JP6876058B2 - フェニルウレア化合物及びその用途 - Google Patents
フェニルウレア化合物及びその用途 Download PDFInfo
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- JP6876058B2 JP6876058B2 JP2018535748A JP2018535748A JP6876058B2 JP 6876058 B2 JP6876058 B2 JP 6876058B2 JP 2018535748 A JP2018535748 A JP 2018535748A JP 2018535748 A JP2018535748 A JP 2018535748A JP 6876058 B2 JP6876058 B2 JP 6876058B2
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- disease
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- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
- A01N47/30—Derivatives containing the group >N—CO—N aryl or >N—CS—N—aryl
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/69—Two or more oxygen atoms
Description
本発明はフェニルウレア化合物及びその用途に関する。
液体担体としては、例えば、水、アルコール類(メタノール、エタノール等)、ケトン類(アセトン、メチルエチルケトン等)、芳香族炭化水素類(トルエン、キシレン、エチルベンゼン、メチルナフタレン等)、脂肪族炭化水素類(ヘキサン、シクロヘキサン、灯油等)、エステル類(酢酸エチル、酢酸ブチル等)、ニトリル類(アセトニトリル、イソブチルニトリル等)、エーテル類(ジイソプロピルエーテル等)、アミド類(ジメチルホルムアミド、ジメチルアセトアミド等)、及びスルホキシド類(ジメチルスルホキシド等)が挙げられる。
本発明の防除方法における本発明化合物の処理量は、処理する植物の種類、防除対象である植物病害の種類や発生頻度、製剤形態、処理時期、処理方法、処理場所、気象条件等によっても異なるが、植物の茎葉に処理する場合又は植物を栽培する土壌に処理する場合は、本発明化合物は、1000m2あたり、通常1〜500gである。
乳剤、水和剤、フロアブル剤等は通常水で希釈して散布することにより処理する。この場合、本発明化合物の濃度は、通常0.0005〜2重量%である。粉剤、粒剤等は通常希釈することなくそのまま処理する。
Aspergillus属、Penicillium属、Fusarium属、Gibberella属、Tricoderma属、Thielaviopsis属、Rhizopus属、Mucor属、Corticium属、Phoma属、Rhizoctonia属、及びDiplodia属菌等によって引き起こされる、各種作物の種子病害又は生育初期の病害。Polymixa属又はOlpidium属等によって媒介される各種作物のウイルス病。
イネの苗立枯細菌病(Burkholderia plantarii);キュウリの灰色疫病(Phytophthora capsici)、苗立枯病(Pythium ultimum)および斑点細菌病(Pseudomonas syringae pv. Lachrymans);ナスの青枯病(Ralstonia solanacearum);カンキツのかいよう病(Xanthomonas citiri);ハクサイの軟腐病(Erwinia carotovora)等。
1H−NMR (DMSO−D6) δ (ppm): 8.56 (1H, d, J = 2.0 Hz), 7.91 (1H, d, J = 7.7 Hz), 7.87 (1H, dd, J = 5.0, 1.4 Hz), 7.56 (1H, d, J = 10.9 Hz), 7.21 (1H, dd, J = 7.9, 1.4 Hz), 6.99 (1H, dd, J = 7.9, 5.0 Hz), 6.24 (2H, s), 4.93 (2H, s), 4.10 (2H, q, J = 7.1 Hz) , 1.15 (3H, t, J = 7.1 Hz).
本発明化合物4.5mgをジメチルスルホキシド100μLで希釈した。希釈液1μLをタイタープレート(96ウェル)に分注したのち、キュウリ灰色疫病菌(Phytophthora capsici)の遊走子を含むジャガイモ煎汁液体培地(PDB培地)を150μL分注した。このプレートを3日間、27℃で培養してキュウリ灰色疫病菌を増殖させたのち、タイタープレートの各ウェルの600nmの吸光度を測定し、キュウリ灰色疫病菌の生育度とした。その生育度をもとに、「式1」を用いて効力を算出したところ、本発明化合物の効力は90%以上であった。
「式1」
効力=100×(X−Y)/X
X:無処理区の菌の生育度
Y:処理区の菌の生育度
なお、本試験例における無処理区とは、本発明化合物を含有するジメチルスルホキシド希釈液の代わりにジメチルスルホキシドを分注する以外は処理区と同じ条件で行った試験区を表す。
一方、欧州特許第1122244号明細書に記載のN−[4−クロロ−2−フルオロ−5−{2−(エトキシカルボニル)メトキシ−3−ピリジルオキシ}フェニル]アセトアミドを用いて同じ試験を行った結果、その効力は50%未満であった。
Claims (4)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2016165422 | 2016-08-26 | ||
JP2016165422 | 2016-08-26 | ||
PCT/JP2017/030246 WO2018038188A1 (ja) | 2016-08-26 | 2017-08-24 | フェニルウレア化合物及びその用途 |
Publications (2)
Publication Number | Publication Date |
---|---|
JPWO2018038188A1 JPWO2018038188A1 (ja) | 2019-06-24 |
JP6876058B2 true JP6876058B2 (ja) | 2021-05-26 |
Family
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Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP2018535748A Active JP6876058B2 (ja) | 2016-08-26 | 2017-08-24 | フェニルウレア化合物及びその用途 |
Country Status (10)
Country | Link |
---|---|
US (1) | US10624343B2 (ja) |
JP (1) | JP6876058B2 (ja) |
CN (1) | CN109563042B (ja) |
AR (1) | AR109405A1 (ja) |
AU (1) | AU2017316907B2 (ja) |
