JPS5583750A - 5-oxo-3,4,5,6,7,8-hexahydrocarbostyril derivative - Google Patents
5-oxo-3,4,5,6,7,8-hexahydrocarbostyril derivativeInfo
- Publication number
- JPS5583750A JPS5583750A JP15905278A JP15905278A JPS5583750A JP S5583750 A JPS5583750 A JP S5583750A JP 15905278 A JP15905278 A JP 15905278A JP 15905278 A JP15905278 A JP 15905278A JP S5583750 A JPS5583750 A JP S5583750A
- Authority
- JP
- Japan
- Prior art keywords
- hexahydrocarbostyril
- oxo
- derivative
- formula
- solvent
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Quinoline Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:A 5-oxo-3,4,5,6,7,8-hexahydrocarbostyril derivative of formula I (R1,2 are lower alkyl, or R1 and R2 together may form an N-containing saturated heterocyclic ring with adjacent N atom).
EXAMPLE: 6-(Piperidinothiocarbonylthiomethyl)-5-oxo-3, 4, 5, 6, 7, 8-hexahydrocarbostyril.
USE: Antibacterial agent especially effective to Mycoplasma.
PROCESS: 5-Oxo-3,4,5,6,7,8-hexahydrocarbostyril of formula II is reacted with formaldehyde and an amine of formula III in a solvent in the presence of a catalyst at 25W 150°C to afford 6-substituted aminomethyl-5-oxo-3,4,5,6,7,8-hexahydrocarbostyril derivative of formula IV, which is converted to the desired compound I by boiling and refluxing with CS2 in a solvent.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP15905278A JPS5583750A (en) | 1978-12-21 | 1978-12-21 | 5-oxo-3,4,5,6,7,8-hexahydrocarbostyril derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP15905278A JPS5583750A (en) | 1978-12-21 | 1978-12-21 | 5-oxo-3,4,5,6,7,8-hexahydrocarbostyril derivative |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5583750A true JPS5583750A (en) | 1980-06-24 |
JPS617194B2 JPS617194B2 (en) | 1986-03-04 |
Family
ID=15685167
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP15905278A Granted JPS5583750A (en) | 1978-12-21 | 1978-12-21 | 5-oxo-3,4,5,6,7,8-hexahydrocarbostyril derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5583750A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5681839A (en) * | 1994-02-10 | 1997-10-28 | John Wyeth & Brother | Nitrogen heterocycles |
-
1978
- 1978-12-21 JP JP15905278A patent/JPS5583750A/en active Granted
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5681839A (en) * | 1994-02-10 | 1997-10-28 | John Wyeth & Brother | Nitrogen heterocycles |
Also Published As
Publication number | Publication date |
---|---|
JPS617194B2 (en) | 1986-03-04 |
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