JP5775452B2 - 肝細胞増殖因子（分散因子）活性の低分子モジュレーターの組成物および方法 - Google Patents

肝細胞増殖因子（分散因子）活性の低分子モジュレーターの組成物および方法 Download PDF

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JP5775452B2
JP5775452B2 JP2011517424A JP2011517424A JP5775452B2 JP 5775452 B2 JP5775452 B2 JP 5775452B2 JP 2011517424 A JP2011517424 A JP 2011517424A JP 2011517424 A JP2011517424 A JP 2011517424A JP 5775452 B2 JP5775452 B2 JP 5775452B2
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alkyl
alkoxy
independently selected
hydroxy
optionally substituted
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JP2011527675A (ja
JP2011527675A5 (enExample
Inventor
ウェイチョン カイ，
ウェイチョン カイ，
プラカッシュ ナラヤン，
プラカッシュ ナラヤン，
ビジョイ パニッカー，
ビジョイ パニッカー，
デイビッド イー． スミス，
デイビッド イー． スミス，
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Elicio Therapeutics Inc
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Angion Biomedica Corp
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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JP2011517424A 2008-07-10 2009-07-09 肝細胞増殖因子（分散因子）活性の低分子モジュレーターの組成物および方法 Expired - Fee Related JP5775452B2 (ja)

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US13448508P 2008-07-10 2008-07-10
US61/134,485 2008-07-10
PCT/US2009/004014 WO2010005580A2 (en) 2008-07-10 2009-07-09 Methods and compositions of small molecule modulators of hepatocyte growth factor (scatter factor) activity

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JP2015012415A Division JP2015108002A (ja) 2008-07-10 2015-01-26 肝細胞増殖因子（分散因子）活性の低分子モジュレーターの組成物および方法

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JP2011527675A JP2011527675A (ja) 2011-11-04
JP2011527675A5 JP2011527675A5 (enExample) 2012-08-23
JP5775452B2 true JP5775452B2 (ja) 2015-09-09

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JP2015012415A Pending JP2015108002A (ja) 2008-07-10 2015-01-26 肝細胞増殖因子（分散因子）活性の低分子モジュレーターの組成物および方法

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US (4) US8772326B2 (enExample)
EP (1) EP2313093A4 (enExample)
JP (2) JP5775452B2 (enExample)
CN (1) CN102149379A (enExample)
CA (1) CA2767331A1 (enExample)
IL (1) IL210544A (enExample)
WO (1) WO2010005580A2 (enExample)

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US20130190376A1 (en) * 2010-10-05 2013-07-25 David E. Smith Methods of use of small molecule modulators of hepatocyte growth factor (scatter factor) activity
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PL2968297T3 (pl) 2013-03-15 2019-04-30 Verseon Corp Wielopodstawione związki aromatyczne jako inhibitory protezy serynowej
EP3194369A4 (en) 2014-09-17 2018-02-28 Verseon Corporation Pyrazolyl-substituted pyridone compounds as serine protease inhibitors
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CA3133803A1 (en) * 2019-04-11 2020-10-15 Angion Biomedica Corp. Solid forms of (e)-3-[2-(2-thienyl)vinyl]-1h-pyrazole
US20230000828A1 (en) * 2019-10-31 2023-01-05 Angion Biomedica Corp. Improving renal function after kidney transplantation
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US8772326B2 (en) 2014-07-08
CA2767331A1 (en) 2010-01-14
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US10899750B2 (en) 2021-01-26
US20110184038A1 (en) 2011-07-28
WO2010005580A2 (en) 2010-01-14
US20190375739A1 (en) 2019-12-12
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IL210544A (en) 2015-09-24

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