JPS55144000A - Preparation of 2-amino-adenosine-3',5'-cyclic phosphoric acid - Google Patents
Preparation of 2-amino-adenosine-3',5'-cyclic phosphoric acidInfo
- Publication number
- JPS55144000A JPS55144000A JP5142279A JP5142279A JPS55144000A JP S55144000 A JPS55144000 A JP S55144000A JP 5142279 A JP5142279 A JP 5142279A JP 5142279 A JP5142279 A JP 5142279A JP S55144000 A JPS55144000 A JP S55144000A
- Authority
- JP
- Japan
- Prior art keywords
- phosphoric acid
- cyclic phosphoric
- adenosine
- formula
- amino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Saccharide Compounds (AREA)
Abstract
PURPOSE: To prepare the title compound useful as an anti-allergic agent, central nervous system depressant, blood platelet coagulation inhibitor, and an intermediate of diuretic, carcinostatic agent, etc., economically, in an industrial scale, by reducing an N6-alkoxy derivative.
CONSTITUTION: The objective compound of formula II is prepared by (1) culturing a specific species of bacteria belonging to Microbacterium genus in a medium containing adenine, xylose, etc. and an inorganic phosphate to obtain adenosine-3',5'- cyclic phosphoric acid, (2) oxidizing the product with H2O2, etc., (3) reacting the resulting 2-imino-6-β-3',5'-cyclic phosphoric acid ribofuranosyl (1,2,4-oxadiazolo [2,3-f]purine) salt of formula I (X is halogen) with an alkyl chloride, (4) subjecting the product to the alkali rearrangement reaction to provide a 2-amino-N6-alkoxy- adenosine-3',5'-cyclic phosphoric acid of formula II (R is lower alkyl), and (5) reducing the compound III with hydrogen in the presence of Pd-C catalyst.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5142279A JPS55144000A (en) | 1979-04-27 | 1979-04-27 | Preparation of 2-amino-adenosine-3',5'-cyclic phosphoric acid |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP5142279A JPS55144000A (en) | 1979-04-27 | 1979-04-27 | Preparation of 2-amino-adenosine-3',5'-cyclic phosphoric acid |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS55144000A true JPS55144000A (en) | 1980-11-10 |
JPS633877B2 JPS633877B2 (en) | 1988-01-26 |
Family
ID=12886480
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP5142279A Granted JPS55144000A (en) | 1979-04-27 | 1979-04-27 | Preparation of 2-amino-adenosine-3',5'-cyclic phosphoric acid |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS55144000A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN106589030A (en) * | 2016-10-28 | 2017-04-26 | 南通宏慈药业有限公司 | Preparation method of adenosine cyclophosphate oxide impurity |
-
1979
- 1979-04-27 JP JP5142279A patent/JPS55144000A/en active Granted
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN106589030A (en) * | 2016-10-28 | 2017-04-26 | 南通宏慈药业有限公司 | Preparation method of adenosine cyclophosphate oxide impurity |
Also Published As
Publication number | Publication date |
---|---|
JPS633877B2 (en) | 1988-01-26 |
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