BR (1) | BR112019002247B1 (ja) |
CA (1) | CA3035001A1 (ja) |
DE (1) | DE112017004271T5 (ja) |
MX (1) | MX2019002233A (ja) |
WO (1) | WO2018038188A1 (ja) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN114787131A (zh) * | 2019-12-11 | 2022-07-22 | 住友化学株式会社 | 吡啶氧基乙酸化合物及其用途 |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA811752B (en) * | 1980-03-18 | 1982-04-28 | Ciba Geigy Ag | Novel ureas haviang herbicidal activity |
US4376646A (en) | 1980-03-18 | 1983-03-15 | Ciba-Geigy Corporation | Herbicidal N-[4-(3'-alkoxyphenoxy)-phenyl]-N'-methylureas |
JPS60142958A (ja) * | 1983-12-01 | 1985-07-29 | バスフ アクチェン ゲゼルシャフト | キノリンオキシフエニル尿素、その製法及び該化合物を含有する除草剤 |
DE3418532A1 (de) * | 1983-12-01 | 1985-06-13 | Basf Ag, 6700 Ludwigshafen | Chinolinoxyphenylharnstoffe, verfahren zu ihrer herstellung und ihre verwendung zur bekaempfung unerwuenschten pflanzenwuchses |
BR9808334A (pt) | 1997-03-14 | 2000-05-16 | Isk Americas Inc | éteres diarìlicos, processos para sua preparação e composições herbicidas e dessecantes contendo os mesmos |
IL141034A0 (en) * | 2000-02-04 | 2002-02-10 | Sumitomo Chemical Co | Uracil compounds and use thereof |
FR2812633A1 (fr) | 2000-08-04 | 2002-02-08 | Aventis Cropscience Sa | Derives de phenyl(thio)urees et phenyl(thio)carbamates fongicides |
CA2588389A1 (en) | 2004-11-23 | 2006-06-22 | Ptc Therapeutics, Inc. | Substituted phenols as active agents inhibiting vegf production |
UY30117A1 (es) | 2006-01-31 | 2007-06-29 | Tanabe Seiyaku Co | Compuesto amina trisustituido |
JP6456196B2 (ja) | 2015-03-10 | 2019-01-23 | テルモ株式会社 | 抗血栓性接着用組成物、ならびに該抗血栓性接着用組成物を利用した医療用具およびその製造方法 |
MX2019002234A (es) * | 2016-08-26 | 2019-06-17 | Sumitomo Chemical Co | Compuesto de 1-fenil-3-carbamoil urea y uso del mismo. |
DE112017004275T5 (de) * | 2016-08-26 | 2019-05-09 | Sumitomo Chemical Company, Limited | 1-acetyl-3-phenylharnstoffverbindung und deren verwendung |
-
2017
- 2017-08-24 AR ARP170102342A patent/AR109405A1/es active IP Right Grant
- 2017-08-24 CN CN201780051329.2A patent/CN109563042B/zh active Active
- 2017-08-24 DE DE112017004271.2T patent/DE112017004271T5/de active Pending
- 2017-08-24 CA CA3035001A patent/CA3035001A1/en active Pending
- 2017-08-24 MX MX2019002233A patent/MX2019002233A/es unknown
- 2017-08-24 WO PCT/JP2017/030246 patent/WO2018038188A1/ja active Application Filing
- 2017-08-24 US US16/328,010 patent/US10624343B2/en active Active
- 2017-08-24 JP JP2018535748A patent/JP6876058B2/ja active Active
- 2017-08-24 AU AU2017316907A patent/AU2017316907B2/en active Active
- 2017-08-24 BR BR112019002247-3A patent/BR112019002247B1/pt active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
MX2019002233A (es) | 2019-06-17 |
WO2018038188A1 (ja) | 2018-03-01 |
AU2017316907B2 (en) | 2020-11-19 |
CN109563042B (zh) | 2021-12-07 |
DE112017004271T5 (de) | 2019-05-16 |
CN109563042A (zh) | 2019-04-02 |
CA3035001A1 (en) | 2018-03-01 |
AU2017316907A1 (en) | 2019-02-21 |
AR109405A1 (es) | 2018-11-28 |
US10624343B2 (en) | 2020-04-21 |
BR112019002247B1 (pt) | 2022-11-22 |
JPWO2018038188A1 (ja) | 2019-06-24 |
BR112019002247A2 (pt) | 2019-05-14 |
US20190223435A1 (en) | 2019-07-25 |
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