JP6483148B2 - ＨＰＴＰ−β阻害剤 - Google Patents

ＨＰＴＰ−β阻害剤 Download PDF

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Publication number
JP6483148B2
JP6483148B2 JP2016556997A JP2016556997A JP6483148B2 JP 6483148 B2 JP6483148 B2 JP 6483148B2 JP 2016556997 A JP2016556997 A JP 2016556997A JP 2016556997 A JP2016556997 A JP 2016556997A JP 6483148 B2 JP6483148 B2 JP 6483148B2
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Japanese (ja)
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JP2017511305A5 (https=
JP2017511305A (ja
Inventor
ジョン ジャヌス，
ジョン ジャヌス，
ジェイムズ コップ，
ジェイムズ コップ，
ケビン ピータース，
ケビン ピータース，
Original Assignee
エアーピオ セラピューティクス インコーポレイテッド
エアーピオ セラピューティクス インコーポレイテッド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2016556997A 2014-03-14 2015-03-13 ＨＰＴＰ−β阻害剤 Active JP6483148B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201461953680P 2014-03-14 2014-03-14
US61/953,680 2014-03-14
PCT/US2015/020425 WO2015138882A1 (en) 2014-03-14 2015-03-13 Hptp-beta inhibitors

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2018246712A Division JP6661744B2 (ja) 2014-03-14 2018-12-28 ＨＰＴＰ−β阻害剤

Publications (3)

Publication Number Publication Date
JP2017511305A JP2017511305A (ja) 2017-04-20
JP2017511305A5 JP2017511305A5 (https=) 2018-04-12
JP6483148B2 true JP6483148B2 (ja) 2019-03-13

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ID=54068203

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2016556997A Active JP6483148B2 (ja) 2014-03-14 2015-03-13 ＨＰＴＰ−β阻害剤
JP2018246712A Active JP6661744B2 (ja) 2014-03-14 2018-12-28 ＨＰＴＰ−β阻害剤
JP2019077696A Withdrawn JP2019108407A (ja) 2014-03-14 2019-04-16 ＨＰＴＰ−β阻害剤

Family Applications After (2)

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JP2018246712A Active JP6661744B2 (ja) 2014-03-14 2018-12-28 ＨＰＴＰ−β阻害剤
JP2019077696A Withdrawn JP2019108407A (ja) 2014-03-14 2019-04-16 ＨＰＴＰ−β阻害剤

Country Status (5)

Country Link
US (3) US9994560B2 (https=)
EP (1) EP3116503A4 (https=)
JP (3) JP6483148B2 (https=)
CN (1) CN106456614A (https=)
WO (1) WO2015138882A1 (https=)

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Also Published As

Publication number Publication date
US9994560B2 (en) 2018-06-12
EP3116503A1 (en) 2017-01-18
US20210130341A1 (en) 2021-05-06
US20180354937A1 (en) 2018-12-13
WO2015138882A1 (en) 2015-09-17
US20150259335A1 (en) 2015-09-17
JP6661744B2 (ja) 2020-03-11
CN106456614A (zh) 2017-02-22
JP2019108407A (ja) 2019-07-04
JP2019048894A (ja) 2019-03-28
US10858354B2 (en) 2020-12-08
EP3116503A4 (en) 2017-08-23
JP2017511305A (ja) 2017-04-20

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