- ester
- optically active
- preparation
- acid
- novel optically
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
NEW MATERIAL:A compound of formulaI(R1 is methyl or ethyl; R2 is H or 1W 4C lower alkyl).
EXAMPLE: 3-Azido-2-D-methylpropionic acid.
USE: Useful as a synthetic intermediate for medicines, e.g. triamcinolone acetonide ester having the anti-inflammatory action.
PROCESS: An optically active 3-organosulfonyloxycarboxylic acid of formula II (R is methyl, ethyl p-methylphenyl or benzyl) or an ester thereof is reacted with an alkali metallic salt of hydrogen azide, e.g. sodium, lithium or potassium salt, in a solvent, e.g. dimethyl sulfoxide or N,N-dimethylformamide, to give the compound of formulaI.
COPYRIGHT: (C)1982,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5032381A JPS57165357A (en) | 1981-04-02 | 1981-04-02 | Novel optically active azidocarboxylic acid or ester thereof and its preparation |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5032381A JPS57165357A (en) | 1981-04-02 | 1981-04-02 | Novel optically active azidocarboxylic acid or ester thereof and its preparation |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS57165357A true JPS57165357A (en) | 1982-10-12 |
JPH0124782B2 JPH0124782B2 (en) | 1989-05-15 |
Family
ID=12855689
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP5032381A Granted JPS57165357A (en) | 1981-04-02 | 1981-04-02 | Novel optically active azidocarboxylic acid or ester thereof and its preparation |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS57165357A (en) |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4855455A (en) * | 1988-01-22 | 1989-08-08 | W. R. Grace & Co.-Conn. | Preparation of amino acid derivatives |
US5580999A (en) * | 1989-12-11 | 1996-12-03 | Hoffmann-La Roche Inc. | Alcohols |
JP2009023933A (en) * | 2007-07-19 | 2009-02-05 | National Institute Of Advanced Industrial & Technology | Nitrogen-containing organic silicon compound |
-
1981
- 1981-04-02 JP JP5032381A patent/JPS57165357A/en active Granted
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4855455A (en) * | 1988-01-22 | 1989-08-08 | W. R. Grace & Co.-Conn. | Preparation of amino acid derivatives |
JPH021447A (en) * | 1988-01-22 | 1990-01-05 | W R Grace & Co | Preparation of amino acid derivative |
US5580999A (en) * | 1989-12-11 | 1996-12-03 | Hoffmann-La Roche Inc. | Alcohols |
JP2009023933A (en) * | 2007-07-19 | 2009-02-05 | National Institute Of Advanced Industrial & Technology | Nitrogen-containing organic silicon compound |
Also Published As
Publication number | Publication date |
---|---|
JPH0124782B2 (en) | 1989-05-15 |
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