JP6019015B2 - 6−シクロヘキシル−1−ヒドロキシ−4−メチル−2(1h)−ピリドンを使用する血液悪性疾患の治療方法 - Google Patents

6−シクロヘキシル−1−ヒドロキシ−4−メチル−2(1h)−ピリドンを使用する血液悪性疾患の治療方法 Download PDF

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JP6019015B2
JP6019015B2 JP2013513289A JP2013513289A JP6019015B2 JP 6019015 B2 JP6019015 B2 JP 6019015B2 JP 2013513289 A JP2013513289 A JP 2013513289A JP 2013513289 A JP2013513289 A JP 2013513289A JP 6019015 B2 JP6019015 B2 JP 6019015B2
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resistant
leukemia
pharmaceutical composition
drug
methyl
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JP2013528620A (ja
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メルクウリオ フランク
メルクウリオ フランク
ダブリュー.エイチ. チャン クイルエ
ダブリュー.エイチ. チャン クイルエ
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ビオトヘルイク, インコーポレイテッド
ビオトヘルイク, インコーポレイテッド
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2013513289A 2010-06-01 2011-06-01 6−シクロヘキシル−1−ヒドロキシ−4−メチル−2(1h)−ピリドンを使用する血液悪性疾患の治療方法 Expired - Fee Related JP6019015B2 (ja)

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US35043810P 2010-06-01 2010-06-01
US61/350,438 2010-06-01
PCT/US2011/038702 WO2011153199A1 (en) 2010-06-01 2011-06-01 Methods of treating hematologic malignancies using 6-cyclohexyl-1-hydroxy-4-methyl-2(1h)-pyridone

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JP2013528620A5 JP2013528620A5 (enExample) 2014-07-17
JP6019015B2 true JP6019015B2 (ja) 2016-11-02

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EP (1) EP2585063A1 (enExample)
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CN (1) CN103153309A (enExample)
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CA (1) CA2801003A1 (enExample)
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Publication number Priority date Publication date Assignee Title
JP5844354B2 (ja) 2010-06-01 2016-01-13 ビオトヘルイク, インコーポレイテッド ヒドロキシピリドン誘導体、その医薬組成物、及び増殖性疾患治療のためのその治療的使用
WO2015195474A1 (en) 2014-06-18 2015-12-23 Biotheryx, Inc. Hydroxypyridone derivatives, pharmaceutical compositions thereof, and their therapeutic use for treating inflammatory, neurodegenerative, or immune-mediated diseases
CN116077522B (zh) * 2023-03-09 2024-01-26 青岛市中心医院 一种用于治疗白血病的治疗制剂

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Publication number Publication date
US20130178503A1 (en) 2013-07-11
US20150342942A1 (en) 2015-12-03
MX2012013878A (es) 2013-06-28
MX342465B (es) 2016-09-30
CA2801003A1 (en) 2011-12-08
CN103153309A (zh) 2013-06-12
AU2011261501B2 (en) 2016-01-21
AU2011261501A1 (en) 2013-01-10
EP2585063A1 (en) 2013-05-01
JP2013528620A (ja) 2013-07-11
WO2011153199A1 (en) 2011-12-08

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