JPH0225465A - ピペリジン誘導体、その製造方法並びにそれを含む抗ヒスタミン剤 - Google Patents

ピペリジン誘導体、その製造方法並びにそれを含む抗ヒスタミン剤

Info

Publication number
JPH0225465A
JPH0225465A JP17514288A JP17514288A JPH0225465A JP H0225465 A JPH0225465 A JP H0225465A JP 17514288 A JP17514288 A JP 17514288A JP 17514288 A JP17514288 A JP 17514288A JP H0225465 A JPH0225465 A JP H0225465A
Authority
JP
Japan
Prior art keywords
group
formula
lower alkyl
general formula
tables
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP17514288A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0533953B2 (enrdf_load_stackoverflow
Inventor
Shoei Eda
江田　昭英
Junichiro Kita
淳一郎 北
Shinji Takamura
真司 高村
Kayoko Yamano
山野　佳代子
Hiroshi Fujiwara
寛 藤原
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Ube Corp
Original Assignee
Ube Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=15991022&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JPH0225465(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ube Industries Ltd filed Critical Ube Industries Ltd
Priority to JP17514288A priority Critical patent/JPH0225465A/ja
Priority to US07/325,306 priority patent/US4929618A/en
Priority to CA000594067A priority patent/CA1340207C/en
Priority to DE89302894T priority patent/DE68906816T2/de
Priority to EP89302894A priority patent/EP0335586B1/en
Priority to ES89302894T priority patent/ES2058504T3/es
Publication of JPH0225465A publication Critical patent/JPH0225465A/ja
Publication of JPH0533953B2 publication Critical patent/JPH0533953B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP17514288A 1988-03-25 1988-07-15 ピペリジン誘導体、その製造方法並びにそれを含む抗ヒスタミン剤 Granted JPH0225465A (ja)

Priority Applications (6)

Application Number Priority Date Filing Date Title
JP17514288A JPH0225465A (ja) 1988-07-15 1988-07-15 ピペリジン誘導体、その製造方法並びにそれを含む抗ヒスタミン剤
US07/325,306 US4929618A (en) 1988-03-25 1989-03-16 Piperdine and piperazine derivatives, and antihistaminic pharmaceutical compositions containing the same
CA000594067A CA1340207C (en) 1988-03-25 1989-03-17 Piperidine and piperazine derivatives, process for preparing the same and pharmaceutical compositions containing the same
DE89302894T DE68906816T2 (de) 1988-03-25 1989-03-22 Piperidin- und Piperazinderivate, Verfahren zu ihrer Herstellung und pharmazeutische Zusammensetzungen, die sie enthalten.
EP89302894A EP0335586B1 (en) 1988-03-25 1989-03-22 Piperidine & piperazine derivatives, process for preparing the same and pharmaceutical compositions containing the same
ES89302894T ES2058504T3 (es) 1988-03-25 1989-03-22 Derivados de piperidina y piperazina, procedimiento para preparar los mismos, y composiciones farmaceuticas que contienen los mismos.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP17514288A JPH0225465A (ja) 1988-07-15 1988-07-15 ピペリジン誘導体、その製造方法並びにそれを含む抗ヒスタミン剤

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP28722891A Division JP2625294B2 (ja) 1991-10-08 1991-10-08 ピペリジン誘導体

Publications (2)

Publication Number Publication Date
JPH0225465A true JPH0225465A (ja) 1990-01-26
JPH0533953B2 JPH0533953B2 (enrdf_load_stackoverflow) 1993-05-20

Family

ID=15991022

Family Applications (1)

Application Number Title Priority Date Filing Date
JP17514288A Granted JPH0225465A (ja) 1988-03-25 1988-07-15 ピペリジン誘導体、その製造方法並びにそれを含む抗ヒスタミン剤

Country Status (1)

Country Link
JP (1) JPH0225465A (enrdf_load_stackoverflow)

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5153207A (en) * 1989-05-22 1992-10-06 Hokuriku Pharmaceutical Co., Ltd. Piperidine derivative, method for preparation thereof, and a pharmaceutical composition comprising the same
JP2000198784A (ja) * 1996-12-26 2000-07-18 Ube Ind Ltd 光学活性ピペリジン誘導体の酸付加塩及びその製法
JP2004051600A (ja) * 2002-07-24 2004-02-19 Iyaku Bunshi Sekkei Kenkyusho:Kk 造血器型プロスタグランジンｄ２合成酵素阻害剤
JPWO2003057675A1 (ja) * 2001-12-28 2005-05-19 興和株式会社 環状ジアミン化合物又はその塩の製造法
WO2008153289A3 (en) * 2007-06-11 2009-03-05 Hanmi Pharm Ind Co Ltd Process for preparing bepotastine and intermediates used therein
JP2012025705A (ja) * 2010-07-26 2012-02-09 Tokuyama Corp （ｓ）−４−〔（４−クロロフェニル）（２−ピリジル）メトキシ〕ピペリジンのジアステレオマー塩の製造方法
JP2012240982A (ja) * 2011-05-23 2012-12-10 Toray Fine Chemicals Co Ltd 光学活性ピペリジン誘導体のベンゼンスルホン酸塩の製造方法

Cited By (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5153207A (en) * 1989-05-22 1992-10-06 Hokuriku Pharmaceutical Co., Ltd. Piperidine derivative, method for preparation thereof, and a pharmaceutical composition comprising the same
JP2000198784A (ja) * 1996-12-26 2000-07-18 Ube Ind Ltd 光学活性ピペリジン誘導体の酸付加塩及びその製法
JP2007145852A (ja) * 1996-12-26 2007-06-14 Ube Ind Ltd 光学活性ピペリジン誘導体の酸付加塩及びその製法
JP2011063619A (ja) * 1996-12-26 2011-03-31 Ube Industries Ltd 光学活性ピペリジン誘導体の酸付加塩及びその製法
JP2012180360A (ja) * 1996-12-26 2012-09-20 Ube Industries Ltd 光学活性ピペリジン誘導体の酸付加塩及びその製法
JPWO2003057675A1 (ja) * 2001-12-28 2005-05-19 興和株式会社 環状ジアミン化合物又はその塩の製造法
JP2004051600A (ja) * 2002-07-24 2004-02-19 Iyaku Bunshi Sekkei Kenkyusho:Kk 造血器型プロスタグランジンｄ２合成酵素阻害剤
WO2008153289A3 (en) * 2007-06-11 2009-03-05 Hanmi Pharm Ind Co Ltd Process for preparing bepotastine and intermediates used therein
JP2012025705A (ja) * 2010-07-26 2012-02-09 Tokuyama Corp （ｓ）−４−〔（４−クロロフェニル）（２−ピリジル）メトキシ〕ピペリジンのジアステレオマー塩の製造方法
JP2012240982A (ja) * 2011-05-23 2012-12-10 Toray Fine Chemicals Co Ltd 光学活性ピペリジン誘導体のベンゼンスルホン酸塩の製造方法

Also Published As

Publication number Publication date
JPH0533953B2 (enrdf_load_stackoverflow) 1993-05-20

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