JP7364663B2 - イミダゾ［４，５－ｃ］キノリン誘導体のＮＬＲＰ３モジュレーター - Google Patents
イミダゾ［４，５－ｃ］キノリン誘導体のＮＬＲＰ３モジュレーター Download PDFInfo
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- JP7364663B2 JP7364663B2 JP2021507787A JP2021507787A JP7364663B2 JP 7364663 B2 JP7364663 B2 JP 7364663B2 JP 2021507787 A JP2021507787 A JP 2021507787A JP 2021507787 A JP2021507787 A JP 2021507787A JP 7364663 B2 JP7364663 B2 JP 7364663B2
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- A61K39/39533—Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
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- Nitrogen Condensed Heterocyclic Rings (AREA)
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| PCT/US2019/046591 WO2020037091A1 (en) | 2018-08-16 | 2019-08-15 | Imidazo[4,5-c]quinoline derived nlrp3-modulators |
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| JP2021534168A JP2021534168A (ja) | 2021-12-09 |
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| US20210269434A1 (en) * | 2020-01-10 | 2021-09-02 | Incyte Corporation | Tricyclic compounds as inhibitors of kras |
| WO2021150613A1 (en) | 2020-01-20 | 2021-07-29 | Incyte Corporation | Spiro compounds as inhibitors of kras |
| CA3179692A1 (en) * | 2020-04-16 | 2021-10-21 | Incyte Corporation | Fused tricyclic kras inhibitors |
| US11739102B2 (en) | 2020-05-13 | 2023-08-29 | Incyte Corporation | Fused pyrimidine compounds as KRAS inhibitors |
| US11999752B2 (en) | 2020-08-28 | 2024-06-04 | Incyte Corporation | Vinyl imidazole compounds as inhibitors of KRAS |
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| WO2022204112A1 (en) | 2021-03-22 | 2022-09-29 | Incyte Corporation | Imidazole and triazole kras inhibitors |
| CN115124524A (zh) * | 2021-03-26 | 2022-09-30 | 浙江海正药业股份有限公司 | 三环类衍生物及其制备方法和用途 |
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