JPH0254348B2 - - Google Patents

Info

Publication number
JPH0254348B2
JPH0254348B2 JP56036521A JP3652181A JPH0254348B2 JP H0254348 B2 JPH0254348 B2 JP H0254348B2 JP 56036521 A JP56036521 A JP 56036521A JP 3652181 A JP3652181 A JP 3652181A JP H0254348 B2 JPH0254348 B2 JP H0254348B2
Authority
JP
Japan
Prior art keywords
formula
group
syn
alkyl group
lower alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP56036521A
Other languages
English (en)
Japanese (ja)
Other versions
JPS57154175A (en
Inventor
Isao Sakano
Tatsuro Yokoyama
Seitaro Kajitani
Yutaka Okazaki
Hiroshi Tokuda
Hiroshi Kawamo
Mikio Kumakura
Okao Nakano
Akira Awaya
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mitsui Toatsu Chemicals Inc
Original Assignee
Mitsui Toatsu Chemicals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsui Toatsu Chemicals Inc filed Critical Mitsui Toatsu Chemicals Inc
Priority to JP56036521A priority Critical patent/JPS57154175A/ja
Priority to GB08232545A priority patent/GB2110674B/en
Priority to PCT/JP1982/000071 priority patent/WO1982003217A1/ja
Priority to EP82900830A priority patent/EP0075600B1/en
Priority to DE3237438T priority patent/DE3237438C2/de
Publication of JPS57154175A publication Critical patent/JPS57154175A/ja
Priority to US06/568,826 priority patent/US4532137A/en
Publication of JPH0254348B2 publication Critical patent/JPH0254348B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
JP56036521A 1981-03-16 1981-03-16 2-thiazoleamine derivative, its preparation, and drug composition comprising it Granted JPS57154175A (en)

Priority Applications (6)

Application Number Priority Date Filing Date Title
JP56036521A JPS57154175A (en) 1981-03-16 1981-03-16 2-thiazoleamine derivative, its preparation, and drug composition comprising it
GB08232545A GB2110674B (en) 1981-03-16 1982-03-16 2-thiazoleamine derivatives, process for their preparation, and medicinal composition containing same
PCT/JP1982/000071 WO1982003217A1 (en) 1981-03-16 1982-03-16 2-thiazoleamine derivatives,process for their preparation,and medicinal composition containing same
EP82900830A EP0075600B1 (en) 1981-03-16 1982-03-16 2-thiazoleamine derivatives, process for their preparation, and medicinal composition containing same
DE3237438T DE3237438C2 (de) 1981-03-16 1982-03-16 2-Thiazolamin-Derivate und dieselben enthaltende pharmazeutische Zusammensetzungen
US06/568,826 US4532137A (en) 1981-03-16 1984-01-06 2-Thiazolamine derivatives, process for preparing same, and pharmaceutical compositions comprising same

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP56036521A JPS57154175A (en) 1981-03-16 1981-03-16 2-thiazoleamine derivative, its preparation, and drug composition comprising it

Publications (2)

Publication Number Publication Date
JPS57154175A JPS57154175A (en) 1982-09-22
JPH0254348B2 true JPH0254348B2 (en, 2012) 1990-11-21

Family

ID=12472115

Family Applications (1)

Application Number Title Priority Date Filing Date
JP56036521A Granted JPS57154175A (en) 1981-03-16 1981-03-16 2-thiazoleamine derivative, its preparation, and drug composition comprising it

Country Status (6)

Country Link
US (1) US4532137A (en, 2012)
EP (1) EP0075600B1 (en, 2012)
JP (1) JPS57154175A (en, 2012)
DE (1) DE3237438C2 (en, 2012)
GB (1) GB2110674B (en, 2012)
WO (1) WO1982003217A1 (en, 2012)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DD283621A5 (de) * 1989-04-20 1990-10-17 �����������@�������������@����������@��@������k�� Verfahren zur herstellung von azylureidoaminothiazoly-abkoemmlingen

