JPS5436262A - Alphaahalomethyl derivative of amino acid - Google Patents

Alphaahalomethyl derivative of amino acid

Info

Publication number
JPS5436262A
JPS5436262A JP9002378A JP9002378A JPS5436262A JP S5436262 A JPS5436262 A JP S5436262A JP 9002378 A JP9002378 A JP 9002378A JP 9002378 A JP9002378 A JP 9002378A JP S5436262 A JPS5436262 A JP S5436262A
Authority
JP
Japan
Prior art keywords
alphaahalomethyl
derivative
amino acid
amino
acid
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP9002378A
Other languages
English (en)
Other versions
JPS6123792B2 (ja
Inventor
Bei Fuiritsupu
Yunku Mishieru
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merrell Toraude et Cie
Original Assignee
Merrell Toraude et Cie
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Toraude et Cie filed Critical Merrell Toraude et Cie
Publication of JPS5436262A publication Critical patent/JPS5436262A/ja
Publication of JPS6123792B2 publication Critical patent/JPS6123792B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP9002378A 1977-07-28 1978-07-25 Alphaahalomethyl derivative of amino acid Granted JPS5436262A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/819,975 US4315095A (en) 1977-07-28 1977-07-28 α-Halomethyl derivatives of amino acids

Publications (2)

Publication Number Publication Date
JPS5436262A true JPS5436262A (en) 1979-03-16
JPS6123792B2 JPS6123792B2 (ja) 1986-06-07

Family

ID=25229573

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9002378A Granted JPS5436262A (en) 1977-07-28 1978-07-25 Alphaahalomethyl derivative of amino acid

Country Status (16)

Country Link
US (1) US4315095A (ja)
JP (1) JPS5436262A (ja)
AU (1) AU521354B2 (ja)
BE (1) BE869322A (ja)
CA (1) CA1120041A (ja)
CH (1) CH638790A5 (ja)
DE (1) DE2832309A1 (ja)
ES (1) ES471594A1 (ja)
FR (1) FR2398736A1 (ja)
GB (1) GB2001626B (ja)
IE (1) IE46928B1 (ja)
IL (1) IL54914A0 (ja)
IT (1) IT1107454B (ja)
NL (1) NL7807871A (ja)
NZ (1) NZ187537A (ja)
ZA (1) ZA783350B (ja)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS591490A (ja) * 1982-06-29 1984-01-06 Dai Ichi Seiyaku Co Ltd ３−セフェム−４−カルボン酸誘導体
JPH06100446A (ja) * 1990-10-15 1994-04-12 Merck & Co Inc （Ｓ）−α−フルオロメチル−ヒスチジン及びそのエステルを使用するぜん息の治療方法

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4413141A (en) * 1977-07-11 1983-11-01 Merrell Toraude Et Compagnie 2-(Difluoromethyl)-2,5-diaminopentanoic acid
CA1302919C (en) * 1985-07-03 1992-06-09 Robert T. Buckler Histamine derivatives, immunogen conjugates and antibodies raised thereto
US6001926A (en) * 1997-10-02 1999-12-14 The United States Of America As Represented By The Secretary Of The Navy Fiber-reinforced phthalonitrile composite cured with low-reactivity aromatic amine curing agent
EP1321169A1 (en) * 2001-12-18 2003-06-25 Biofrontera Pharmaceuticals AG Combination of a serotonin receptor antagonist with a histidine decarboxylase inhibitor as a medicament

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3169971A (en) * 1965-02-16 A-alkyl histidines
GB715182A (en) * 1951-09-19 1954-09-08 Roche Products Ltd A novel imidazole derivative and process for the manufacture thereof
FR1493402A (fr) * 1962-01-22 1967-09-01 Merck & Co Inc Hydrazino-acides
US3387031A (en) * 1961-06-08 1968-06-04 Union Carbide Corp Synthesis of alpha-amino acid amide hydrohalides
FR1457259A (fr) * 1961-08-18 1966-01-24 Merck & Co Inc Production d'amino-acides du type alpha-alkyl-histidine
NZ187377A (en) * 1977-06-01 1981-05-15 Merck & Co Inc A-amino-a-substituted alkyl-a-fluoromethylacetic acids

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS591490A (ja) * 1982-06-29 1984-01-06 Dai Ichi Seiyaku Co Ltd ３−セフェム−４−カルボン酸誘導体
JPH0251434B2 (ja) * 1982-06-29 1990-11-07 Daiichi Seiyaku Co
JPH06100446A (ja) * 1990-10-15 1994-04-12 Merck & Co Inc （Ｓ）−α−フルオロメチル−ヒスチジン及びそのエステルを使用するぜん息の治療方法

Also Published As

Publication number Publication date
IL54914A0 (en) 1978-08-31
US4315095A (en) 1982-02-09
IT7850463A0 (it) 1978-07-25
DE2832309A1 (de) 1979-02-08
GB2001626B (en) 1982-04-07
NL7807871A (nl) 1979-01-30
FR2398736B1 (ja) 1980-09-19
DE2832309C2 (ja) 1989-07-06
IE46928B1 (en) 1983-11-02
IT1107454B (it) 1985-11-25
ZA783350B (en) 1979-06-27
NZ187537A (en) 1980-08-26
FR2398736A1 (fr) 1979-02-23
IE781149L (en) 1979-01-28
ES471594A1 (es) 1979-10-01
CH638790A5 (de) 1983-10-14
JPS6123792B2 (ja) 1986-06-07
AU521354B2 (en) 1982-04-01
AU3731778A (en) 1980-01-03
CA1120041A (en) 1982-03-16
BE869322A (fr) 1978-11-16
GB2001626A (en) 1979-02-07

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