JPH0317824B2 - - Google Patents

Info

Publication number
JPH0317824B2
JPH0317824B2 JP63086213A JP8621388A JPH0317824B2 JP H0317824 B2 JPH0317824 B2 JP H0317824B2 JP 63086213 A JP63086213 A JP 63086213A JP 8621388 A JP8621388 A JP 8621388A JP H0317824 B2 JPH0317824 B2 JP H0317824B2
Authority
JP
Japan
Prior art keywords
adpoc
bzl
thr
formula
phe
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP63086213A
Other languages
English (en)
Japanese (ja)
Other versions
JPS6452748A (en
Inventor
Karubatsuhaa Hyuubaato
Borutaa Borufugangu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of JPS6452748A publication Critical patent/JPS6452748A/ja
Publication of JPH0317824B2 publication Critical patent/JPH0317824B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • C07K5/06156—Dipeptides with the first amino acid being heterocyclic and Trp-amino acid; Derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D209/20—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals substituted additionally by nitrogen atoms, e.g. tryptophane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
    • C07K1/063—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for alpha-amino functions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
    • C07K1/064—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for omega-amino or -guanidino functions
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C07K1/061—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
    • C07K1/068—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for heterocyclic side chains
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/655—Somatostatins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
    • C07K5/1013—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing O or S as heteroatoms, e.g. Cys, Ser

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Analytical Chemistry (AREA)
  • Endocrinology (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP63086213A 1978-09-07 1988-04-06 Urethanes of novel substituted carbonic acid Granted JPS6452748A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
LU80207A LU80207A1 (de) 1978-09-07 1978-09-07 Neue substituierte kohlensaeureester und urethane,verfahren zu ihrer herstellung und deren verwendung

Publications (2)

Publication Number Publication Date
JPS6452748A JPS6452748A (en) 1989-02-28
JPH0317824B2 true JPH0317824B2 (enExample) 1991-03-11

Family

ID=19728996

Family Applications (2)

Application Number Title Priority Date Filing Date
JP54115646A Expired - Lifetime JPH0662511B2 (ja) 1978-09-07 1979-09-07 新規な置換炭酸のエステル類及びそれらの製造法
JP63086213A Granted JPS6452748A (en) 1978-09-07 1988-04-06 Urethanes of novel substituted carbonic acid

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP54115646A Expired - Lifetime JPH0662511B2 (ja) 1978-09-07 1979-09-07 新規な置換炭酸のエステル類及びそれらの製造法

Country Status (6)

Country Link
US (1) US4440692A (enExample)
EP (1) EP0010587B1 (enExample)
JP (2) JPH0662511B2 (enExample)
AT (1) ATE3634T1 (enExample)
DE (1) DE2965574D1 (enExample)
LU (1) LU80207A1 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
LU80207A1 (de) * 1978-09-07 1980-04-21 H Kalbacher Neue substituierte kohlensaeureester und urethane,verfahren zu ihrer herstellung und deren verwendung
FR2559764B1 (fr) * 1984-02-16 1988-01-29 Poudres & Explosifs Ste Nale Nouveaux carbonates a-chlores, leur procede de fabrication et leur application a la protection des fonctions amine des amino-acides
US4818704A (en) * 1986-05-16 1989-04-04 Eka Nobel Ab Method for the separation and determination of enantiomeric amine compounds using an optically active agent
US4713480A (en) * 1987-01-07 1987-12-15 Ortho Pharmaceutical Corporation Method for the production of crystalline amino-protected-beta-benzyl-L-aspartic acid
GB8900376D0 (en) * 1989-01-09 1989-03-08 Nycomed As Iodinated esters
US5175333A (en) * 1990-09-14 1992-12-29 Lever Brothers Company, Division Of Conopco, Inc. Transesterification route to quaternary ammonium substituted carbonate esters
KR20010014005A (ko) * 1998-04-21 2001-02-26 고지마 아끼로, 오가와 다이스께 아다만탄메탄올 유도체 및 그의 제조 방법
JP4503109B2 (ja) * 1999-02-09 2010-07-14 ダイセル化学工業株式会社 重合性脂環式化合物
KR100584810B1 (ko) * 2002-06-11 2006-05-30 주식회사 이엔에프테크놀로지 비닐 알킬(1-아다만틸) 에테르 및 그 제조방법
GB2402132B (en) * 2003-05-28 2005-10-19 Reckitt Benckiser Nv Dishwasher anti-corrosion composition
PL1673426T3 (pl) * 2003-10-17 2008-07-31 Reckitt Benckiser Finish Bv Kompozycja ochronna do wyrobów szklanych w zmywarkach

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1050422A (enExample) * 1963-03-06
NL130998C (enExample) * 1965-01-21
DE1930330A1 (de) * 1969-06-14 1970-12-17 Hoechst Ag Cysteinhaltige Peptide und deren Derivate und Verfahren zu ihrer Herstellung
DE1924802A1 (de) * 1969-05-14 1970-11-19 Hoechst Ag Verfahren zur Herstellung argininhaltiger Peptiden
US3705213A (en) * 1969-07-01 1972-12-05 Smith Kline French Lab Adamantoyl and adamantyl (alkyl) glycerophosphoryl (and phosphonyl)ethanolamines
DE2063087A1 (de) * 1969-12-29 1971-08-19 Eli Lilly and Co , Indianapolis, Ind (V St A) Histidin und Tryptophanderivate
IE46462B1 (en) * 1977-02-22 1983-06-15 American Home Prod Somatostatin peptide analogues
LU80207A1 (de) * 1978-09-07 1980-04-21 H Kalbacher Neue substituierte kohlensaeureester und urethane,verfahren zu ihrer herstellung und deren verwendung

Also Published As

Publication number Publication date
DE2965574D1 (en) 1983-07-07
US4440692A (en) 1984-04-03
JPS6452748A (en) 1989-02-28
JPS5543087A (en) 1980-03-26
JPH0662511B2 (ja) 1994-08-17
ATE3634T1 (de) 1983-06-15
EP0010587A1 (de) 1980-05-14
EP0010587B1 (de) 1983-06-01
LU80207A1 (de) 1980-04-21

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