JPH036158B2 - - Google Patents
Info
- Publication number
- JPH036158B2 JPH036158B2 JP57011927A JP1192782A JPH036158B2 JP H036158 B2 JPH036158 B2 JP H036158B2 JP 57011927 A JP57011927 A JP 57011927A JP 1192782 A JP1192782 A JP 1192782A JP H036158 B2 JPH036158 B2 JP H036158B2
- Authority
- JP
- Japan
- Prior art keywords
- group
- compound
- here
- formula
- carbon atoms
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by an uninterrupted chain of only two carbon atoms, e.g. pregnane derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
- C07J5/0046—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa
- C07J5/0053—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond substituted in position 17 alfa not substituted in position 16
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8101688A FR2498607A1 (fr) | 1981-01-29 | 1981-01-29 | Nouveau procede de preparation de 17a-hydroxy 17b-hydroxyacetyle steroides, produits intermediaires correspondants et produits finals obtenus |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS57144299A JPS57144299A (en) | 1982-09-06 |
| JPH036158B2 true JPH036158B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1991-01-29 |
Family
ID=9254633
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP57011927A Granted JPS57144299A (en) | 1981-01-29 | 1982-01-29 | Novel manufacture of 17 alpha-hydroxy-17 beta- hydroxyacetylsteroid and corresponding intermediate therefrom |
Country Status (10)
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0123736A1 (en) * | 1983-04-29 | 1984-11-07 | Gist-Brocades N.V. | New process for the preparation of 21-hydroxy-20-keto-delta 16-steroids and new intermediate compounds formed in this process |
| US4910191A (en) * | 1988-06-28 | 1990-03-20 | Merrell Dow Pharmaceuticals Inc. | 19-substituted progesterone derivatives useful as 19-hydroxylase inhibitors |
| US5202316A (en) * | 1989-03-22 | 1993-04-13 | Roussel Uclaf | N,N,N',N'-6-(1-piperazinyl)-2,5-pyridinediamines |
| FR2683530B1 (fr) * | 1991-11-08 | 1994-01-21 | Roussel Uclaf | Nouveau procede de preparation de derives 20-oxo 17 alpha, 21-dihydroxyles du pregnane et nouveaux intermediaires. |
| FR2719588B1 (fr) * | 1994-05-03 | 1996-06-07 | Roussel Uclaf | Nouveau procédé de préparation de la substance "S" et nouveaux intermédiaires. |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3793350A (en) * | 1971-10-01 | 1974-02-19 | Syntex Corp | Process for preparing 17alpha,21-dihydroxy-20-keto-pregnanes,derivatives and intermediates thereof |
| DE2603266A1 (de) * | 1976-01-29 | 1977-08-11 | Hoechst Ag | 17-hydroxyacetylsteroide und verfahren zu ihrer herstellung |
| DE2655104A1 (de) * | 1976-12-04 | 1978-06-08 | Hoechst Ag | Verfahren zur herstellung von 17alpha-hydroxy-21-acetoxy-progesteron |
| DE2704130A1 (de) * | 1977-01-28 | 1978-08-10 | Schering Ag | Verfahren zur herstellung von 17 beta- hydroxy-20-alkoxy-pregnan-21-saeure-derivaten |
| FR2462445A1 (fr) * | 1979-07-31 | 1981-02-13 | Roussel Uclaf | Nouveaux derives 17-/(hydroxymethyl) (formamido) methylene/steroides, leur procede de preparation et leur application a l'introduction de la chaine laterale hydroxyacetyle |
-
1981
- 1981-01-29 FR FR8101688A patent/FR2498607A1/fr active Granted
-
1982
- 1982-01-08 EP EP82400026A patent/EP0058097B1/fr not_active Expired
- 1982-01-08 AT AT82400026T patent/ATE8638T1/de not_active IP Right Cessation
- 1982-01-08 DE DE8282400026T patent/DE3260408D1/de not_active Expired
- 1982-01-26 FI FI820240A patent/FI77462C/fi not_active IP Right Cessation
