JPS5321192A - Cephalosporin derivatives and their preparation - Google Patents

Cephalosporin derivatives and their preparation

Info

Publication number
JPS5321192A
JPS5321192A JP9584976A JP9584976A JPS5321192A JP S5321192 A JPS5321192 A JP S5321192A JP 9584976 A JP9584976 A JP 9584976A JP 9584976 A JP9584976 A JP 9584976A JP S5321192 A JPS5321192 A JP S5321192A
Authority
JP
Japan
Prior art keywords
lower alkyl
cephalosporin derivatives
preparation
substituted
cephem4
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP9584976A
Other languages
English (en)
Japanese (ja)
Other versions
JPS5653312B2 (enExample
Inventor
Senji Kakeya
Yoshinobu Yoshimura
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Priority to JP9584976A priority Critical patent/JPS5321192A/ja
Priority to CH954077A priority patent/CH628057A5/de
Priority to FR7724017A priority patent/FR2361406A1/fr
Priority to DE19772735732 priority patent/DE2735732A1/de
Priority to GB7733178A priority patent/GB1542051A/en
Publication of JPS5321192A publication Critical patent/JPS5321192A/ja
Priority to US06/076,545 priority patent/US4260607A/en
Publication of JPS5653312B2 publication Critical patent/JPS5653312B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP9584976A 1976-08-10 1976-08-10 Cephalosporin derivatives and their preparation Granted JPS5321192A (en)

Priority Applications (6)

Application Number Priority Date Filing Date Title
JP9584976A JPS5321192A (en) 1976-08-10 1976-08-10 Cephalosporin derivatives and their preparation
CH954077A CH628057A5 (de) 1976-08-10 1977-08-03 Verfahren zur herstellung eines cephalosporin-derivates.
FR7724017A FR2361406A1 (fr) 1976-08-10 1977-08-04 Esters de cephalosporines
DE19772735732 DE2735732A1 (de) 1976-08-10 1977-08-08 Cephalosporinester
GB7733178A GB1542051A (en) 1976-08-10 1977-08-08 Cephalosporin esters
US06/076,545 US4260607A (en) 1976-08-10 1979-09-18 Cephalosporin esters

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP9584976A JPS5321192A (en) 1976-08-10 1976-08-10 Cephalosporin derivatives and their preparation

Publications (2)

Publication Number Publication Date
JPS5321192A true JPS5321192A (en) 1978-02-27
JPS5653312B2 JPS5653312B2 (enExample) 1981-12-17

Family

ID=14148810

Family Applications (1)

Application Number Title Priority Date Filing Date
JP9584976A Granted JPS5321192A (en) 1976-08-10 1976-08-10 Cephalosporin derivatives and their preparation

Country Status (6)

Country Link
US (1) US4260607A (enExample)
JP (1) JPS5321192A (enExample)
CH (1) CH628057A5 (enExample)
DE (1) DE2735732A1 (enExample)
FR (1) FR2361406A1 (enExample)
GB (1) GB1542051A (enExample)

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57123190A (en) * 1980-12-12 1982-07-31 Ciba Geigy Ag Novel esters, manufacture and medicine containing same
JPS5989690A (ja) * 1982-09-30 1984-05-23 Fujisawa Pharmaceut Co Ltd ７−アシルアミノ−３−ビニルセフアロスポラン酸誘導体、その製法およびそれを含有する抗菌剤
JPS59116291A (ja) * 1982-12-06 1984-07-05 Fujisawa Pharmaceut Co Ltd ７−置換−３−セフエム−４−カルボン酸エステルおよびその製法
JPS59190995A (ja) * 1983-04-14 1984-10-29 Takeda Chem Ind Ltd セフアロスポリン誘導体
JPS59184292U (ja) * 1983-05-26 1984-12-07 日立造船株式会社 舟艇の揚収装置
JPS59225193A (ja) * 1983-06-02 1984-12-18 Takeda Chem Ind Ltd セフアロスポリンエステル
JPS59225191A (ja) * 1983-06-02 1984-12-18 Takeda Chem Ind Ltd 経口用セフアロスポリン誘導体
JPS6084292A (ja) * 1983-09-30 1985-05-13 Fujisawa Pharmaceut Co Ltd セフエムエステル化合物の製造法

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS58159496A (ja) * 1983-03-02 1983-09-21 Kyoto Yakuhin Kogyo Kk セフエム系化合物
EP0136266A3 (de) * 1983-09-22 1986-03-26 Ciba-Geigy Ag 7beta-Acylamido-3-cephem-4-carbonsäureester, Verfahren zu ihrer Herstellung, pharmazeutische Präparate, welche diese Verbindungen enthalten, und Verwendung von letzteren
JPS60178891A (ja) * 1984-02-24 1985-09-12 Kureha Chem Ind Co Ltd セファロスポリン誘導体及び該誘導体を含有する医薬
CN101948446B (zh) * 2010-08-30 2013-05-15 江苏华旭药业有限公司 一种2-氨基噻唑-4-基乙酸盐酸盐的制造方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1425933A (en) * 1972-03-13 1976-02-25 Astra Laekemedel Ab Cephalosporins
NZ176206A (en) * 1973-12-25 1978-03-06 Takeda Chemical Industries Ltd Cephalosporins
JPS5119765A (en) * 1974-08-09 1976-02-17 Takeda Chemical Industries Ltd Aminochiazoorujudotaino seizoho

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS57123190A (en) * 1980-12-12 1982-07-31 Ciba Geigy Ag Novel esters, manufacture and medicine containing same
JPS5989690A (ja) * 1982-09-30 1984-05-23 Fujisawa Pharmaceut Co Ltd ７−アシルアミノ−３−ビニルセフアロスポラン酸誘導体、その製法およびそれを含有する抗菌剤
JPS59116291A (ja) * 1982-12-06 1984-07-05 Fujisawa Pharmaceut Co Ltd ７−置換−３−セフエム−４−カルボン酸エステルおよびその製法
JPS59190995A (ja) * 1983-04-14 1984-10-29 Takeda Chem Ind Ltd セフアロスポリン誘導体
JPS59184292U (ja) * 1983-05-26 1984-12-07 日立造船株式会社 舟艇の揚収装置
JPS59225193A (ja) * 1983-06-02 1984-12-18 Takeda Chem Ind Ltd セフアロスポリンエステル
JPS59225191A (ja) * 1983-06-02 1984-12-18 Takeda Chem Ind Ltd 経口用セフアロスポリン誘導体
JPS6084292A (ja) * 1983-09-30 1985-05-13 Fujisawa Pharmaceut Co Ltd セフエムエステル化合物の製造法

Also Published As

Publication number Publication date
GB1542051A (en) 1979-03-14
JPS5653312B2 (enExample) 1981-12-17
DE2735732A1 (de) 1978-02-16
CH628057A5 (de) 1982-02-15
FR2361406A1 (fr) 1978-03-10
US4260607A (en) 1981-04-07
FR2361406B1 (enExample) 1981-06-19

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