IT7850463A0 - Derivati alfa-alogenometilici di amminoacidi e relativo procedimentodi produzione - Google Patents

Derivati alfa-alogenometilici di amminoacidi e relativo procedimentodi produzione

Info

Publication number
IT7850463A0
IT7850463A0 IT7850463A IT5046378A IT7850463A0 IT 7850463 A0 IT7850463 A0 IT 7850463A0 IT 7850463 A IT7850463 A IT 7850463A IT 5046378 A IT5046378 A IT 5046378A IT 7850463 A0 IT7850463 A0 IT 7850463A0
Authority
IT
Italy
Prior art keywords
alpha
amino acids
production procedure
related production
halogenomethyl
Prior art date
Application number
IT7850463A
Other languages
English (en)
Other versions
IT1107454B (it
Original Assignee
Merrell Toraude & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Toraude & Co filed Critical Merrell Toraude & Co
Publication of IT7850463A0 publication Critical patent/IT7850463A0/it
Application granted granted Critical
Publication of IT1107454B publication Critical patent/IT1107454B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IT50463/78A 1977-07-28 1978-07-25 Derivati alfa-alogenometilici di amminoacidi e relativo procedimento di produzione IT1107454B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/819,975 US4315095A (en) 1977-07-28 1977-07-28 α-Halomethyl derivatives of amino acids

Publications (2)

Publication Number Publication Date
IT7850463A0 true IT7850463A0 (it) 1978-07-25
IT1107454B IT1107454B (it) 1985-11-25

Family

ID=25229573

Family Applications (1)

Application Number Title Priority Date Filing Date
IT50463/78A IT1107454B (it) 1977-07-28 1978-07-25 Derivati alfa-alogenometilici di amminoacidi e relativo procedimento di produzione

Country Status (16)

Country Link
US (1) US4315095A (it)
JP (1) JPS5436262A (it)
AU (1) AU521354B2 (it)
BE (1) BE869322A (it)
CA (1) CA1120041A (it)
CH (1) CH638790A5 (it)
DE (1) DE2832309A1 (it)
ES (1) ES471594A1 (it)
FR (1) FR2398736A1 (it)
GB (1) GB2001626B (it)
IE (1) IE46928B1 (it)
IL (1) IL54914A0 (it)
IT (1) IT1107454B (it)
NL (1) NL7807871A (it)
NZ (1) NZ187537A (it)
ZA (1) ZA783350B (it)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4413141A (en) * 1977-07-11 1983-11-01 Merrell Toraude Et Compagnie 2-(Difluoromethyl)-2,5-diaminopentanoic acid
JPS591490A (ja) * 1982-06-29 1984-01-06 Dai Ichi Seiyaku Co Ltd 3−セフェム−4−カルボン酸誘導体
CA1302919C (en) * 1985-07-03 1992-06-09 Robert T. Buckler Histamine derivatives, immunogen conjugates and antibodies raised thereto
US5030645A (en) * 1990-10-15 1991-07-09 Merck & Co., Inc. Method of treating asthma using (S)-α-fluoromethyl-histidine and esters thereof
US6001926A (en) * 1997-10-02 1999-12-14 The United States Of America As Represented By The Secretary Of The Navy Fiber-reinforced phthalonitrile composite cured with low-reactivity aromatic amine curing agent
EP1321169A1 (en) * 2001-12-18 2003-06-25 Biofrontera Pharmaceuticals AG Combination of a serotonin receptor antagonist with a histidine decarboxylase inhibitor as a medicament

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3169971A (en) * 1965-02-16 A-alkyl histidines
GB715182A (en) * 1951-09-19 1954-09-08 Roche Products Ltd A novel imidazole derivative and process for the manufacture thereof
FR1493402A (fr) * 1962-01-22 1967-09-01 Merck & Co Inc Hydrazino-acides
US3387031A (en) * 1961-06-08 1968-06-04 Union Carbide Corp Synthesis of alpha-amino acid amide hydrohalides
FR1457259A (fr) * 1961-08-18 1966-01-24 Merck & Co Inc Production d'amino-acides du type alpha-alkyl-histidine
GR64495B (en) * 1977-06-01 1980-03-31 Merck & Co Inc Novel fluorinated amino acids