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5760345B2 (en, 2012) * 1974-12-19 1982-12-18 Takeda Chemical Industries Ltd
US4203899A (en) * 1974-12-19 1980-05-20 Takeda Chemical Industries, Ltd. Thiazolylacetamido compounds
DK154939C (da) * 1974-12-19 1989-06-12 Takeda Chemical Industries Ltd Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
GB1536281A (en) * 1975-06-09 1978-12-20 Takeda Chemical Industries Ltd Cephem compounds
SE440655B (sv) * 1976-01-23 1985-08-12 Roussel Uclaf Sett att framstella nya oximderivat av 7-amino-tiazolyl-acetamido-cefalosporansyra
US4166115A (en) * 1976-04-12 1979-08-28 Fujisawa Pharmaceutical Co., Ltd. Syn 7-oxoimino substituted derivatives of cephalosporanic acid
GB1576625A (en) * 1976-04-12 1980-10-08 Fujisawa Pharmaceutical Co Syn isomer 3,7 disubstituted 3 cephem 4 carboxylic acid compounds and processes for the preparation thereof
US4304770A (en) * 1976-04-12 1981-12-08 Fujisawa Pharmaceutical Co., Ltd. Syn-isomer of 3,7-disubstituted-3-cephem-4-carboxylic acid compounds and processes for the preparation thereof
DE2714880A1 (de) * 1977-04-02 1978-10-26 Hoechst Ag Cephemderivate und verfahren zu ihrer herstellung
FR2406634A1 (fr) * 1977-10-19 1979-05-18 Fabre Sa Pierre Immunostimulants derives d'amino thiazoles
US4217355A (en) * 1978-04-24 1980-08-12 Pfizer Inc. Amide therapeutic agents
DK150068C (da) * 1978-06-02 1987-06-29 Pfizer Analogifremgangsmaade til fremstilling af aminothiazoler
DE2826482A1 (de) * 1978-06-16 1980-01-03 Bayer Ag Beta -lactam-verbindungen
EP0009008A3 (de) * 1978-09-08 1980-05-14 Ciba-Geigy Ag Cephalosporinderivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Präparate
AU518218B2 (en) * 1978-10-16 1981-09-17 Takeda Chemical Industries Ltd. Thiazolylacetic acid compounds
US4313945A (en) * 1978-11-23 1982-02-02 Ciba-Geigy Corporation 7-Thiazolyl-acetamido-cephem derivatives with terminal aminocarboxylic acid grouping
JPS56100772A (en) * 1980-01-18 1981-08-12 Denki Kagaku Kogyo Kk Preparation of 2- 2-aminothiazol-4-yl -2-alkoxyiminoacetic acid derivative

Also Published As

Publication number Publication date
EP0075600A4 (en) 1983-05-16
US4532137A (en) 1985-07-30
EP0075600A1 (en) 1983-04-06
WO1982003217A1 (en) 1982-09-30
JPS57154175A (en) 1982-09-22
EP0075600B1 (en) 1986-12-30
GB2110674A (en) 1983-06-22
GB2110674B (en) 1985-04-17
DE3237438C2 (de) 1985-02-14
DE3237438T1 (de) 1983-12-01

Similar Documents

Publication Publication Date Title
US4225610A (en) Immunoactivators derived from amino thiazoles
KR930009790B1 (ko) 벤조티아졸 및 그를 유효성분으로 함유하는 항류머티스제
US3852293A (en) 4-phenyl-2-(3-pyridyl)-thiazole carboxamides
EP0069784B1 (en) Thiazolylurea derivatives, process for their preparation, and medicinal composition containing same
NZ188770A (en) Thiazolinylguanidine derivatives and pharmaceutical compositions
JPS6324514B2 (en, 2012)
US3896223A (en) Anti-inflammatory thiazole compositions and methods for using same
US4501750A (en) Thiazole compounds, a process for preparing same and a pharmaceutical composition containing the thiazole compounds
US3852292A (en) 2-(pyridyl)-imidazole-4,5-dicarboxylic acid and derivatives
JPH0254348B2 (en, 2012)
JPH01228975A (ja) ベンゾチアジン―１，１―ジオキシド誘導体及びそれを含有する医薬組成物
US4301167A (en) 2-Amino thiazoline derivatives
JPH0135831B2 (en, 2012)
US4348403A (en) 2-Amino-4-(4-benzyloxyphenyl)thiazoles, and their use in hyperlipemia
JPH0260670B2 (en, 2012)
JPH0254347B2 (en, 2012)
JPS6254306B2 (en, 2012)
EP0068033B1 (en) N-(4-phenyl-2-thiazolyl)carbamate derivatives, process for their preparation, and medicinal composition containing same
JPH0254354B2 (en, 2012)
JPH0255426B2 (en, 2012)
JPS6345669B2 (en, 2012)
JPH0255427B2 (en, 2012)
JPH0255428B2 (en, 2012)
JP2804276B2 (ja) イミダゾ［２，１―ｂ］チアゾール類
JPH0260672B2 (en, 2012)