JP5791611B2 - ピリド［３，４−ｂ］インドールおよび使用方法 - Google Patents
ピリド［３，４−ｂ］インドールおよび使用方法 Download PDFInfo
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- JP5791611B2 JP5791611B2 JP2012531043A JP2012531043A JP5791611B2 JP 5791611 B2 JP5791611 B2 JP 5791611B2 JP 2012531043 A JP2012531043 A JP 2012531043A JP 2012531043 A JP2012531043 A JP 2012531043A JP 5791611 B2 JP5791611 B2 JP 5791611B2
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- General Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Medicinal Chemistry (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
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| US24514809P | 2009-09-23 | 2009-09-23 | |
| US61/245,148 | 2009-09-23 | ||
| PCT/US2010/050079 WO2011038162A1 (en) | 2009-09-23 | 2010-09-23 | Pyrido(3,4-b)indoles and methods of use |
Publications (3)
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| JP2013505946A JP2013505946A (ja) | 2013-02-21 |
| JP2013505946A5 JP2013505946A5 (https=) | 2013-11-07 |
| JP5791611B2 true JP5791611B2 (ja) | 2015-10-07 |
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| US (2) | US20130137705A1 (https=) |
| EP (1) | EP2480079A4 (https=) |
| JP (1) | JP5791611B2 (https=) |
| CN (1) | CN102711467A (https=) |
| AU (1) | AU2010298167B2 (https=) |
| BR (1) | BR112012006644A2 (https=) |
| CA (1) | CA2775129A1 (https=) |
| WO (1) | WO2011038162A1 (https=) |
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| RU2007139634A (ru) | 2007-10-25 | 2009-04-27 | Сергей Олегович Бачурин (RU) | Новые тиазол-, триазол- или оксадиазол-содержащие тетрациклические соединения |
| RU2544856C2 (ru) | 2008-01-25 | 2015-03-20 | Сергей Олегович Бачурин | НОВЫЕ ПРОИЗВОДНЫЕ 2,3,4,5-ТЕТРАГИДРО-1-ПИРИДО[4,3-b]ИНДОЛА И СПОСОБЫ ИХ ПРИМЕНЕНИЯ |
| TWI443098B (zh) | 2008-03-24 | 2014-07-01 | Medivation Technologies Inc | 吡啶并〔３，４－ｂ〕吲哚及使用方法 |
| CN102046625B (zh) | 2008-03-24 | 2015-04-08 | 梅迪维新技术公司 | 桥连杂环化合物及其使用方法 |
| AU2009308706C1 (en) | 2008-10-31 | 2016-01-21 | Medivation Technologies, Inc. | Pyrido (4,3-b) indoles containing rigid moieties |
| WO2010051503A1 (en) | 2008-10-31 | 2010-05-06 | Medivation Technologies, Inc. | Azepino [4, 5-b] indoles and methods of use |
| US9162980B2 (en) | 2009-01-09 | 2015-10-20 | Board Of Regents Of The University Of Texas System | Anti-depression compounds |
| US8362277B2 (en) | 2009-01-09 | 2013-01-29 | Board Of Regents Of The University Of Texas System | Pro-neurogenic compounds |
| EP2385829B1 (en) | 2009-01-09 | 2018-08-01 | Board of Regents of the University of Texas System | Pro-neurogenic compounds |
| US9095572B2 (en) | 2009-01-09 | 2015-08-04 | Board Of Regents Of The University Of Texas System | Pro-neurogenic compounds |
| US9962368B2 (en) | 2009-01-09 | 2018-05-08 | Board Of Regents Of The University Of Texas System | Pro-neurogenic compounds |
| JP5827943B2 (ja) | 2009-04-29 | 2015-12-02 | メディベイション テクノロジーズ， インコーポレイテッド | ピリド［４，３−ｂ］インドールおよびその使用方法 |
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- 2010-09-23 AU AU2010298167A patent/AU2010298167B2/en not_active Ceased
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- 2010-09-23 JP JP2012531043A patent/JP5791611B2/ja not_active Expired - Fee Related
- 2010-09-23 BR BR112012006644A patent/BR112012006644A2/pt not_active IP Right Cessation
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- 2010-09-23 CN CN2010800528027A patent/CN102711467A/zh active Pending
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| WO2011038162A1 (en) | 2011-03-31 |
| BR112012006644A2 (pt) | 2019-09-24 |
| CA2775129A1 (en) | 2011-03-31 |
| JP2013505946A (ja) | 2013-02-21 |
| CN102711467A (zh) | 2012-10-03 |
| US20130123277A1 (en) | 2013-05-16 |
| AU2010298167A1 (en) | 2012-04-12 |
| EP2480079A1 (en) | 2012-08-01 |
| EP2480079A4 (en) | 2015-04-08 |
| AU2010298167B2 (en) | 2015-12-24 |
| US20130137705A1 (en) | 2013-05-30 |
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