Also Published As

Publication number Publication date
DE2832309C2 (it) 1989-07-06
CH638790A5 (de) 1983-10-14
AU521354B2 (en) 1982-04-01
JPS6123792B2 (it) 1986-06-07
IT1107454B (it) 1985-11-25
GB2001626B (en) 1982-04-07
BE869322A (fr) 1978-11-16
GB2001626A (en) 1979-02-07
IL54914A0 (en) 1978-08-31
NZ187537A (en) 1980-08-26
JPS5436262A (en) 1979-03-16
ZA783350B (en) 1979-06-27
IE46928B1 (en) 1983-11-02
ES471594A1 (es) 1979-10-01
US4315095A (en) 1982-02-09
AU3731778A (en) 1980-01-03
FR2398736B1 (it) 1980-09-19
CA1120041A (en) 1982-03-16
NL7807871A (nl) 1979-01-30
DE2832309A1 (de) 1979-02-08
FR2398736A1 (fr) 1979-02-23
IE781149L (en) 1979-01-28

Similar Documents

Publication Publication Date Title
IT1112112B (it) Derivati acilici sostituiti di amminoacidi e relativo procedimento di produzione
IT1132392B (it) Derivati di acidi chinolincarbossilici e relativo procedimento di preparazione
IT1096306B (it) Derivati di idantoina ad azione terapeutica e relativo procedimento di preparazione
PL197963A1 (pl) Sposob wytwarzania merkaptocylowych pochodnych aminokwasow
IT7852280A0 (it) Procedimento per la produzione di derivati ammidici in particolare acilanilidi sostituite e prodotto ottenuto
IT1078981B (it) Derivati di acidi fenossi-fenossipropionici
IT7851499A0 (it) Procedimento per la produzione di derivati della xantina e prodotto relativo
IT1105176B (it) Derivati della morfina e relativo procedimento di produzione
IT1092179B (it) Derivati di acidi tiazolidincarbossilici e elativo procedimento di produzione
IT1102599B (it) Derivati di p-amminometil-benzen-solfonammide procedimento di preparazione ed applicazioni
IT1143671B (it) Procedimento per la fabbricazione di triptofano e di suoi derivati
IT7850129A0 (it) Derivati alfa-acetilenici e vinilici di amminoacidi e relativo procedimento di produzione
IT7850463A0 (it) Derivati alfa-alogenometilici di amminoacidi e relativo procedimentodi produzione
IT1134448B (it) Derivati esterei di acidi ciclopropancarbossilici
IT1105172B (it) Derivati della morfina e relativo procedimento di produzione
IT1106121B (it) Derivati 25-alchilcolesterolici e relativo procedimento di produzione
IT1094043B (it) Derivati di acidi ossi-alcanoici
IT1140954B (it) Amminpacil derivati di acidi mercaptoacil amminici
IT1113140B (it) Derivati di amminoalcoli
IT7825800A0 (it) Procedimento per la fabbricazione di p-idrossifenilglicina e suoi derivati
IT7848192A0 (it) Procedimento per la produzione di derivati di 9-2-idrossietossimetilguanina e prodotto ottenuto
IT7850147A0 (it) Derivati di 4-omoisotwistano e relativo procedimento di produzione
IT7850128A0 (it) Derivati di amminoacidi alfa-vinili ci utili in particolare come composti farmaceutici e relativo procedimento di produzione
IT7849828A0 (it) Derivati di 24-deidrovitamina d3 eloro preparazione
IT7949253A0 (it) Derivati della idantoina e relativo procedimento di produzione