JP5918386B2 - キラル触媒およびそれらの塩の製造方法 - Google Patents

キラル触媒およびそれらの塩の製造方法 Download PDF

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JP5918386B2
JP5918386B2 JP2014543996A JP2014543996A JP5918386B2 JP 5918386 B2 JP5918386 B2 JP 5918386B2 JP 2014543996 A JP2014543996 A JP 2014543996A JP 2014543996 A JP2014543996 A JP 2014543996A JP 5918386 B2 JP5918386 B2 JP 5918386B2
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compound
formula
group
benzyl
iii
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Expired - Fee Related
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JP2014543996A
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Japanese (ja)
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JP2015505827A (ja
JP2015505827A5 (https=
Inventor
ポール ヘンシュケ ジュリアン
ポール ヘンシュケ ジュリアン
ピン−ユ ウー
ピン−ユ ウー
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サイノファーム タイワン，リミティド
サイノファーム タイワン，リミティド
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B53/00—Asymmetric syntheses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2014543996A 2011-11-30 2012-11-29 キラル触媒およびそれらの塩の製造方法 Expired - Fee Related JP5918386B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161565449P 2011-11-30 2011-11-30
US61/565,449 2011-11-30
PCT/IB2012/002910 WO2013080049A2 (en) 2011-11-30 2012-11-29 A process for the manufacture of chiral catalysts and their salts

Publications (3)

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JP2015505827A JP2015505827A (ja) 2015-02-26
JP2015505827A5 JP2015505827A5 (https=) 2016-03-31
JP5918386B2 true JP5918386B2 (ja) 2016-05-18

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ID=48536192

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JP2014543996A Expired - Fee Related JP5918386B2 (ja) 2011-11-30 2012-11-29 キラル触媒およびそれらの塩の製造方法

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Country Link
US (1) US8859765B2 (https=)
EP (1) EP2785688B1 (https=)
JP (1) JP5918386B2 (https=)
KR (1) KR101647415B1 (https=)
CN (1) CN103974932B (https=)
AU (1) AU2012346860B2 (https=)
BR (1) BR112014013285A8 (https=)
CA (1) CA2855751C (https=)
IL (1) IL232574A (https=)
TW (1) TWI483926B (https=)
WO (1) WO2013080049A2 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9553397B2 (en) 2014-09-18 2017-01-24 Lsis Co., Ltd. Electric connector and housing having a simple mounting structure

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6261111B2 (ja) * 2013-07-17 2018-01-17 国立大学法人名古屋大学 アレーンスルホンアミドの還元方法及びアレーンスルホン酸の製法
CN114436911B (zh) * 2022-03-17 2023-04-28 南京林业大学 一种樟脑磺酰苄胺类化合物的制备方法及其应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201136904A (en) * 2010-04-30 2011-11-01 Nat Univ Tsing Hua Method for preparing 2-morpholinoisobornane-10-thiol and intermediates formed therein
US8168835B2 (en) * 2010-05-26 2012-05-01 National Tsing Hua University Method for preparing propargylic alcohol catalyzed by 2-morpholinoisobornane-10-thiol

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9553397B2 (en) 2014-09-18 2017-01-24 Lsis Co., Ltd. Electric connector and housing having a simple mounting structure

Also Published As

Publication number Publication date
BR112014013285A2 (pt) 2017-06-13
CA2855751C (en) 2017-02-21
EP2785688A4 (en) 2015-07-15
WO2013080049A3 (en) 2013-08-08
TWI483926B (zh) 2015-05-11
WO2013080049A2 (en) 2013-06-06
EP2785688A2 (en) 2014-10-08
US20130150574A1 (en) 2013-06-13
IL232574A (en) 2017-02-28
JP2015505827A (ja) 2015-02-26
EP2785688B1 (en) 2017-09-13
BR112014013285A8 (pt) 2017-06-20
KR101647415B1 (ko) 2016-08-10
CA2855751A1 (en) 2013-06-06
KR20140097517A (ko) 2014-08-06
CN103974932A (zh) 2014-08-06
AU2012346860A1 (en) 2014-05-29
AU2012346860B2 (en) 2015-09-24
US8859765B2 (en) 2014-10-14
IL232574A0 (en) 2014-06-30
CN103974932B (zh) 2016-05-18
TW201335127A (zh) 2013-09-01

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