- 1982-01-27 US US06/343,357 patent/US4565656A/en not_active Expired - Fee Related
- 1982-01-27 PT PT74343A patent/PT74343B/pt not_active IP Right Cessation
- 1982-01-28 DK DK37782A patent/DK37782A/da not_active Application Discontinuation
- 1982-01-28 HU HU82259A patent/HU187843B/hu not_active IP Right Cessation
- 1982-01-29 JP JP57011927A patent/JPS57144299A/ja active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| US4565656A (en) | 1986-01-21 |
| JPS57144299A (en) | 1982-09-06 |
| FR2498607A1 (fr) | 1982-07-30 |
| FI77462C (fi) | 1989-03-10 |
| HU187843B (en) | 1986-02-28 |
| ATE8638T1 (de) | 1984-08-15 |
| PT74343B (fr) | 1984-05-30 |
| EP0058097A2 (fr) | 1982-08-18 |
| DK37782A (da) | 1982-07-30 |
| PT74343A (fr) | 1982-02-01 |
| FR2498607B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1983-07-29 |
| EP0058097A3 (en) | 1982-10-27 |
| FI820240L (fi) | 1982-07-30 |
| FI77462B (fi) | 1988-11-30 |
| DE3260408D1 (en) | 1984-08-30 |
| EP0058097B1 (fr) | 1984-07-25 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| SU1340593A3 (ru) | Способ получени производных @ @ 19-норстероидов | |
| EP0057115A2 (fr) | Nouveaux dérivés stéroides substitués en 11beta, procédé de préparation, leur application comme médicament et les compositions les renfermant | |
| PT85891B (pt) | Processo para a preparacao de 9-alfa-hidroxi-esteroides e dos respectivos derivados 9(11)-deidro bem como de composicoes farmaceuticas que os contem | |
| AU725606B2 (en) | Process for the preparation of 17-esters of 9alpha,21- dihalo-pregnane-11beta,17alpha-diol-20-ones | |
| EP0023856B1 (fr) | Dérivés 17-((hydroxyméthyl)(formamido) méthylène) stéroides, leur préparation, leur application à l'introduction de la chaîne latérale hydroxyacétyle | |
| EP1242444B1 (en) | Process for preparing 17alpha-acetoxy-11beta- 4-n,n-(dimethylamino)phenyl]-21-methoxy-19-norpregna-4,9-diene-3,20-dione, intermediates useful in the process, and processes for preparing such intermediates | |
| EP0176399B1 (fr) | Nouveaux stéroides substitués en position 10 par un radical comportant une double ou triple liaison, leur procédé de préparation, leur application comme médicaments, les compositions pharmaceutiques les renfermant | |
| JPH0440360B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| JPH036158B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| US5998639A (en) | Sulfatation of estrogen mixtures | |
| JPH0276896A (ja) | ステロイド化合物およびその製造方法 | |
| EP0181442B1 (de) | Verfahren zur Herstellung von Pregnan-Derivaten | |
| JP3037508B2 (ja) | プレグナ−１，４−ジエン−３，２０−ジオンの新規な置換された１６−メチルステロイド誘導体、それらの製造法、それらの１６−メチレンステロイドの製造への用途及び新規な中間体 | |
| JPH0320399B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| JPH0776231B2 (ja) | １７α―エチニル―１７β―ヒドロキシ―１８―メチル―４，１５―エストラジエン―３―オンの製法 | |
| EP0110434B1 (fr) | Nouveaux produits intermédiaires stéroides substitués en 11-beta et procédé de préparation de ces produits | |
| JP4361976B2 (ja) | エストロゲン混合物の硫酸化 | |
| US4585591A (en) | 17β-ethynylsteroids and process for preparing same | |
| JPS641480B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| JPS6210238B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| JPH0153680B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| JPS6360038B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| JPS6353995B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| JPS6352637B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | ||
| JPH0148917B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) |